BR112012032333A2 - composto, uso de um composto, composição farmacêutica, combinação de um composto e dispositivo - Google Patents
composto, uso de um composto, composição farmacêutica, combinação de um composto e dispositivoInfo
- Publication number
- BR112012032333A2 BR112012032333A2 BR112012032333A BR112012032333A BR112012032333A2 BR 112012032333 A2 BR112012032333 A2 BR 112012032333A2 BR 112012032333 A BR112012032333 A BR 112012032333A BR 112012032333 A BR112012032333 A BR 112012032333A BR 112012032333 A2 BR112012032333 A2 BR 112012032333A2
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- combination
- pharmaceutical composition
- pharmaceutical
- composition
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pulmonology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP10166898 | 2010-06-22 | ||
PCT/EP2011/058801 WO2011160918A1 (en) | 2010-06-22 | 2011-05-30 | Alkaloid aminoester derivatives and medicinal composition thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112012032333A2 true BR112012032333A2 (pt) | 2016-11-08 |
Family
ID=43303945
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112012032333A BR112012032333A2 (pt) | 2010-06-22 | 2011-05-30 | composto, uso de um composto, composição farmacêutica, combinação de um composto e dispositivo |
Country Status (11)
Country | Link |
---|---|
US (1) | US8629160B2 (pt) |
EP (1) | EP2585457B1 (pt) |
KR (1) | KR20130111968A (pt) |
CN (1) | CN102947298B (pt) |
AR (1) | AR081965A1 (pt) |
BR (1) | BR112012032333A2 (pt) |
CA (1) | CA2803416A1 (pt) |
ES (1) | ES2545812T3 (pt) |
HK (1) | HK1181047A1 (pt) |
RU (1) | RU2569846C2 (pt) |
WO (1) | WO2011160918A1 (pt) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2206712A1 (en) | 2008-12-23 | 2010-07-14 | CHIESI FARMACEUTICI S.p.A. | "Alkaloid aminoester derivatives and medicinal composition thereof" |
CA2803459A1 (en) * | 2010-06-22 | 2011-12-29 | Chiesi Farmaceutici S.P.A. | Alkaloid aminoester derivatives and medicinal compositions thereof |
RU2585767C2 (ru) | 2010-11-26 | 2016-06-10 | КЬЕЗИ ФАРМАЧЕУТИЧИ С.п.А. | Производные глицина и их применение в качестве антагонистов мускариновых рецепторов |
CN104011043B (zh) | 2011-12-30 | 2016-11-16 | 奇斯药制品公司 | 作为抗毒蕈碱剂的1-氮杂杂环基乙酸的奎宁环酯、它们的制备方法及其药用组合物 |
US9427376B2 (en) | 2013-10-10 | 2016-08-30 | Chiesi Farmaceutici S.P.A. | Process for preparing pharmaceutical formulations for inhalation comprising a high-dosage strength active ingredient |
Family Cites Families (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2824106A (en) * | 1958-02-18 | Quaternary tropeine compounds and a process of making same | ||
US2856407A (en) * | 1956-08-08 | 1958-10-14 | Lakeside Lab Inc | Aminoacid esters of n-substituted 3 and 4-piperidinols |
GB8923590D0 (en) * | 1989-10-19 | 1989-12-06 | Pfizer Ltd | Antimuscarinic bronchodilators |
US6169075B1 (en) * | 1996-09-10 | 2001-01-02 | British Biotech Pharmaceuticals Limited | Cytostatic agents |
JP2001520222A (ja) * | 1997-10-22 | 2001-10-30 | ゼネカ・リミテッド | イミダゾール誘導体およびファルネシルタンパク質トランスフェラーゼインヒビターとしてのそれらの使用 |
IL156499A0 (en) * | 2000-12-22 | 2004-01-04 | Almirall Prodesfarma Ag | Quinuclidine carbamate derivatives and their use as m3 antagonists |
MXPA04006206A (es) | 2001-12-20 | 2004-12-06 | S A L V A T Lab Sa | Derivados de 1-alquil-azoniabiciclo(2.2.2(octano carbamato y su uso como antagonistas del receptor musrcarinico. |
GB0424284D0 (en) * | 2004-11-02 | 2004-12-01 | Novartis Ag | Organic compounds |
EP1882691A1 (en) * | 2006-07-26 | 2008-01-30 | CHIESI FARMACEUTICI S.p.A. | Quinuclidine derivatives as M3 antagonists |
GB0621830D0 (en) * | 2006-11-02 | 2006-12-13 | Chroma Therapeutics Ltd | Inhibitors of p38 mitogen-activated protein kinase |
TW200825084A (en) * | 2006-11-14 | 2008-06-16 | Astrazeneca Ab | New compounds 521 |
ES2385681T3 (es) * | 2006-12-19 | 2012-07-30 | Astrazeneca Ab | Derivados de quinuclidinol como antagonistas de receptores muscarínicos |
WO2008075006A1 (en) * | 2006-12-19 | 2008-06-26 | Astrazeneca Ab | Piperldinum compounds for treatment of obstructive pulmonary diseases ( copd) |
EP2154136A1 (en) | 2008-08-08 | 2010-02-17 | CHIESI FARMACEUTICI S.p.A. | Quinuclidine carbonate derivatives and medicinal compositions thereof |
EP2206712A1 (en) | 2008-12-23 | 2010-07-14 | CHIESI FARMACEUTICI S.p.A. | "Alkaloid aminoester derivatives and medicinal composition thereof" |
EP2585458B1 (en) * | 2010-06-22 | 2015-01-07 | Chiesi Farmaceutici S.p.A. | Alkaloid aminoester derivatives and medicinal compositions thereof |
AU2011269238A1 (en) * | 2010-06-22 | 2013-01-10 | Chiesi Farmaceutici S.P.A. | Dry powder formulation comprising an antimuscarinic drug |
CA2803459A1 (en) * | 2010-06-22 | 2011-12-29 | Chiesi Farmaceutici S.P.A. | Alkaloid aminoester derivatives and medicinal compositions thereof |
US20120220557A1 (en) * | 2011-02-17 | 2012-08-30 | Chiesi Farmaceutici S.P.A. | Liquid propellant-free formulation comprising an antimuscarinic drug |
-
2011
- 2011-05-30 CN CN201180030597.9A patent/CN102947298B/zh not_active Expired - Fee Related
- 2011-05-30 ES ES11724157.0T patent/ES2545812T3/es active Active
- 2011-05-30 CA CA2803416A patent/CA2803416A1/en not_active Abandoned
- 2011-05-30 KR KR1020127033567A patent/KR20130111968A/ko not_active Application Discontinuation
- 2011-05-30 EP EP11724157.0A patent/EP2585457B1/en active Active
- 2011-05-30 RU RU2012155690/04A patent/RU2569846C2/ru active
- 2011-05-30 BR BR112012032333A patent/BR112012032333A2/pt not_active IP Right Cessation
- 2011-05-30 WO PCT/EP2011/058801 patent/WO2011160918A1/en active Application Filing
- 2011-06-21 AR ARP110102147A patent/AR081965A1/es unknown
- 2011-06-22 US US13/165,936 patent/US8629160B2/en active Active
-
2013
- 2013-07-16 HK HK13108338.9A patent/HK1181047A1/zh not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
CN102947298A (zh) | 2013-02-27 |
EP2585457A1 (en) | 2013-05-01 |
US20110311461A1 (en) | 2011-12-22 |
US8629160B2 (en) | 2014-01-14 |
AR081965A1 (es) | 2012-10-31 |
RU2012155690A (ru) | 2014-06-27 |
HK1181047A1 (zh) | 2013-11-01 |
ES2545812T3 (es) | 2015-09-16 |
WO2011160918A1 (en) | 2011-12-29 |
CA2803416A1 (en) | 2011-12-29 |
RU2569846C2 (ru) | 2015-11-27 |
CN102947298B (zh) | 2016-03-02 |
EP2585457B1 (en) | 2015-07-22 |
KR20130111968A (ko) | 2013-10-11 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] | ||
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |