SK281079B6 - Deriváty benzazepín-, benzoxazepín- a benztiazepín-n-octovej kyseliny, spôsob ich prípravy a liečivo s ich obsahom - Google Patents

Deriváty benzazepín-, benzoxazepín- a benztiazepín-n-octovej kyseliny, spôsob ich prípravy a liečivo s ich obsahom Download PDF

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Publication number
SK281079B6
SK281079B6 SK354-96A SK35496A SK281079B6 SK 281079 B6 SK281079 B6 SK 281079B6 SK 35496 A SK35496 A SK 35496A SK 281079 B6 SK281079 B6 SK 281079B6
Authority
SK
Slovakia
Prior art keywords
formula
acid
group
compounds
solution
Prior art date
Application number
SK354-96A
Other languages
English (en)
Slovak (sk)
Other versions
SK35496A3 (en
Inventor
Harald Waldeck
Dagmar H�Ltje
Josef Messinger
Jochen Antel
Michael Wurl
Dirk Thorm�Hlen
Original Assignee
Solvay Pharmaceuticals Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Solvay Pharmaceuticals Gmbh filed Critical Solvay Pharmaceuticals Gmbh
Publication of SK35496A3 publication Critical patent/SK35496A3/sk
Publication of SK281079B6 publication Critical patent/SK281079B6/sk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D223/16—Benzazepines; Hydrogenated benzazepines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10—Antioedematous agents; Diuretics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
SK354-96A 1995-03-23 1996-03-15 Deriváty benzazepín-, benzoxazepín- a benztiazepín-n-octovej kyseliny, spôsob ich prípravy a liečivo s ich obsahom SK281079B6 (sk)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19510566A DE19510566A1 (de) 1995-03-23 1995-03-23 Benzazepin-, Benzoxazepin- und Benzothiazepin-N-essigsäurederivate sowie Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel

Publications (2)

Publication Number Publication Date
SK35496A3 SK35496A3 (en) 1997-02-05
SK281079B6 true SK281079B6 (sk) 2000-11-07

Family

ID=7757471

Family Applications (1)

Application Number Title Priority Date Filing Date
SK354-96A SK281079B6 (sk) 1995-03-23 1996-03-15 Deriváty benzazepín-, benzoxazepín- a benztiazepín-n-octovej kyseliny, spôsob ich prípravy a liečivo s ich obsahom

Country Status (25)

Country Link
US (1) US5677297A (cs)
EP (1) EP0733642B1 (cs)
JP (1) JP3942670B2 (cs)
KR (1) KR100482499B1 (cs)
CN (1) CN1059436C (cs)
AR (1) AR023289A1 (cs)
AT (1) ATE197801T1 (cs)
AU (1) AU701271B2 (cs)
CA (1) CA2172354C (cs)
CZ (1) CZ289245B6 (cs)
DE (2) DE19510566A1 (cs)
DK (1) DK0733642T3 (cs)
DZ (1) DZ2003A1 (cs)
ES (1) ES2152444T3 (cs)
GR (1) GR3035410T3 (cs)
HU (1) HU226064B1 (cs)
IL (1) IL117265A (cs)
NO (1) NO305904B1 (cs)
NZ (1) NZ286224A (cs)
PL (1) PL184336B1 (cs)
PT (1) PT733642E (cs)
RU (1) RU2159768C2 (cs)
SK (1) SK281079B6 (cs)
UA (1) UA44712C2 (cs)
ZA (1) ZA961243B (cs)

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* Cited by examiner, † Cited by third party
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FR2781483A1 (fr) * 1998-07-21 2000-01-28 Hoechst Marion Roussel Inc Derives de thioazepinone, procede de preparation et intermediaires de ce procede, application a titre de medicament et compositions pharmaceutiques les renfermant
DE19906310A1 (de) * 1999-02-16 2000-08-17 Solvay Pharm Gmbh Arzneimittel zur Behandlung von Bluthochdruck
DE19932555A1 (de) * 1999-07-13 2001-01-18 Solvay Pharm Gmbh Arzneimittel mit protektiver Wirkung gegen oxidativ-toxische und insbesondere gegen kardiotoxische Substanzen
US20020052370A1 (en) * 2000-07-06 2002-05-02 Barber Christopher Gordon Cyclopentyl-substituted glutaramide derivatives as inhibitors of neutral endopeptidase
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JP4824573B2 (ja) * 2003-11-18 2011-11-30 ゾルファイ ファーマスーティカルズ ゲゼルシャフト ミット ベシュレンクテル ハフツング 腎不全、腎疾患または腎障害、特に糖尿病患者におけるこれらの治療のための医薬組成物
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JP6591530B2 (ja) 2014-08-07 2019-10-16 イントラ−セルラー・セラピーズ・インコーポレイテッドＩｎｔｒａ−Ｃｅｌｌｕｌａｒ Ｔｈｅｒａｐｉｅｓ， Ｉｎｃ． 有機化合物
KR102345318B1 (ko) 2014-12-02 2021-12-31 현대모비스 주식회사 에이밍 보정 구조를 구비한 차량용 램프
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Also Published As

Publication number Publication date
IL117265A0 (en) 1996-06-18
ZA961243B (en) 1996-08-27
ATE197801T1 (de) 2000-12-15
IL117265A (en) 2000-07-16
JPH08269011A (ja) 1996-10-15
NO961181L (no) 1996-09-24
CN1147506A (zh) 1997-04-16
HUP9600680A3 (en) 1998-07-28
NO961181D0 (no) 1996-03-22
CN1059436C (zh) 2000-12-13
CZ86396A3 (en) 1996-10-16
AU701271B2 (en) 1999-01-21
AR023289A1 (es) 2002-09-04
CA2172354C (en) 2002-10-08
GR3035410T3 (en) 2001-05-31
PL313433A1 (en) 1996-09-30
AU4821096A (en) 1996-10-03
HUP9600680A2 (en) 1997-01-28
NO305904B1 (no) 1999-08-16
UA44712C2 (uk) 2002-03-15
DZ2003A1 (fr) 2002-07-20
HU226064B1 (en) 2008-04-28
CA2172354A1 (en) 1996-09-24
JP3942670B2 (ja) 2007-07-11
RU2159768C2 (ru) 2000-11-27
DE59606160D1 (de) 2001-01-04
CZ289245B6 (cs) 2001-12-12
PL184336B1 (pl) 2002-10-31
PT733642E (pt) 2001-03-30
KR100482499B1 (ko) 2006-08-23
SK35496A3 (en) 1997-02-05
DK0733642T3 (da) 2001-01-15
DE19510566A1 (de) 1996-09-26
EP0733642B1 (de) 2000-11-29
KR960034178A (ko) 1996-10-22
HU9600680D0 (en) 1996-05-28
NZ286224A (en) 1997-09-22
EP0733642A1 (de) 1996-09-25
US5677297A (en) 1997-10-14
ES2152444T3 (es) 2001-02-01

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