SI1534390T1 - Z dimetilfenil dihidro metil okso H pirazol iliden hidrazino hidroksi bifenil karboksilna kislina bis monoetanolamin - Google Patents

Z dimetilfenil dihidro metil okso H pirazol iliden hidrazino hidroksi bifenil karboksilna kislina bis monoetanolamin

Info

Publication number
SI1534390T1
SI1534390T1 SI200331773T SI200331773T SI1534390T1 SI 1534390 T1 SI1534390 T1 SI 1534390T1 SI 200331773 T SI200331773 T SI 200331773T SI 200331773 T SI200331773 T SI 200331773T SI 1534390 T1 SI1534390 T1 SI 1534390T1
Authority
SI
Slovenia
Prior art keywords
hydrazino
ylidene
pyrazol
dimethylphenyl
monoethanolamine
Prior art date
Application number
SI200331773T
Other languages
English (en)
Inventor
Stephen Moore
Original Assignee
Glaxosmithkline Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=29584468&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI1534390(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Glaxosmithkline Llc filed Critical Glaxosmithkline Llc
Publication of SI1534390T1 publication Critical patent/SI1534390T1/sl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/44—Oxygen and nitrogen or sulfur and nitrogen atoms
    • C07D231/46—Oxygen atom in position 3 or 5 and nitrogen atom in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4152—1,2-Diazoles having oxo groups directly attached to the heterocyclic ring, e.g. antipyrine, phenylbutazone, sulfinpyrazone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/19—Cytokines; Lymphokines; Interferons
    • A61K38/193—Colony stimulating factors [CSF]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/04—Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/06—Antianaemics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D231/08—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with oxygen or sulfur atoms directly attached to ring carbon atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Zoology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
SI200331773T 2002-05-22 2003-05-21 Z dimetilfenil dihidro metil okso H pirazol iliden hidrazino hidroksi bifenil karboksilna kislina bis monoetanolamin SI1534390T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US38287102P 2002-05-22 2002-05-22
EP03731335A EP1534390B1 (en) 2002-05-22 2003-05-21 3'- (2z)- 1-(3,4-dimethylphenyl)-1,5-dihydro-3-methyl-5-oxo-4h-pyrazol-4-ylidene hydrazino -2'-hydroxy- 1,1'-biphenyl -3-carboxylic acid bis-(monoethanolamine)
PCT/US2003/016255 WO2003098992A2 (en) 2002-05-22 2003-05-21 3'-[(2z)-[1-(3,4-dimethylphenyl)-1,5-dihydro-3-methyl-5-oxo-4h-pyrazol-4-ylidene]hydrazino]-2'-hydroxy-[1,1'-biphenyl]-3-carboxylic acid bis-(monoethanolamine)

Publications (1)

Publication Number Publication Date
SI1534390T1 true SI1534390T1 (sl) 2010-05-31

Family

ID=29584468

Family Applications (1)

Application Number Title Priority Date Filing Date
SI200331773T SI1534390T1 (sl) 2002-05-22 2003-05-21 Z dimetilfenil dihidro metil okso H pirazol iliden hidrazino hidroksi bifenil karboksilna kislina bis monoetanolamin

Country Status (29)

Country Link
US (6) US7547719B2 (sl)
EP (2) EP2206533A3 (sl)
JP (2) JP4612414B2 (sl)
KR (2) KR101090643B1 (sl)
CN (1) CN100542530C (sl)
AR (1) AR040083A1 (sl)
AT (1) ATE452683T1 (sl)
AU (1) AU2003241587B2 (sl)
BR (1) BRPI0310094B8 (sl)
CA (1) CA2486697C (sl)
CY (1) CY1109912T1 (sl)
DE (1) DE60330674D1 (sl)
DK (1) DK1534390T3 (sl)
ES (1) ES2338108T3 (sl)
HK (1) HK1078039A1 (sl)
IL (2) IL164966A0 (sl)
IS (1) IS2770B (sl)
LT (1) LTC1534390I2 (sl)
MX (1) MXPA04011522A (sl)
MY (1) MY142390A (sl)
NO (1) NO330160B1 (sl)
NZ (1) NZ536272A (sl)
PL (1) PL212682B1 (sl)
PT (1) PT1534390E (sl)
RU (1) RU2284994C9 (sl)
SI (1) SI1534390T1 (sl)
TW (1) TWI280128B (sl)
WO (1) WO2003098992A2 (sl)
ZA (1) ZA200408701B (sl)

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TW200407128A (en) 2004-05-16
US20140037580A1 (en) 2014-02-06
CA2486697A1 (en) 2003-12-04
EP2206533A3 (en) 2010-09-15
ATE452683T1 (de) 2010-01-15
US7547719B2 (en) 2009-06-16
US20120189576A1 (en) 2012-07-26
EP1534390A4 (en) 2008-03-12
DE60330674D1 (de) 2010-02-04
US20150079030A1 (en) 2015-03-19
US8088813B2 (en) 2012-01-03
LTC1534390I2 (lt) 2020-06-10
RU2284994C2 (ru) 2006-10-10
HK1078039A1 (en) 2006-03-03
IL199438A (en) 2011-06-30
MXPA04011522A (es) 2005-02-14
NZ536272A (en) 2007-08-31
CN100542530C (zh) 2009-09-23
RU2004137491A (ru) 2005-06-10
AU2003241587B2 (en) 2007-10-04
LTPA2010007I1 (lt) 2019-11-11
US7795293B2 (en) 2010-09-14
IS2770B (is) 2011-12-15
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DK1534390T3 (da) 2010-04-26
BRPI0310094B1 (pt) 2018-10-23
CA2486697C (en) 2009-01-06
EP1534390B1 (en) 2009-12-23
EP2206533A2 (en) 2010-07-14
PL372440A1 (en) 2005-07-25
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