FI964114A - Uusia 1-(5-metaanisulfonamidoindolyyli-2-karbonyyli)-4-(3-(1-metyylietyyliamino)-2-pyridinyyli)piperatsiinin kiteisiä muotoja - Google Patents

Uusia 1-(5-metaanisulfonamidoindolyyli-2-karbonyyli)-4-(3-(1-metyylietyyliamino)-2-pyridinyyli)piperatsiinin kiteisiä muotoja Download PDF

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Publication number
FI964114A
FI964114A FI964114A FI964114A FI964114A FI 964114 A FI964114 A FI 964114A FI 964114 A FI964114 A FI 964114A FI 964114 A FI964114 A FI 964114A FI 964114 A FI964114 A FI 964114A
Authority
FI
Finland
Prior art keywords
methanesulfonamidoindolyl
methylethylamino
pyridinyl
carbonyl
piperazine
Prior art date
Application number
FI964114A
Other languages
English (en)
Swedish (sv)
Other versions
FI964114A0 (fi
FI111364B (fi
Inventor
Jeffrey L Havens
Donald P Smith
Michael S Bergren
Mark A Lyster
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of FI964114A publication Critical patent/FI964114A/fi
Publication of FI964114A0 publication Critical patent/FI964114A0/fi
Application granted granted Critical
Publication of FI111364B publication Critical patent/FI111364B/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Immunology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Virology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Indole Compounds (AREA)
FI964114A 1994-04-15 1996-10-14 Uusia 1-[5-metaanisulfonamidoindolyyli-2-karbonyyli]-4-[3-(1-metyylietyyliamino)-2-pyridinyyli]piperatsiinin kidemuotoja FI111364B (fi)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US22786094A 1994-04-15 1994-04-15
US22786094 1994-04-15
US31178094A 1994-09-23 1994-09-23
US31178094 1994-09-23
US9502166 1995-03-01
PCT/US1995/002166 WO1995028398A1 (en) 1994-04-15 1995-03-01 Novel crystal forms of 1-[5-methanesulfonamidoindolyl-2-carbonyl]-4-[3-(1-methylethylamino)-2-pyridinyl]piperazine

Publications (3)

Publication Number Publication Date
FI964114A true FI964114A (fi) 1996-10-14
FI964114A0 FI964114A0 (fi) 1996-10-14
FI111364B FI111364B (fi) 2003-07-15

Family

ID=26921831

Family Applications (1)

Application Number Title Priority Date Filing Date
FI964114A FI111364B (fi) 1994-04-15 1996-10-14 Uusia 1-[5-metaanisulfonamidoindolyyli-2-karbonyyli]-4-[3-(1-metyylietyyliamino)-2-pyridinyyli]piperatsiinin kidemuotoja

Country Status (26)

Country Link
US (1) US6452007B1 (fi)
EP (1) EP0755393B1 (fi)
JP (1) JP3817261B2 (fi)
KR (1) KR100364941B1 (fi)
CN (1) CN1147253A (fi)
AT (1) ATE207481T1 (fi)
AU (1) AU693939B2 (fi)
CA (1) CA2184598C (fi)
CZ (1) CZ287164B6 (fi)
DE (1) DE69523447T2 (fi)
DK (1) DK0755393T3 (fi)
ES (1) ES2164147T3 (fi)
FI (1) FI111364B (fi)
HU (1) HU226827B1 (fi)
IL (1) IL113162A (fi)
LV (1) LV12957B (fi)
MX (1) MX9604831A (fi)
MY (1) MY116830A (fi)
NO (1) NO310024B1 (fi)
NZ (1) NZ282211A (fi)
PL (1) PL180776B1 (fi)
PT (1) PT755393E (fi)
RU (1) RU2136677C1 (fi)
SK (1) SK282424B6 (fi)
TW (1) TW393478B (fi)
WO (1) WO1995028398A1 (fi)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69934582T2 (de) 1998-06-11 2007-10-04 Pharmacia & Upjohn Co. Llc, Kalamazoo Delavirdin tablettenformulierung
US6872811B1 (en) 1998-09-30 2005-03-29 Millennium Pharmaceuticals, Inc. HRPCa9 and HRPCa10 nucleic acids and polypeptides
DE102011113749A1 (de) * 2011-09-14 2013-03-14 Aicuris Gmbh & Co. Kg Sulfonsäuresalze Heterocyclylamid-substituiertr Imidazole

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3565924A (en) 1968-07-01 1971-02-23 Wisconsin Alumni Res Found 25-hydroxycholfcalciferol
US3833622A (en) 1969-03-17 1974-09-03 Upjohn Co Crystalline 25-hydroxycholecalciferol hydrate and structurally related compounds
GB1532682A (en) 1976-04-27 1978-11-22 Bristol Myers Co Process for the preparation of cephadroxil
IL63968A (en) 1980-10-01 1985-10-31 Glaxo Group Ltd Form 2 ranitidine hydrochloride,its preparation and pharmaceutical compositions containing it
US5563142A (en) * 1989-12-28 1996-10-08 The Upjohn Company Diaromatic substituted compounds as anti-HIV-1 agents
HUT61296A (en) * 1989-12-28 1992-12-28 Upjohn Co Process for producing substituted diaromatic compounds against aids and pharmaceutical compositions comprising same
US5599930A (en) * 1991-07-03 1997-02-04 The Upjohn Company Substituted indoles as anti-AIDS pharmaceuticals

Also Published As

Publication number Publication date
KR970702275A (ko) 1997-05-13
DK0755393T3 (da) 2001-12-17
CZ287164B6 (en) 2000-10-11
NO964386D0 (no) 1996-10-15
HUT76467A (en) 1997-09-29
JPH09512007A (ja) 1997-12-02
PL316688A1 (en) 1997-02-03
WO1995028398A1 (en) 1995-10-26
EP0755393B1 (en) 2001-10-24
DE69523447T2 (de) 2002-05-16
PT755393E (pt) 2002-04-29
MY116830A (en) 2004-04-30
EP0755393A1 (en) 1997-01-29
SK282424B6 (sk) 2002-01-07
NZ282211A (en) 1997-10-24
SK122996A3 (en) 1997-05-07
MX9604831A (es) 1998-05-31
IL113162A (en) 1999-04-11
JP3817261B2 (ja) 2006-09-06
AU3513695A (en) 1995-11-10
FI964114A0 (fi) 1996-10-14
NO964386L (no) 1996-10-15
KR100364941B1 (ko) 2003-02-19
US6452007B1 (en) 2002-09-17
AU693939B2 (en) 1998-07-09
CA2184598C (en) 2005-05-03
CZ294296A3 (en) 1997-01-15
LV12957B (en) 2003-04-20
RU2136677C1 (ru) 1999-09-10
PL180776B1 (pl) 2001-04-30
NO310024B1 (no) 2001-05-07
FI111364B (fi) 2003-07-15
TW393478B (en) 2000-06-11
CA2184598A1 (en) 1995-10-26
HU226827B1 (en) 2009-11-30
CN1147253A (zh) 1997-04-09
DE69523447D1 (de) 2001-11-29
IL113162A0 (en) 1995-06-29
ATE207481T1 (de) 2001-11-15
ES2164147T3 (es) 2002-02-16
HU9602857D0 (en) 1996-12-30

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MA Patent expired