SI1811999T1 - Kinuklidinski derivati in njihova uporaba kot antagonisti muskarinskega M3 receptorja - Google Patents

Kinuklidinski derivati in njihova uporaba kot antagonisti muskarinskega M3 receptorja

Info

Publication number
SI1811999T1
SI1811999T1 SI200531188T SI200531188T SI1811999T1 SI 1811999 T1 SI1811999 T1 SI 1811999T1 SI 200531188 T SI200531188 T SI 200531188T SI 200531188 T SI200531188 T SI 200531188T SI 1811999 T1 SI1811999 T1 SI 1811999T1
Authority
SI
Slovenia
Prior art keywords
muscarinic
receptor antagonists
quinuclidine derivatives
quinuclidine
derivatives
Prior art date
Application number
SI200531188T
Other languages
English (en)
Inventor
Neil John Press
Stephen Paul Collingwood
Urs Baettig
Brian Cox
Sudhakar Devidasrao Garad
Hyungchul Kim
Dimitris Papoutsakis
Simon James Watson
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=33515948&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI1811999(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of SI1811999T1 publication Critical patent/SI1811999T1/sl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/16—Central respiratory analeptics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
SI200531188T 2004-11-02 2005-10-31 Kinuklidinski derivati in njihova uporaba kot antagonisti muskarinskega M3 receptorja SI1811999T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0424284.8A GB0424284D0 (en) 2004-11-02 2004-11-02 Organic compounds
EP05798470A EP1811999B1 (en) 2004-11-02 2005-10-31 Quinuclidine derivatives and their use as muscarinic m3 receptor antagonists
PCT/EP2005/011662 WO2006048225A1 (en) 2004-11-02 2005-10-31 Quinuclidine derivatives and their use as muscarinic m3 receptor antagonists

Publications (1)

Publication Number Publication Date
SI1811999T1 true SI1811999T1 (sl) 2011-01-31

Family

ID=33515948

Family Applications (1)

Application Number Title Priority Date Filing Date
SI200531188T SI1811999T1 (sl) 2004-11-02 2005-10-31 Kinuklidinski derivati in njihova uporaba kot antagonisti muskarinskega M3 receptorja

Country Status (33)

Country Link
US (2) US7723356B2 (sl)
EP (2) EP2206499A1 (sl)
JP (1) JP4950896B2 (sl)
KR (1) KR101252307B1 (sl)
CN (1) CN101056634B (sl)
AR (1) AR054090A1 (sl)
AT (1) ATE481099T1 (sl)
AU (1) AU2005300710B2 (sl)
BR (1) BRPI0517945A (sl)
CA (1) CA2583237C (sl)
CY (1) CY1110952T1 (sl)
DE (1) DE602005023639D1 (sl)
DK (1) DK1811999T3 (sl)
EC (1) ECSP077424A (sl)
ES (1) ES2353142T3 (sl)
GB (1) GB0424284D0 (sl)
HR (1) HRP20100693T1 (sl)
IL (1) IL182695A0 (sl)
JO (1) JO2613B1 (sl)
MA (1) MA29080B1 (sl)
MX (1) MX2007005189A (sl)
MY (1) MY145207A (sl)
NO (1) NO20072371L (sl)
NZ (1) NZ554302A (sl)
PE (1) PE20060609A1 (sl)
PL (1) PL1811999T3 (sl)
PT (1) PT1811999E (sl)
RU (1) RU2399620C2 (sl)
SI (1) SI1811999T1 (sl)
TN (1) TNSN07164A1 (sl)
TW (1) TW200628154A (sl)
WO (1) WO2006048225A1 (sl)
ZA (1) ZA200702772B (sl)

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JP5902612B2 (ja) 2009-04-09 2016-04-13 ノバルティス アーゲー ピロリジニウム塩の調製方法
EP2585457B1 (en) * 2010-06-22 2015-07-22 Chiesi Farmaceutici S.p.A. Alkaloid aminoester derivatives and medicinal composition thereof
AU2011269238A1 (en) * 2010-06-22 2013-01-10 Chiesi Farmaceutici S.P.A. Dry powder formulation comprising an antimuscarinic drug
US8637516B2 (en) 2010-09-09 2014-01-28 Irm Llc Compounds and compositions as TRK inhibitors
WO2012034095A1 (en) 2010-09-09 2012-03-15 Irm Llc Compounds and compositions as trk inhibitors
CN103492384B (zh) 2011-02-25 2016-05-11 诺华股份有限公司 作为trk抑制剂的化合物和组合物
JP2011195593A (ja) * 2011-06-30 2011-10-06 Astrazeneca Ab ムスカリンｍ３受容体アンタゴニストとしてのキヌクリジン誘導体
EA028509B1 (ru) 2012-12-19 2017-11-30 Новартис Аг Ингибиторы аутотаксина, фармацевтические композиции и комбинации, содержащие их, и их применение в лечении заболеваний и состояний, опосредованных аутотаксином
WO2015162558A1 (en) 2014-04-24 2015-10-29 Novartis Ag Autotaxin inhibitors
CA3193201A1 (en) * 2014-05-06 2015-11-12 Anthony G. Visco Methods of treating or preventing preterm labor
CN109851615B (zh) * 2019-04-22 2021-06-08 上海旭东海普药业有限公司 纯化戊乙奎醚的方法

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