SK281761B6 - Fenylindolová zlúčenina, farmaceutický prostriedok s jej obsahom a jej použitie - Google Patents

Fenylindolová zlúčenina, farmaceutický prostriedok s jej obsahom a jej použitie Download PDF

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Publication number
SK281761B6
SK281761B6 SK534-96A SK53496A SK281761B6 SK 281761 B6 SK281761 B6 SK 281761B6 SK 53496 A SK53496 A SK 53496A SK 281761 B6 SK281761 B6 SK 281761B6
Authority
SK
Slovakia
Prior art keywords
fluorophenyl
chloro
ethyl
piperidin
indol
Prior art date
Application number
SK534-96A
Other languages
English (en)
Slovak (sk)
Other versions
SK53496A3 (en
Inventor
Jens Perregaard
Ejner Knud Moltzen
Kim Andersen
Henrik Pedersen
Klaus Peter Bogeso
Andre Pernet
Barbara Bopp
Darcy Mulford
Kiyoshi Sakamoto
Original Assignee
H. Lundbeck A/S
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by H. Lundbeck A/S filed Critical H. Lundbeck A/S
Publication of SK53496A3 publication Critical patent/SK53496A3/sk
Publication of SK281761B6 publication Critical patent/SK281761B6/sk

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Sewing Machines And Sewing (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Polyurethanes Or Polyureas (AREA)
SK534-96A 1993-11-01 1994-10-28 Fenylindolová zlúčenina, farmaceutický prostriedok s jej obsahom a jej použitie SK281761B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DK931234A DK123493D0 (da) 1993-11-01 1993-11-01 Compounds
PCT/DK1994/000407 WO1995012591A1 (en) 1993-11-01 1994-10-28 Phenylindole compounds

Publications (2)

Publication Number Publication Date
SK53496A3 SK53496A3 (en) 1996-11-06
SK281761B6 true SK281761B6 (sk) 2001-07-10

Family

ID=8102507

Family Applications (1)

Application Number Title Priority Date Filing Date
SK534-96A SK281761B6 (sk) 1993-11-01 1994-10-28 Fenylindolová zlúčenina, farmaceutický prostriedok s jej obsahom a jej použitie

Country Status (27)

Country Link
US (1) US5703087A (ko)
EP (1) EP0726898B1 (ko)
JP (1) JP3898219B2 (ko)
KR (1) KR100350550B1 (ko)
CN (1) CN1134149A (ko)
AT (1) ATE198199T1 (ko)
AU (1) AU683700B2 (ko)
CA (1) CA2175498C (ko)
CZ (1) CZ291403B6 (ko)
DE (1) DE69426462T2 (ko)
DK (2) DK123493D0 (ko)
ES (1) ES2154303T3 (ko)
FI (1) FI116623B (ko)
GR (1) GR3035462T3 (ko)
HK (1) HK1013817A1 (ko)
HU (1) HUT76063A (ko)
IL (2) IL111394A (ko)
LV (1) LV12805B (ko)
NO (1) NO309038B1 (ko)
NZ (1) NZ275086A (ko)
PL (1) PL176391B1 (ko)
PT (1) PT726898E (ko)
RU (1) RU2156249C2 (ko)
SI (1) SI0726898T1 (ko)
SK (1) SK281761B6 (ko)
WO (1) WO1995012591A1 (ko)
ZA (1) ZA948589B (ko)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6489341B1 (en) * 1999-06-02 2002-12-03 Sepracor Inc. Methods for the treatment of neuroleptic and related disorders using sertindole derivatives
JP2003509509A (ja) * 1999-09-09 2003-03-11 ハー・ルンドベック・アクチエゼルスカベット 5−アミノアルキル及び5−アミノカルボニル置換されたインドール類
US20070212412A1 (en) * 2005-09-08 2007-09-13 H. Lundbeck A/S Stable solid formulation of sertindole
TW200821296A (en) * 2006-06-01 2008-05-16 Lundbeck & Co As H Use of sertindole for the preventive treatment of suicidal behaviour
PL2509961T3 (pl) 2009-12-11 2016-09-30 Pochodne imidazolidynodionu
US8933072B2 (en) 2010-06-16 2015-01-13 Vitae Pharmaceuticals, Inc. Substituted 5-,6- and 7-membered heterocycles, medicaments containing such compounds, and their use
US9346790B2 (en) 2010-12-06 2016-05-24 Autifony Therapeutics Limited Hydantoin derivatives useful as Kv3 inhibitors
JP6008953B2 (ja) * 2011-06-07 2016-10-19 アウトイフオンイ トヘラペウトイクス リミテッド Kv3阻害剤としてのヒダントイン誘導体
MX356813B (es) * 2011-12-06 2018-06-13 Autifony Therapeutics Ltd Derivados de hidantoina utiles como inhibidores de kv3.
EP2852588B8 (en) 2012-05-22 2018-01-10 Autifony Therapeutics Limited Hydantoin derivatives as kv3 inhibitors
EP2852589B1 (en) 2012-05-22 2021-04-28 Autifony Therapeutics Limited Triazoles as kv3 inhibitors

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE58370B1 (en) * 1985-04-10 1993-09-08 Lundbeck & Co As H Indole derivatives
GB8908085D0 (en) * 1989-04-11 1989-05-24 Lundbeck & Co As H New therapeutic use
DK152090D0 (da) * 1990-06-22 1990-06-22 Lundbaek A S H Piperidylsubstituerede indolderivater

Also Published As

Publication number Publication date
IL111395A (en) 1999-06-20
WO1995012591A1 (en) 1995-05-11
HU9601144D0 (en) 1996-07-29
LV12805A (en) 2002-03-20
NO309038B1 (no) 2000-12-04
KR100350550B1 (ko) 2002-12-12
PT726898E (pt) 2001-05-31
AU8057794A (en) 1995-05-23
DK0726898T3 (da) 2001-04-30
CZ124896A3 (en) 1996-09-11
US5703087A (en) 1997-12-30
FI961844A (fi) 1996-04-30
ES2154303T3 (es) 2001-04-01
FI116623B (fi) 2006-01-13
RU2156249C2 (ru) 2000-09-20
NO961746D0 (no) 1996-04-30
HUT76063A (en) 1997-06-30
NZ275086A (en) 1997-10-24
HK1013817A1 (en) 1999-09-10
SI0726898T1 (en) 2001-04-30
AU683700B2 (en) 1997-11-20
JPH09506083A (ja) 1997-06-17
ZA948589B (en) 1995-06-26
PL176391B1 (pl) 1999-05-31
GR3035462T3 (en) 2001-05-31
CN1134149A (zh) 1996-10-23
DK123493D0 (da) 1993-11-01
SK53496A3 (en) 1996-11-06
ATE198199T1 (de) 2001-01-15
EP0726898A1 (en) 1996-08-21
CA2175498C (en) 2005-07-26
IL111394A0 (en) 1994-12-29
JP3898219B2 (ja) 2007-03-28
KR960705814A (ko) 1996-11-08
PL314181A1 (en) 1996-08-19
NO961746L (no) 1996-06-28
IL111395A0 (en) 1994-12-29
DE69426462T2 (de) 2001-04-26
CA2175498A1 (en) 1995-05-11
IL111394A (en) 1998-08-16
FI961844A0 (fi) 1996-04-30
LV12805B (lv) 2002-05-20
CZ291403B6 (cs) 2003-03-12
EP0726898B1 (en) 2000-12-20
DE69426462D1 (de) 2001-01-25

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Legal Events

Date Code Title Description
MM4A Patent lapsed due to non-payment of maintenance fees

Effective date: 20091028