SI1963280T1 - 2-feniletilamino derivati kot modulatorji kalcijevih in/ali natrijevih kanalčkov - Google Patents
2-feniletilamino derivati kot modulatorji kalcijevih in/ali natrijevih kanalčkovInfo
- Publication number
- SI1963280T1 SI1963280T1 SI200632017T SI200632017T SI1963280T1 SI 1963280 T1 SI1963280 T1 SI 1963280T1 SI 200632017 T SI200632017 T SI 200632017T SI 200632017 T SI200632017 T SI 200632017T SI 1963280 T1 SI1963280 T1 SI 1963280T1
- Authority
- SI
- Slovenia
- Prior art keywords
- calcium
- sodium channel
- channel modulators
- phenylethylamino derivatives
- phenylethylamino
- Prior art date
Links
- OYPRJOBELJOOCE-UHFFFAOYSA-N Calcium Chemical compound [Ca] OYPRJOBELJOOCE-UHFFFAOYSA-N 0.000 title 1
- 108090000312 Calcium Channels Proteins 0.000 title 1
- 102000003922 Calcium Channels Human genes 0.000 title 1
- 108010052164 Sodium Channels Proteins 0.000 title 1
- 102000018674 Sodium Channels Human genes 0.000 title 1
- 239000011575 calcium Substances 0.000 title 1
- 229910052791 calcium Inorganic materials 0.000 title 1
- 125000003395 phenylethylamino group Chemical group [H]N(*)C([H])([H])C([H])([H])C1=C([H])C([H])=C([H])C([H])=C1[H] 0.000 title 1
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- C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
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- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
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- C07C2601/02—Systems containing only non-condensed rings with a three-membered ring
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Epidemiology (AREA)
- Endocrinology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Gastroenterology & Hepatology (AREA)
- Rheumatology (AREA)
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- Hospice & Palliative Care (AREA)
- Vascular Medicine (AREA)
- Reproductive Health (AREA)
- Diabetes (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP05028147 | 2005-12-22 | ||
| PCT/EP2006/011443 WO2007071311A1 (en) | 2005-12-22 | 2006-11-29 | 2 -phenylethylamino derivatives as calcium and/or sodium channel modulators |
| EP06829177.2A EP1963280B1 (en) | 2005-12-22 | 2006-11-29 | 2-phenylethylamino derivatives as calcium and/or sodium channel modulators |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SI1963280T1 true SI1963280T1 (sl) | 2016-02-29 |
Family
ID=36178203
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SI200632017T SI1963280T1 (sl) | 2005-12-22 | 2006-11-29 | 2-feniletilamino derivati kot modulatorji kalcijevih in/ali natrijevih kanalčkov |
Country Status (25)
| Country | Link |
|---|---|
| US (3) | US7855227B2 (enExample) |
| EP (1) | EP1963280B1 (enExample) |
| JP (1) | JP5271087B2 (enExample) |
| KR (1) | KR101380137B1 (enExample) |
| CN (1) | CN101309909B (enExample) |
| AR (1) | AR058720A1 (enExample) |
| AU (1) | AU2006329040C1 (enExample) |
| BR (1) | BRPI0620239B8 (enExample) |
| CA (1) | CA2629065C (enExample) |
| CY (1) | CY1117094T1 (enExample) |
| DK (1) | DK1963280T3 (enExample) |
| ES (1) | ES2556937T3 (enExample) |
| HR (1) | HRP20160005T1 (enExample) |
| HU (1) | HUE028329T2 (enExample) |
| IL (1) | IL191255A (enExample) |
| IN (1) | IN266803B (enExample) |
| NO (1) | NO341296B1 (enExample) |
| NZ (1) | NZ567540A (enExample) |
| PL (1) | PL1963280T3 (enExample) |
| PT (1) | PT1963280E (enExample) |
| RS (1) | RS54522B1 (enExample) |
| RU (1) | RU2397160C9 (enExample) |
| SI (1) | SI1963280T1 (enExample) |
| TW (1) | TWI379828B (enExample) |
| WO (1) | WO2007071311A1 (enExample) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
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| IL173886A (en) * | 2003-08-25 | 2012-09-24 | Newron Pharm Spa | Alpha-aminoamide derivatives for treating inflammatory disorders |
| RU2397160C9 (ru) * | 2005-12-22 | 2012-10-27 | НЬЮРОН ФАРМАСЬЮТИКАЛЗ С.п.А. | 2-фенилэтиламинопроизводные в качестве модуляторов кальциевых и/или натриевых каналов |
| DK2155663T3 (en) * | 2007-06-15 | 2018-01-22 | Newron Pharm Spa | SUBSTITUTED 2- [2- (PHENYL) ETHYLAMINO] ALKANAMIDE DERIVATIVES AND THEIR USE AS SODIUM AND / OR CALCIUM CHANNEL MODULATORS |
| CA2707646C (en) | 2007-12-19 | 2016-09-13 | Newron Pharmaceuticals S.P.A. | Alpha-aminoamide derivatives useful in the treatment of psychiatric disorders |
| HUE030031T2 (en) | 2011-06-27 | 2017-04-28 | Newron Pharm Spa | Fluorinated arylalkylaminocarboxamide derivatives |
| UA109220C2 (uk) | 2011-10-26 | 2015-07-27 | Пфайзер Лімітед | Похідні (4-фенілімідазол-2-іл)етиламіну як модулятори натрієвих каналів |
| CN103804341B (zh) * | 2012-11-13 | 2018-04-10 | 中国人民解放军军事医学科学院毒物药物研究所 | 酰胺衍生物及其医药用途 |
| CN104761531B (zh) * | 2014-01-03 | 2017-12-01 | 中国人民解放军军事医学科学院毒物药物研究所 | 镇痛活性化合物及其医药用途 |
| CA2963371C (en) | 2014-10-02 | 2020-06-02 | Korea Institute Of Science And Technology | Alpha-aminoamide derivative compound and pharmaceutical composition containing the same |
| US10034861B2 (en) | 2016-07-04 | 2018-07-31 | H. Lundbeck A/S | 1H-pyrazolo[4,3-b]pyridines as PDE1 inhibitors |
| HRP20211784T1 (hr) | 2017-12-14 | 2022-02-18 | H. Lundbeck A/S | Kombinacijski tretmani koji se sastoje od primjene 1h-pirazolo[4,3-b]piridina |
| AR113926A1 (es) | 2017-12-14 | 2020-07-01 | H Lundbeck As | Derivados de 1h-pirazolo[4,3-b]piridinas |
| EP3728250A1 (en) | 2017-12-20 | 2020-10-28 | H. Lundbeck A/S | PYRAZOLO[3,4-beta]PYRIDINES AND IMIDAZO[1,5-beta]PYRIDAZINES AS PDE1 INHIBITORS |
| EP3725768A1 (en) * | 2019-04-17 | 2020-10-21 | Newron Pharmaceuticals S.p.A. | Process for the production of substituted 2-[2-(phenyl) ethylamino]alkaneamide derivatives |
| EP3725769A1 (en) * | 2019-04-17 | 2020-10-21 | Newron Pharmaceuticals S.p.A. | Process for the production of substituted 2-[2-(phenyl) ethylamino]alkaneamide derivatives |
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| ATE165977T1 (de) * | 1991-12-30 | 1998-05-15 | Neurex Corp | Methoden zur erzeugung von analgesie und zur verstärkung von opiat-analgesie |
| FR2696934B1 (fr) | 1992-10-20 | 1995-06-02 | Conservatoire Nal Arts Metiers | Dérivés de stéroïdes naturels 3B hydroxyles ayant des propriétés de déclenchement et de stimulation de l'immunité, composition les contenant et procédé pour les obtenir. |
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| AU8668598A (en) * | 1997-08-20 | 1999-03-08 | University Of Oklahoma, The | Gaba analogs to prevent and treat gastrointestinal damage |
| DE19740110A1 (de) | 1997-09-12 | 1999-03-18 | Boehringer Ingelheim Pharma | Substituierte 1,2,3,4,5,6-Hexahydro-2,6-methano-3-benzazocin-10-ole, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
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| RU2397160C9 (ru) * | 2005-12-22 | 2012-10-27 | НЬЮРОН ФАРМАСЬЮТИКАЛЗ С.п.А. | 2-фенилэтиламинопроизводные в качестве модуляторов кальциевых и/или натриевых каналов |
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2006
- 2006-11-29 RU RU2008130045/04A patent/RU2397160C9/ru active
- 2006-11-29 DK DK06829177.2T patent/DK1963280T3/en active
- 2006-11-29 EP EP06829177.2A patent/EP1963280B1/en active Active
- 2006-11-29 HU HUE06829177A patent/HUE028329T2/en unknown
- 2006-11-29 CA CA2629065A patent/CA2629065C/en active Active
- 2006-11-29 US US12/158,491 patent/US7855227B2/en active Active
- 2006-11-29 ES ES06829177.2T patent/ES2556937T3/es active Active
- 2006-11-29 JP JP2008546171A patent/JP5271087B2/ja active Active
- 2006-11-29 PL PL06829177T patent/PL1963280T3/pl unknown
- 2006-11-29 KR KR1020087018027A patent/KR101380137B1/ko active Active
- 2006-11-29 WO PCT/EP2006/011443 patent/WO2007071311A1/en not_active Ceased
- 2006-11-29 CN CN2006800424801A patent/CN101309909B/zh active Active
- 2006-11-29 IN IN3820CHN2008 patent/IN266803B/en unknown
- 2006-11-29 PT PT68291772T patent/PT1963280E/pt unknown
- 2006-11-29 BR BRPI0620239A patent/BRPI0620239B8/pt active IP Right Grant
- 2006-11-29 HR HRP20160005TT patent/HRP20160005T1/hr unknown
- 2006-11-29 RS RS20160004A patent/RS54522B1/sr unknown
- 2006-11-29 SI SI200632017T patent/SI1963280T1/sl unknown
- 2006-11-29 AU AU2006329040A patent/AU2006329040C1/en active Active
- 2006-11-29 NZ NZ567540A patent/NZ567540A/en unknown
- 2006-12-18 TW TW095147414A patent/TWI379828B/zh active
- 2006-12-21 AR ARP060105699A patent/AR058720A1/es active IP Right Grant
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2008
- 2008-05-05 IL IL191255A patent/IL191255A/en active IP Right Grant
- 2008-07-21 NO NO20083237A patent/NO341296B1/no unknown
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- 2010-09-09 US US12/878,831 patent/US8129427B2/en active Active
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2012
- 2012-01-26 US US13/359,285 patent/US8470877B2/en active Active
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2015
- 2015-12-30 CY CY20151101204T patent/CY1117094T1/el unknown
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