SG11201805004TA - Substituted 4-phenyl pyridine compounds as non-systemic tgr5 agonists - Google Patents

Substituted 4-phenyl pyridine compounds as non-systemic tgr5 agonists

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Publication number
SG11201805004TA
SG11201805004TA SG11201805004TA SG11201805004TA SG11201805004TA SG 11201805004T A SG11201805004T A SG 11201805004TA SG 11201805004T A SG11201805004T A SG 11201805004TA SG 11201805004T A SG11201805004T A SG 11201805004TA SG 11201805004T A SG11201805004T A SG 11201805004TA
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SG
Singapore
Prior art keywords
california
international
avenue
co7d
pct
Prior art date
Application number
SG11201805004TA
Other languages
English (en)
Inventor
Jason G Lewis
Michael Robert Leadbetter
Jeremy Caldwell
Dean Dragoli
Noah Bell
Jeffrey W Jacobs
Patricia Finn
Rakesh Jain
Tao Chen
Matthew Siegel
Original Assignee
Ardelyx Inc
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Publication date
Application filed by Ardelyx Inc filed Critical Ardelyx Inc
Publication of SG11201805004TA publication Critical patent/SG11201805004TA/en

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    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/26—Acyclic or carbocyclic radicals, substituted by hetero rings
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4418—Non condensed pyridines; Hydrogenated derivatives thereof having a carbocyclic group directly attached to the heterocyclic ring, e.g. cyproheptadine
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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