SK12722000A3 - Deriváty indolu a farmaceutické prostriedky, ktoré ich obsahujú - Google Patents

Deriváty indolu a farmaceutické prostriedky, ktoré ich obsahujú Download PDF

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Publication number
SK12722000A3
SK12722000A3 SK1272-2000A SK12722000A SK12722000A3 SK 12722000 A3 SK12722000 A3 SK 12722000A3 SK 12722000 A SK12722000 A SK 12722000A SK 12722000 A3 SK12722000 A3 SK 12722000A3
Authority
SK
Slovakia
Prior art keywords
carbon atom
ethyl
trifluoroethyl
pharmaceutically acceptable
configuration
Prior art date
Application number
SK1272-2000A
Other languages
English (en)
Slovak (sk)
Inventor
Makio Kitazawa
Toshiaki Yamaguchi
Hiroshi Miyata
Yukiyoshi Ajisawa
Original Assignee
Kissei Pharmaceutical Co., Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kissei Pharmaceutical Co., Ltd filed Critical Kissei Pharmaceutical Co., Ltd
Publication of SK12722000A3 publication Critical patent/SK12722000A3/sk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
SK1272-2000A 1998-02-27 1999-02-19 Deriváty indolu a farmaceutické prostriedky, ktoré ich obsahujú SK12722000A3 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP9057298 1998-02-27
PCT/JP1999/000732 WO1999043652A1 (fr) 1998-02-27 1999-02-19 Derives de l'indole et compositions medicales les renfermant

Publications (1)

Publication Number Publication Date
SK12722000A3 true SK12722000A3 (sk) 2001-03-12

Family

ID=14002150

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1272-2000A SK12722000A3 (sk) 1998-02-27 1999-02-19 Deriváty indolu a farmaceutické prostriedky, ktoré ich obsahujú

Country Status (24)

Country Link
US (1) US6310086B1 (da)
EP (1) EP1057813B1 (da)
JP (1) JP4342101B2 (da)
KR (1) KR100576207B1 (da)
CN (1) CN1157375C (da)
AR (1) AR014964A1 (da)
AT (1) ATE264841T1 (da)
AU (1) AU766088B2 (da)
BR (1) BR9908301A (da)
CA (1) CA2321547C (da)
DE (1) DE69916586T2 (da)
DK (1) DK1057813T3 (da)
ES (1) ES2220043T3 (da)
HK (1) HK1036974A1 (da)
HU (1) HUP0100680A3 (da)
NO (1) NO317257B1 (da)
NZ (1) NZ506497A (da)
PE (1) PE20000329A1 (da)
PL (1) PL342477A1 (da)
RU (1) RU2212404C2 (da)
SK (1) SK12722000A3 (da)
TW (2) TWI241293B (da)
WO (1) WO1999043652A1 (da)
ZA (1) ZA991590B (da)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SK12722000A3 (sk) 1998-02-27 2001-03-12 Kissei Pharmaceutical Co., Ltd Deriváty indolu a farmaceutické prostriedky, ktoré ich obsahujú
JP4634560B2 (ja) * 2000-01-14 2011-02-16 キッセイ薬品工業株式会社 光学活性なインドリン誘導体の製造方法およびその製造中間体
US6849655B2 (en) 2000-05-15 2005-02-01 Kissei Pharmaceutical Co., Ltd. Aqueous liquid formulations
WO2001087834A1 (fr) * 2000-05-16 2001-11-22 Takeda Chemical Industries, Ltd. Antagoniste de l'hormone de concentration de la melanine
JP4921646B2 (ja) * 2001-03-08 2012-04-25 キッセイ薬品工業株式会社 １−（３−ベンジルオキシプロピル）−５−（２−置換プロピル）インドリン誘導体およびその使用方法
CA2453476A1 (en) * 2001-07-13 2003-01-23 Kissei Pharmaceutical Co., Ltd. Medicinal compositions for opthalmic use
HU225505B1 (en) * 2002-09-09 2007-01-29 Richter Gedeon Vegyeszet Process for the preparation of r-(-)-tamsulosin hydrochloride and novel intermediates
AR050253A1 (es) 2004-06-24 2006-10-11 Smithkline Beecham Corp Compuesto derivado de indazol carboxamida, composicion que lo comprende y su uso para la preparacion de un medicamento
ATE508113T1 (de) * 2004-10-27 2011-05-15 Kissei Pharmaceutical Indolinverbindung und verfahren zu deren herstellung
EP1902731B1 (en) * 2005-06-21 2013-04-10 Kowa Company, Ltd. Preventive or remedy for glaucoma
US8063071B2 (en) 2007-10-31 2011-11-22 GlaxoSmithKline, LLC Chemical compounds
US8013007B2 (en) * 2007-02-26 2011-09-06 Concert Pharmaceuticals, Inc. Alpha 1A-adrenoceptor antagonists
US20100076010A1 (en) * 2007-02-26 2010-03-25 Concert Pharmaceuticals, Inc. Alpha 1a-adrenoceptor antagonists
AR065804A1 (es) 2007-03-23 2009-07-01 Smithkline Beecham Corp Compuesto de indol carboxamida, composicion farmaceutica que lo comprende y uso de dicho compuesto para preparar un medicamento
WO2010102968A1 (en) 2009-03-10 2010-09-16 Glaxo Group Limited Indole derivatives as ikk2 inhibitors
CN104211631A (zh) * 2013-05-30 2014-12-17 中国科学院上海药物研究所 一类吲哚类化合物、其制备方法、药物组合物及应用
WO2016042441A1 (en) 2014-09-18 2016-03-24 Mankind Research Centre A novel process for the preparation of considerably pure silodosin
ES2607639B1 (es) 2015-09-30 2018-02-28 Urquima, S.A Sal de ácido maleico de un intermedio de silodosina

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5021410A (en) * 1989-05-22 1991-06-04 Allergan, Inc. Combinations of selective alpha-adrenergic agonists and antagonists useful in lowering intraocular pressure
DE69319551T2 (de) * 1992-12-02 1998-10-29 Kissei Pharmaceutical Indolin Verbindungen zur Behandlung von Dysurien
JP3331047B2 (ja) * 1994-06-01 2002-10-07 キッセイ薬品工業株式会社 インドリン誘導体
JP3331048B2 (ja) 1994-06-01 2002-10-07 キッセイ薬品工業株式会社 インドール誘導体
JPH08143557A (ja) * 1994-11-24 1996-06-04 Toyobo Co Ltd 新規なフェニルピペラジン誘導体、その塩及びその溶媒和物
JPH0912563A (ja) * 1995-06-30 1997-01-14 Toyobo Co Ltd 新規ベンジルアルコ−ル誘導体、その製造方法およびその用途
AU9095998A (en) * 1997-09-22 1999-04-12 Kissei Pharmaceutical Co. Ltd. Remedies for dysuria resulting from prostatic hypertrophy
SK12722000A3 (sk) 1998-02-27 2001-03-12 Kissei Pharmaceutical Co., Ltd Deriváty indolu a farmaceutické prostriedky, ktoré ich obsahujú

Also Published As

Publication number Publication date
NO20004277D0 (no) 2000-08-25
CA2321547A1 (en) 1999-09-02
DK1057813T3 (da) 2004-08-16
NZ506497A (en) 2004-12-24
KR20010041403A (ko) 2001-05-15
ATE264841T1 (de) 2004-05-15
AU766088B2 (en) 2003-10-09
NO20004277L (no) 2000-09-11
EP1057813A4 (en) 2001-11-21
TWI241293B (en) 2005-10-11
KR100576207B1 (ko) 2006-05-03
CN1157375C (zh) 2004-07-14
HUP0100680A2 (hu) 2001-08-28
AU2547899A (en) 1999-09-15
US6310086B1 (en) 2001-10-30
CN1291976A (zh) 2001-04-18
NO317257B1 (no) 2004-09-27
HK1036974A1 (en) 2002-01-25
PE20000329A1 (es) 2000-04-13
DE69916586T2 (de) 2004-09-16
PL342477A1 (en) 2001-06-04
JP4342101B2 (ja) 2009-10-14
CA2321547C (en) 2010-01-19
EP1057813A1 (en) 2000-12-06
HUP0100680A3 (en) 2001-09-28
RU2212404C2 (ru) 2003-09-20
ES2220043T3 (es) 2004-12-01
ZA991590B (en) 1999-08-27
DE69916586D1 (de) 2004-05-27
WO1999043652A1 (fr) 1999-09-02
TWI249525B (en) 2006-02-21
BR9908301A (pt) 2000-10-31
AR014964A1 (es) 2001-04-11
EP1057813B1 (en) 2004-04-21

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