SI2070536T1 - Farmacevtska sestava vsebujoča derivat fenilamidina in postopek z uporabo farmacevtske sestave vkombinaciji s protiglivičnim sredstvom - Google Patents

Farmacevtska sestava vsebujoča derivat fenilamidina in postopek z uporabo farmacevtske sestave vkombinaciji s protiglivičnim sredstvom

Info

Publication number
SI2070536T1
SI2070536T1 SI200730827T SI200730827T SI2070536T1 SI 2070536 T1 SI2070536 T1 SI 2070536T1 SI 200730827 T SI200730827 T SI 200730827T SI 200730827 T SI200730827 T SI 200730827T SI 2070536 T1 SI2070536 T1 SI 2070536T1
Authority
SI
Slovenia
Prior art keywords
pharmaceutical composition
antifungal agents
combination
phenylamidine derivative
agents
Prior art date
Application number
SI200730827T
Other languages
English (en)
Inventor
Hiroshi Nishikawa
Original Assignee
Toyama Chemical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Toyama Chemical Co Ltd filed Critical Toyama Chemical Co Ltd
Publication of SI2070536T1 publication Critical patent/SI2070536T1/sl

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4465Non condensed piperidines, e.g. piperocaine only substituted in position 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41961,2,4-Triazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4453Non condensed piperidines, e.g. piperocaine only substituted in position 1, e.g. propipocaine, diperodon
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965Non-condensed pyrazines
    • A61K31/497Non-condensed pyrazines containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
SI200730827T 2006-10-06 2007-10-03 Farmacevtska sestava vsebujoča derivat fenilamidina in postopek z uporabo farmacevtske sestave vkombinaciji s protiglivičnim sredstvom SI2070536T1 (sl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2006274709 2006-10-06

Publications (1)

Publication Number Publication Date
SI2070536T1 true SI2070536T1 (sl) 2012-03-30

Family

ID=39282771

Family Applications (1)

Application Number Title Priority Date Filing Date
SI200730827T SI2070536T1 (sl) 2006-10-06 2007-10-03 Farmacevtska sestava vsebujoča derivat fenilamidina in postopek z uporabo farmacevtske sestave vkombinaciji s protiglivičnim sredstvom

Country Status (21)

Country Link
US (1) US8173157B2 (sl)
EP (1) EP2070536B1 (sl)
JP (1) JP5132569B2 (sl)
KR (1) KR101409258B1 (sl)
CN (1) CN101522195B (sl)
AT (1) ATE538789T1 (sl)
AU (1) AU2007305626B2 (sl)
BR (1) BRPI0719157A2 (sl)
CA (1) CA2664915C (sl)
CY (1) CY1112617T1 (sl)
DK (1) DK2070536T3 (sl)
ES (1) ES2376130T3 (sl)
MX (1) MX2009003533A (sl)
NO (1) NO20091101L (sl)
NZ (1) NZ575714A (sl)
PL (1) PL2070536T3 (sl)
PT (1) PT2070536E (sl)
RU (1) RU2429843C2 (sl)
SI (1) SI2070536T1 (sl)
WO (1) WO2008044562A1 (sl)
ZA (1) ZA200902053B (sl)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI385169B (zh) 2005-10-31 2013-02-11 Eisai R&D Man Co Ltd 經雜環取代之吡啶衍生物及含有彼之抗真菌劑
TW200841879A (en) 2007-04-27 2008-11-01 Eisai R&D Man Co Ltd Pyridine derivatives substituted by heterocyclic ring and phosphonoamino group, and anti-fungal agent containing same
TWI395735B (zh) 2007-07-04 2013-05-11 Toyama Chemical Co Ltd 4-{3-〔4-(3-{4-〔胺基(丁氧基羰基亞胺基)甲基〕苯氧基}丙基)-1-哌啶基〕丙氧基}-n’-(丁氧基羰基)苄脒之新穎結晶
US20130288956A1 (en) 2010-11-05 2013-10-31 Eisai R&D Management Co., Ltd. Combined pharmaceutical composition as antifungal agent
JP6181044B2 (ja) 2012-04-20 2017-08-16 エーザイ・アール・アンド・ディー・マネジメント株式会社 カプセル剤
WO2018081513A1 (en) 2016-10-31 2018-05-03 Biocryst Pharmaceuticals, Inc. Prodrugs of kallikrein inhibitors

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4782059A (en) * 1986-09-29 1988-11-01 Merck & Co., Inc. Method of controlling mycotic infections and compositions therefor
JPH03288051A (ja) 1990-03-30 1991-12-18 Mazda Motor Corp カムシャフトおよびその製造方法
GB9509631D0 (en) * 1995-05-12 1995-07-05 Sandoz Ltd Antifungal combination
WO1998010782A1 (en) * 1996-09-12 1998-03-19 Merck & Co., Inc. Antifungal combination therapy
AUPQ066399A0 (en) * 1999-05-31 1999-06-24 Fujisawa Pharmaceutical Co., Ltd. Antifungal combination use
KR100915979B1 (ko) * 2002-03-06 2009-09-10 토야마 케미칼 컴퍼니 리미티드 신규의 아릴아미딘 유도체 또는 그 염
WO2005026323A2 (en) * 2003-09-05 2005-03-24 Merck & Co., Inc. Stationary phases and a purification process using the stationary phases
JP4937506B2 (ja) * 2003-09-05 2012-05-23 富山化学工業株式会社 新規なアリールアミジン誘導体またはその塩
CA2572161C (en) * 2004-06-30 2012-10-02 Toyama Chemical Co., Ltd. Novel arylamidine derivative, salt thereof, and antifungal containing these
CN1596897A (zh) * 2004-07-26 2005-03-23 范敏华 一种伊曲康唑注射剂及其制备方法
JP5021308B2 (ja) * 2004-07-28 2012-09-05 富山化学工業株式会社 新規なアリールアミジン誘導体およびその塩ならびにそれらを含有する抗真菌剤
ZA200708530B (en) 2005-04-07 2009-04-29 Toyama Chemical Co Ltd Pharmaceutical composition and method using antifungal agent in combination
JP5314284B2 (ja) 2005-11-09 2013-10-16 富山化学工業株式会社 4−(3−(4−(3−(4−シアノフェノキシ)プロピル)−1−ピペリジニル)プロポキシ)ベンゾニトリルの製造法およびその中間体
DK1967190T3 (da) * 2005-12-29 2010-11-22 Toyama Chemical Co Ltd Nyt arylamidin-derivat, salt deraf og svampebekæmpelsesmiddel indeholdende dette

Also Published As

Publication number Publication date
RU2009117207A (ru) 2010-11-20
PT2070536E (pt) 2012-03-06
ZA200902053B (en) 2010-07-28
EP2070536B1 (en) 2011-12-28
CA2664915A1 (en) 2008-04-17
BRPI0719157A2 (pt) 2014-02-04
AU2007305626B2 (en) 2013-01-10
DK2070536T3 (da) 2012-04-10
ATE538789T1 (de) 2012-01-15
JP5132569B2 (ja) 2013-01-30
AU2007305626A1 (en) 2008-04-17
PL2070536T3 (pl) 2012-06-29
RU2429843C2 (ru) 2011-09-27
EP2070536A1 (en) 2009-06-17
EP2070536A4 (en) 2010-02-10
ES2376130T3 (es) 2012-03-09
US8173157B2 (en) 2012-05-08
JPWO2008044562A1 (ja) 2010-02-12
CN101522195B (zh) 2012-01-18
NO20091101L (no) 2009-04-27
KR101409258B1 (ko) 2014-06-18
WO2008044562A1 (fr) 2008-04-17
NZ575714A (en) 2011-05-27
US20100098750A1 (en) 2010-04-22
KR20090069317A (ko) 2009-06-30
CN101522195A (zh) 2009-09-02
CA2664915C (en) 2014-01-07
CY1112617T1 (el) 2016-02-10
MX2009003533A (es) 2009-07-17

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