SI3412673T1 - Postopek za pripravo pirolo(3,2-d)pirimidinske spojine in njenih intermediatov - Google Patents

Postopek za pripravo pirolo(3,2-d)pirimidinske spojine in njenih intermediatov

Info

Publication number
SI3412673T1
SI3412673T1 SI201730605T SI201730605T SI3412673T1 SI 3412673 T1 SI3412673 T1 SI 3412673T1 SI 201730605 T SI201730605 T SI 201730605T SI 201730605 T SI201730605 T SI 201730605T SI 3412673 T1 SI3412673 T1 SI 3412673T1
Authority
SI
Slovenia
Prior art keywords
intermediates
pyrimidine compound
preparing pyrrolo
pyrrolo
preparing
Prior art date
Application number
SI201730605T
Other languages
English (en)
Slovenian (sl)
Inventor
Zhaozhong Ding
Fei Sun
Yinghu Hu
Yilong Zhou
Rui Zhao
Ling Yang
Original Assignee
Chia Tai Tianqing Pharmaceutical Group Co., Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chia Tai Tianqing Pharmaceutical Group Co., Ltd filed Critical Chia Tai Tianqing Pharmaceutical Group Co., Ltd
Publication of SI3412673T1 publication Critical patent/SI3412673T1/sl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
SI201730605T 2016-02-05 2017-02-04 Postopek za pripravo pirolo(3,2-d)pirimidinske spojine in njenih intermediatov SI3412673T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN201610082028.3A CN107043378A (zh) 2016-02-05 2016-02-05 一种吡咯并[3,2-d]嘧啶类化合物的制备方法及其中间体
PCT/CN2017/072893 WO2017133686A1 (zh) 2016-02-05 2017-02-04 一种吡咯并[3,2-d]嘧啶类化合物的制备方法及其中间体
EP17747006.9A EP3412673B1 (en) 2016-02-05 2017-02-04 Method for preparing pyrrolo[3,2-d]pyrimidine compound, and intermediates thereof

Publications (1)

Publication Number Publication Date
SI3412673T1 true SI3412673T1 (sl) 2021-04-30

Family

ID=59500148

Family Applications (1)

Application Number Title Priority Date Filing Date
SI201730605T SI3412673T1 (sl) 2016-02-05 2017-02-04 Postopek za pripravo pirolo(3,2-d)pirimidinske spojine in njenih intermediatov

Country Status (28)

Country Link
US (2) US10654856B2 (cg-RX-API-DMAC7.html)
EP (1) EP3412673B1 (cg-RX-API-DMAC7.html)
JP (1) JP6877449B2 (cg-RX-API-DMAC7.html)
KR (1) KR102371500B1 (cg-RX-API-DMAC7.html)
CN (2) CN107043378A (cg-RX-API-DMAC7.html)
AR (1) AR107549A1 (cg-RX-API-DMAC7.html)
AU (1) AU2017214134B2 (cg-RX-API-DMAC7.html)
BR (1) BR112018015879B1 (cg-RX-API-DMAC7.html)
CA (1) CA3013520C (cg-RX-API-DMAC7.html)
CL (1) CL2018002094A1 (cg-RX-API-DMAC7.html)
DK (1) DK3412673T3 (cg-RX-API-DMAC7.html)
EA (1) EA034581B1 (cg-RX-API-DMAC7.html)
ES (1) ES2852323T3 (cg-RX-API-DMAC7.html)
HR (1) HRP20210103T1 (cg-RX-API-DMAC7.html)
HU (1) HUE053455T2 (cg-RX-API-DMAC7.html)
IL (1) IL260999B (cg-RX-API-DMAC7.html)
LT (1) LT3412673T (cg-RX-API-DMAC7.html)
MX (1) MX374298B (cg-RX-API-DMAC7.html)
MY (1) MY190551A (cg-RX-API-DMAC7.html)
NZ (1) NZ744885A (cg-RX-API-DMAC7.html)
PH (1) PH12018501642A1 (cg-RX-API-DMAC7.html)
PL (1) PL3412673T3 (cg-RX-API-DMAC7.html)
PT (1) PT3412673T (cg-RX-API-DMAC7.html)
SG (1) SG11201806685VA (cg-RX-API-DMAC7.html)
SI (1) SI3412673T1 (cg-RX-API-DMAC7.html)
TW (1) TW201728590A (cg-RX-API-DMAC7.html)
UA (1) UA124100C2 (cg-RX-API-DMAC7.html)
WO (1) WO2017133686A1 (cg-RX-API-DMAC7.html)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN107043380A (zh) * 2016-02-05 2017-08-15 正大天晴药业集团股份有限公司 一种tlr7激动剂的马来酸盐、其晶型c、晶型d、晶型e、制备方法和用途
MA44007A (fr) 2016-02-05 2018-12-19 Denali Therapeutics Inc Inhibiteurs du récepteur interagissant avec protéine kinase 1
WO2020162705A1 (ko) 2019-02-08 2020-08-13 성균관대학교산학협력단 톨-유사 수용체 7 또는 8 작용자와 콜레스테롤의 결합체 및 그 용도
US20230100429A1 (en) 2020-03-02 2023-03-30 Progeneer Inc. Live-pathogen-mimetic nanoparticles based on pathogen cell wall skeleton, and production method thereof
JP7690222B2 (ja) 2020-08-04 2025-06-10 プロジェニア インコーポレイテッド 動力学的制御が可能なアジュバントを含むmRNAワクチン
JP2023536954A (ja) 2020-08-04 2023-08-30 プロジェニア インコーポレイテッド 活性化部位が一時的に不活性化したトール様受容体7または8作用薬と機能性薬物の結合体およびその用途
WO2022031011A1 (ko) 2020-08-04 2022-02-10 성균관대학교산학협력단 동력학적으로 작용하는 아주번트 앙상블
IL314082A (en) 2022-01-12 2024-09-01 Denali Therapeutics Inc Crystal forms of (S)-5-benzyl-N-(5-methyl-4-oxo-2,3,4,5-tetrahydropyrido[3,2-b][1,4]oxazapin-3-yl)- H4- 1,2,4-triazole-3-carboxamide

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009082247A1 (en) * 2007-12-21 2009-07-02 Industrial Research Limited Process for preparing immucillins having a methylene link
EA021377B9 (ru) 2008-12-09 2015-09-30 Джилид Сайэнс, Инк. Модуляторы толл-подобных рецепторов
EP2906563B1 (en) * 2012-10-10 2018-02-28 Janssen Sciences Ireland UC Pyrrolo[3,2-d]pyrimidine derivatives for the treatment of viral infections and other diseases
AU2013348217B2 (en) * 2012-11-20 2016-10-06 Glaxosmithkline Llc Novel compounds
SG11201503282RA (en) * 2012-11-20 2015-06-29 Glaxosmithkline Llc Novel compounds
MX362341B (es) * 2014-05-01 2019-01-11 Novartis Ag Compuestos y composiciones como agonistas del receptor tipo toll 7.
MX386981B (es) 2014-08-15 2025-03-19 Chia Tai Tianqing Pharmaceutical Group Co Ltd Compuestos de pirrolopirimidina usados como agonistas del receptor de tipo toll 7 (tlr7).
CN105367576A (zh) 2014-08-15 2016-03-02 正大天晴药业集团股份有限公司 作为tlr7激动剂的吡咯并嘧啶化合物
ES2833927T3 (es) 2015-11-05 2021-06-16 Chai Tai Tianqing Pharmaceutical Group Co Ltd Compuesto de 7-(tiazol-5-il)pirrolopirimidina como agonista de TLR7
CN107043379A (zh) * 2016-02-05 2017-08-15 正大天晴药业集团股份有限公司 一种tlr7激动剂的晶型a、其制备方法和医药用途
CN107043377A (zh) * 2016-02-05 2017-08-15 正大天晴药业集团股份有限公司 一种tlr7激动剂的三氟乙酸盐、晶型b及其制备方法、药物组合物和用途
CN107043380A (zh) * 2016-02-05 2017-08-15 正大天晴药业集团股份有限公司 一种tlr7激动剂的马来酸盐、其晶型c、晶型d、晶型e、制备方法和用途

Also Published As

Publication number Publication date
HK1259183A1 (zh) 2019-11-29
MY190551A (en) 2022-04-27
KR20180104724A (ko) 2018-09-21
BR112018015879A2 (pt) 2018-12-26
EA034581B1 (ru) 2020-02-21
CN107043378A (zh) 2017-08-15
LT3412673T (lt) 2021-03-10
US20190040072A1 (en) 2019-02-07
WO2017133686A1 (zh) 2017-08-10
US10654856B2 (en) 2020-05-19
EA201891769A1 (ru) 2019-04-30
UA124100C2 (uk) 2021-07-21
HUE053455T2 (hu) 2021-06-28
CA3013520A1 (en) 2017-08-10
ES2852323T3 (es) 2021-09-13
AU2017214134B2 (en) 2020-08-27
AU2017214134A1 (en) 2018-08-23
CN108602832A (zh) 2018-09-28
PH12018501642B1 (en) 2019-06-03
KR102371500B1 (ko) 2022-03-07
CA3013520C (en) 2022-07-19
SG11201806685VA (en) 2018-09-27
NZ744885A (en) 2022-07-01
JP6877449B2 (ja) 2021-05-26
TW201728590A (zh) 2017-08-16
CN108602832B (zh) 2020-10-09
MX2018009502A (es) 2018-12-11
IL260999B (en) 2021-02-28
MX374298B (es) 2025-03-06
PH12018501642A1 (en) 2019-06-03
DK3412673T3 (da) 2021-01-18
PT3412673T (pt) 2021-02-15
JP2019505531A (ja) 2019-02-28
CL2018002094A1 (es) 2018-12-07
BR112018015879B1 (pt) 2024-02-15
PL3412673T3 (pl) 2021-07-26
EP3412673B1 (en) 2020-11-25
EP3412673A4 (en) 2019-07-03
AR107549A1 (es) 2018-05-09
HRP20210103T1 (hr) 2021-03-05
EP3412673A1 (en) 2018-12-12
US20200239484A1 (en) 2020-07-30

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