SG10202100915RA - 3-alkyl-4-amido-bicyclic [4,5,0] hydroxamic acids as hdac inhibitors - Google Patents
3-alkyl-4-amido-bicyclic [4,5,0] hydroxamic acids as hdac inhibitorsInfo
- Publication number
- SG10202100915RA SG10202100915RA SG10202100915RA SG10202100915RA SG10202100915RA SG 10202100915R A SG10202100915R A SG 10202100915RA SG 10202100915R A SG10202100915R A SG 10202100915RA SG 10202100915R A SG10202100915R A SG 10202100915RA SG 10202100915R A SG10202100915R A SG 10202100915RA
- Authority
- SG
- Singapore
- Prior art keywords
- amido
- bicyclic
- alkyl
- hdac inhibitors
- hydroxamic acids
- Prior art date
Links
Classifications
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- C07D267/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D267/02—Seven-membered rings
- C07D267/08—Seven-membered rings having the hetero atoms in positions 1 and 4
- C07D267/12—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D267/14—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/553—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one oxygen as ring hetero atoms, e.g. loxapine, staurosporine
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- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
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- C07D267/08—Seven-membered rings having the hetero atoms in positions 1 and 4
- C07D267/12—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
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- Animal Behavior & Ethology (AREA)
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Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
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US201562110716P | 2015-02-02 | 2015-02-02 | |
US201562205438P | 2015-08-14 | 2015-08-14 |
Publications (1)
Publication Number | Publication Date |
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SG10202100915RA true SG10202100915RA (en) | 2021-02-25 |
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Family Applications (4)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SG10202100916PA SG10202100916PA (en) | 2015-02-02 | 2016-02-02 | 3-aryl-4-amido-bicyclic [4,5,0] hydroxamic acids as hdac inhibitors |
SG11201708622UA SG11201708622UA (en) | 2015-02-02 | 2016-02-02 | 3-aryl-4-amido-bicyclic [4,5,0] hydroxamic acids as hdac inhibitors |
SG10202100915RA SG10202100915RA (en) | 2015-02-02 | 2016-02-02 | 3-alkyl-4-amido-bicyclic [4,5,0] hydroxamic acids as hdac inhibitors |
SG11201706146UA SG11201706146UA (en) | 2015-02-02 | 2016-02-02 | 3-alkyl-4-amido-bicyclic [4,5,0] hydroxamic acids as hdac inhibitors |
Family Applications Before (2)
Application Number | Title | Priority Date | Filing Date |
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SG10202100916PA SG10202100916PA (en) | 2015-02-02 | 2016-02-02 | 3-aryl-4-amido-bicyclic [4,5,0] hydroxamic acids as hdac inhibitors |
SG11201708622UA SG11201708622UA (en) | 2015-02-02 | 2016-02-02 | 3-aryl-4-amido-bicyclic [4,5,0] hydroxamic acids as hdac inhibitors |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
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SG11201706146UA SG11201706146UA (en) | 2015-02-02 | 2016-02-02 | 3-alkyl-4-amido-bicyclic [4,5,0] hydroxamic acids as hdac inhibitors |
Country Status (27)
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US (32) | US10112915B2 (es) |
EP (3) | EP3253747B1 (es) |
JP (1) | JP6668362B2 (es) |
KR (1) | KR102633628B1 (es) |
CN (3) | CN114057765A (es) |
AU (4) | AU2016215431B2 (es) |
BR (1) | BR112017016493B1 (es) |
CA (2) | CA2990165C (es) |
CL (1) | CL2017001968A1 (es) |
CO (1) | CO2017007863A2 (es) |
DK (1) | DK3292116T3 (es) |
EA (2) | EA036711B1 (es) |
EC (1) | ECSP17055491A (es) |
ES (2) | ES2770123T3 (es) |
HK (2) | HK1251550A1 (es) |
HU (1) | HUE057623T2 (es) |
IL (4) | IL280856B (es) |
MA (1) | MA42032A (es) |
MX (2) | MX2017009950A (es) |
MY (1) | MY191591A (es) |
PH (1) | PH12017501383A1 (es) |
PL (1) | PL3292116T3 (es) |
PT (1) | PT3292116T (es) |
SA (1) | SA517382027B1 (es) |
SG (4) | SG10202100916PA (es) |
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