SE512835C2 - Doseringsform innehållande en mångfald enheter alla inneslutande syralabil H+K+ATPas-hämmare - Google Patents
Doseringsform innehållande en mångfald enheter alla inneslutande syralabil H+K+ATPas-hämmareInfo
- Publication number
- SE512835C2 SE512835C2 SE9600073A SE9600073A SE512835C2 SE 512835 C2 SE512835 C2 SE 512835C2 SE 9600073 A SE9600073 A SE 9600073A SE 9600073 A SE9600073 A SE 9600073A SE 512835 C2 SE512835 C2 SE 512835C2
- Authority
- SE
- Sweden
- Prior art keywords
- dosage form
- tableted
- effervescent
- units
- individual
- Prior art date
Links
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- FEWJPZIEWOKRBE-UHFFFAOYSA-N Tartaric acid Natural products [H+].[H+].[O-]C(=O)C(O)C(O)C([O-])=O FEWJPZIEWOKRBE-UHFFFAOYSA-N 0.000 description 1
- 239000003929 acidic solution Substances 0.000 description 1
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- 229910052784 alkaline earth metal Inorganic materials 0.000 description 1
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- 229960004543 anhydrous citric acid Drugs 0.000 description 1
- 239000012736 aqueous medium Substances 0.000 description 1
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- 208000027687 belching Diseases 0.000 description 1
- 235000019658 bitter taste Nutrition 0.000 description 1
- 229910000019 calcium carbonate Inorganic materials 0.000 description 1
- AXCZMVOFGPJBDE-UHFFFAOYSA-L calcium dihydroxide Chemical compound [OH-].[OH-].[Ca+2] AXCZMVOFGPJBDE-UHFFFAOYSA-L 0.000 description 1
- 239000000920 calcium hydroxide Substances 0.000 description 1
- 229910001861 calcium hydroxide Inorganic materials 0.000 description 1
- 239000000378 calcium silicate Substances 0.000 description 1
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- 125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 description 1
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- CEYULKASIQJZGP-UHFFFAOYSA-L disodium;2-(carboxymethyl)-2-hydroxybutanedioate Chemical compound [Na+].[Na+].[O-]C(=O)CC(O)(C(=O)O)CC([O-])=O CEYULKASIQJZGP-UHFFFAOYSA-L 0.000 description 1
- 239000002270 dispersing agent Substances 0.000 description 1
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- 229960003276 erythromycin Drugs 0.000 description 1
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- 235000013355 food flavoring agent Nutrition 0.000 description 1
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- XLYOFNOQVPJJNP-UHFFFAOYSA-M hydroxide Chemical compound [OH-] XLYOFNOQVPJJNP-UHFFFAOYSA-M 0.000 description 1
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- 229920000639 hydroxypropylmethylcellulose acetate succinate Polymers 0.000 description 1
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- 239000000347 magnesium hydroxide Substances 0.000 description 1
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- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 description 1
- FYFFGSSZFBZTAH-UHFFFAOYSA-N methylaminomethanetriol Chemical compound CNC(O)(O)O FYFFGSSZFBZTAH-UHFFFAOYSA-N 0.000 description 1
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- 229920000620 organic polymer Polymers 0.000 description 1
- 230000000149 penetrating effect Effects 0.000 description 1
- PNJWIWWMYCMZRO-UHFFFAOYSA-N pent‐4‐en‐2‐one Natural products CC(=O)CC=C PNJWIWWMYCMZRO-UHFFFAOYSA-N 0.000 description 1
- 150000003022 phthalic acids Chemical class 0.000 description 1
- 229920001223 polyethylene glycol Polymers 0.000 description 1
- 229940068965 polysorbates Drugs 0.000 description 1
- 239000002243 precursor Substances 0.000 description 1
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- HNJBEVLQSNELDL-UHFFFAOYSA-N pyrrolidin-2-one Chemical compound O=C1CCCN1 HNJBEVLQSNELDL-UHFFFAOYSA-N 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
- A61K9/0007—Effervescent
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Priority Applications (33)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE9600073A SE512835C2 (sv) | 1996-01-08 | 1996-01-08 | Doseringsform innehållande en mångfald enheter alla inneslutande syralabil H+K+ATPas-hämmare |
| PT96944727T PT814783E (pt) | 1996-01-08 | 1996-12-20 | Formas de dosagem efervescente de unidades multiplas que compreendem um inibidor da bomba de protoes |
| KR1019970706237A KR100459363B1 (ko) | 1996-01-08 | 1996-12-20 | 양성자펌프억제제를함유하는다단위발포성제형 |
| NZ325978A NZ325978A (en) | 1996-01-08 | 1996-12-20 | Enteric coated effervescent tablet containing a proton pump inhibitor, in particular, s-omeprazole |
| CNB961937637A CN100335043C (zh) | 1996-01-08 | 1996-12-20 | 片剂化多重单元泡腾剂剂型口服药物组合物及其生产方法 |
| IL12165396A IL121653A (en) | 1996-01-08 | 1996-12-20 | Vibrant dosage forms with multiple units that include a proton pump inhibitor |
| PCT/SE1996/001738 WO1997025030A1 (en) | 1996-01-08 | 1996-12-20 | Multiple unit effervescent dosage forms comprising protonpump inhibitor |
| BR9607367A BR9607367A (pt) | 1996-01-08 | 1996-12-20 | Forma de múltipla dosagem unitária em tablete efervecente processos para preparação da mesma para a inibição de secreção de ácido gástrico em mamíferos e no homem e para o tratamento de doenças gastrointestinais inflamatórias em maniferos e no homem e uso da forma de dosagem em tablete efervecente |
| DE69630286T DE69630286T2 (de) | 1996-01-08 | 1996-12-20 | Aus mehreren einzeleinheiten zusammengesetzte dosierungsformen enthaltend einem protonen pumpen inhibitor |
| ES96944727T ES2208775T3 (es) | 1996-01-08 | 1996-12-20 | Formas de dosificacion efervescentes de multiples unidades que comprenden inhibidor de la bomba de protones. |
| CA002214027A CA2214027C (en) | 1996-01-08 | 1996-12-20 | Multiple unit effervescent dosage forms comprising proton pump inhibitor |
| EP96944727A EP0814783B1 (en) | 1996-01-08 | 1996-12-20 | Multiple unit effervescent dosage forms comprising protonpump inhibitor |
| SK1171-97A SK117197A3 (en) | 1996-01-08 | 1996-12-20 | Multiple unit effervescent dosage forms comprising protonpump inhibitor |
| PL96322161A PL322161A1 (en) | 1996-01-08 | 1996-12-20 | Multiple-component single-dose effervescent administration forms containing the protonic pump inhibitor |
| CZ972807A CZ280797A3 (cs) | 1996-01-08 | 1996-12-20 | Vícesložková efervescentní léková forma zahrnující inhibitor protonové pumpy |
| JP52513297A JP4638561B2 (ja) | 1996-01-08 | 1996-12-20 | プロトンポンプ抑制剤を含有するマルチプルユニットの沸騰剤形 |
| DK96944727T DK0814783T3 (da) | 1996-01-08 | 1996-12-20 | Opbruselige multienhedsdoseringsformer, der omfatter en protonpumpeinhibitor |
| AU13242/97A AU712325B2 (en) | 1996-01-08 | 1996-12-20 | Multiple unit effervescent dosage forms comprising protonpump inhibitor |
| US08/793,077 US6132770A (en) | 1996-01-08 | 1996-12-20 | Multiple unit effervescent dosage forms comprising proton pump inhibitor |
| EE9700189A EE9700189A (et) | 1996-01-08 | 1996-12-20 | Mitmikühikuline kihisev annusvorm, mis sisaldab prootonpumba inhibiitorit |
| AT96944727T ATE251451T1 (de) | 1996-01-08 | 1996-12-20 | Aus mehreren einzeleinheiten zusammengesetzte dosierungsformen enthaltend einem protonen pumpen inhibitor |
| MX9706768A MX9706768A (es) | 1996-01-08 | 1996-12-20 | Formas de dosificacion efervecente de unidades multiples que contienen inhibidor de la bomba de protones. |
| TR97/00918T TR199700918T1 (xx) | 1996-01-08 | 1996-12-20 | �oklu birimli efervesan dozaj formlar�. |
| SI9630657T SI0814783T1 (sl) | 1996-01-08 | 1996-12-20 | Multiple enotske šumeče dozirne oblike, ki obsegajo inhibitor protonske črpalke |
| HU0000976A HUP0000976A3 (en) | 1996-01-08 | 1996-12-20 | Multiple unit effervescent tablet dosage forms comprising protonpump inhibitor |
| YU70196A YU70196A (sh) | 1996-01-08 | 1996-12-26 | Tabletirani šumeći oblici doziranja i postupci za njihovo dobijanje |
| ARP960105897A AR005280A1 (es) | 1996-01-08 | 1996-12-26 | Forma de dosis efervescente unitaria multiple en tabletas, proceso para su fabricacion y uso de dicha forma para la fabricacion de medicamentos. |
| ZA9610939A ZA9610939B (en) | 1996-01-08 | 1996-12-30 | Multiple unit effervescent dosage forms |
| HR9600073-2A HRP970005A2 (en) | 1996-01-08 | 1997-01-03 | Multiple unit effervescent dosage forms |
| TNTNSN97002A TNSN97002A1 (fr) | 1996-01-08 | 1997-01-06 | Presentations effervescentes a unites de prise multiples |
| IDP970023A ID15819A (id) | 1996-01-08 | 1997-01-08 | Bentuk sediaan efervesen satuan ganda |
| IS4551A IS4551A (is) | 1996-01-08 | 1997-08-25 | Freyðandi fjöleininga-skammtaform sem inniheldur prótónupumpublokkara |
| NO19974051A NO319999B1 (no) | 1996-01-08 | 1997-09-03 | Tabletterte, brusende multippelenhet-doseringsformer omfattende en protonpumpeinhibitor, fremgangsmate for fremstilling av slike doseringsformer, og anvendelse derav. |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE9600073A SE512835C2 (sv) | 1996-01-08 | 1996-01-08 | Doseringsform innehållande en mångfald enheter alla inneslutande syralabil H+K+ATPas-hämmare |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| SE9600073D0 SE9600073D0 (sv) | 1996-01-08 |
| SE9600073L SE9600073L (sv) | 1997-07-09 |
| SE512835C2 true SE512835C2 (sv) | 2000-05-22 |
Family
ID=20400971
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SE9600073A SE512835C2 (sv) | 1996-01-08 | 1996-01-08 | Doseringsform innehållande en mångfald enheter alla inneslutande syralabil H+K+ATPas-hämmare |
Country Status (33)
| Country | Link |
|---|---|
| US (1) | US6132770A (sl) |
| EP (1) | EP0814783B1 (sl) |
| JP (1) | JP4638561B2 (sl) |
| KR (1) | KR100459363B1 (sl) |
| CN (1) | CN100335043C (sl) |
| AR (1) | AR005280A1 (sl) |
| AT (1) | ATE251451T1 (sl) |
| AU (1) | AU712325B2 (sl) |
| BR (1) | BR9607367A (sl) |
| CA (1) | CA2214027C (sl) |
| CZ (1) | CZ280797A3 (sl) |
| DE (1) | DE69630286T2 (sl) |
| DK (1) | DK0814783T3 (sl) |
| EE (1) | EE9700189A (sl) |
| ES (1) | ES2208775T3 (sl) |
| HR (1) | HRP970005A2 (sl) |
| HU (1) | HUP0000976A3 (sl) |
| ID (1) | ID15819A (sl) |
| IL (1) | IL121653A (sl) |
| IS (1) | IS4551A (sl) |
| MX (1) | MX9706768A (sl) |
| NO (1) | NO319999B1 (sl) |
| NZ (1) | NZ325978A (sl) |
| PL (1) | PL322161A1 (sl) |
| PT (1) | PT814783E (sl) |
| SE (1) | SE512835C2 (sl) |
| SI (1) | SI0814783T1 (sl) |
| SK (1) | SK117197A3 (sl) |
| TN (1) | TNSN97002A1 (sl) |
| TR (1) | TR199700918T1 (sl) |
| WO (1) | WO1997025030A1 (sl) |
| YU (1) | YU70196A (sl) |
| ZA (1) | ZA9610939B (sl) |
Families Citing this family (62)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6558952B1 (en) * | 1992-12-14 | 2003-05-06 | Waratah Pharmaceuticals, Inc. | Treatment for diabetes |
| US5840737A (en) | 1996-01-04 | 1998-11-24 | The Curators Of The University Of Missouri | Omeprazole solution and method for using same |
| US6699885B2 (en) | 1996-01-04 | 2004-03-02 | The Curators Of The University Of Missouri | Substituted benzimidazole dosage forms and methods of using same |
| US6645988B2 (en) | 1996-01-04 | 2003-11-11 | Curators Of The University Of Missouri | Substituted benzimidazole dosage forms and method of using same |
| US6489346B1 (en) * | 1996-01-04 | 2002-12-03 | The Curators Of The University Of Missouri | Substituted benzimidazole dosage forms and method of using same |
| US20050054682A1 (en) * | 1996-01-04 | 2005-03-10 | Phillips Jeffrey O. | Pharmaceutical compositions comprising substituted benzimidazoles and methods of using same |
| SE512835C2 (sv) * | 1996-01-08 | 2000-05-22 | Astrazeneca Ab | Doseringsform innehållande en mångfald enheter alla inneslutande syralabil H+K+ATPas-hämmare |
| SE9702533D0 (sv) | 1997-07-01 | 1997-07-01 | Astra Ab | New oral formulation |
| JP4546643B2 (ja) * | 1997-12-08 | 2010-09-15 | ニコメッド ゲゼルシャフト ミット ベシュレンクテル ハフツング | 酸不安定な活性化合物を含有する新規の坐剤形 |
| EP1056456A4 (en) * | 1998-01-30 | 2006-10-25 | Sepracor Inc | R-LANSOPRAZOL COMPOSITIONS AND TREATMENTS THEREFOR |
| US6328994B1 (en) * | 1998-05-18 | 2001-12-11 | Takeda Chemical Industries, Ltd. | Orally disintegrable tablets |
| TWI257311B (en) * | 1998-07-28 | 2006-07-01 | Takeda Chemical Industries Ltd | Rapidly disintegrable solid preparation |
| AU4040800A (en) * | 1999-03-29 | 2000-10-16 | American Home Products Corporation | Coating system |
| US6174902B1 (en) | 1999-04-28 | 2001-01-16 | Sepracor Inc. | R-rabeprazole compositions and methods |
| AU775995B2 (en) | 1999-06-07 | 2004-08-19 | Nycomed Gmbh | Novel preparation and administration form comprising an acid-labile active compound |
| US6316020B1 (en) | 1999-08-26 | 2001-11-13 | Robert R. Whittle | Pharmaceutical formulations |
| US20020064555A1 (en) * | 2000-09-29 | 2002-05-30 | Dan Cullen | Proton pump inhibitor formulation |
| ATE541564T1 (de) | 2000-12-07 | 2012-02-15 | Nycomed Gmbh | Schnell zerfallende tablette mit einem säurelabilen wirkstoff |
| UA80393C2 (uk) | 2000-12-07 | 2007-09-25 | Алтана Фарма Аг | Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці |
| US20020192299A1 (en) * | 2000-12-28 | 2002-12-19 | Rajneesh Taneja | Pharmaceutical compositions of a non-enteric coated proton pump inhibitor with a carbonate salt and bicarbonate salt combination |
| MXPA04007169A (es) * | 2002-01-25 | 2004-10-29 | Santarus Inc | Suministro transmucosal de inhibidores de bomba de protones. |
| MY140561A (en) | 2002-02-20 | 2009-12-31 | Nycomed Gmbh | Dosage form containing pde 4 inhibitor as active ingredient |
| PL372409A1 (en) | 2002-03-27 | 2005-07-25 | Altana Pharma Ag | Novel alkoxypyridine-derivatives |
| FR2838647B1 (fr) * | 2002-04-23 | 2006-02-17 | Particules enrobees a liberation prolongee, leur procede de preparation et comprimes les contenant | |
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- 1996-12-20 WO PCT/SE1996/001738 patent/WO1997025030A1/en active IP Right Grant
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| NUG | Patent has lapsed |