SE408642B - Analogiforfarande for framstellning av n-tienylmettlderivat av morfinaner och bensomorfaner - Google Patents

Analogiforfarande for framstellning av n-tienylmettlderivat av morfinaner och bensomorfaner

Info

Publication number
SE408642B
SE408642B SE7305148A SE7305148A SE408642B SE 408642 B SE408642 B SE 408642B SE 7305148 A SE7305148 A SE 7305148A SE 7305148 A SE7305148 A SE 7305148A SE 408642 B SE408642 B SE 408642B
Authority
SE
Sweden
Prior art keywords
formula
compound
acid
hydroxy
thienylmethyl
Prior art date
Application number
SE7305148A
Other languages
English (en)
Swedish (sv)
Inventor
H Merz
A Langbein
K Stockhaus
H Wick
Original Assignee
Boehringer Sohn Ingelheim
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Sohn Ingelheim filed Critical Boehringer Sohn Ingelheim
Publication of SE408642B publication Critical patent/SE408642B/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/485Morphinan derivatives, e.g. morphine, codeine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/22Bridged ring systems
    • C07D221/26Benzomorphans

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
SE7305148A 1972-04-12 1973-04-11 Analogiforfarande for framstellning av n-tienylmettlderivat av morfinaner och bensomorfaner SE408642B (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2217420A DE2217420C3 (de) 1972-04-12 1972-04-12 N-Thienylmethyl-Heterocyclen, Verfahren zu deren Herstellung und diese enthaltende pharmazeutische Zubereitungen

Publications (1)

Publication Number Publication Date
SE408642B true SE408642B (sv) 1979-06-25

Family

ID=5841625

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7305148A SE408642B (sv) 1972-04-12 1973-04-11 Analogiforfarande for framstellning av n-tienylmettlderivat av morfinaner och bensomorfaner

Country Status (7)

Country Link
US (1) US3917606A (da)
DE (1) DE2217420C3 (da)
DK (1) DK133555C (da)
FI (1) FI57409C (da)
GB (1) GB1425347A (da)
NO (1) NO137695C (da)
SE (1) SE408642B (da)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2437610A1 (de) * 1974-08-05 1976-02-26 Boehringer Sohn Ingelheim Neue 5,9-beta-disubstituierte 2-tetrahydrofurfuryl-6,7-benzomorphane, deren saeureadditionssalze, ihre verwendung als arzneimittel und verfahren zu deren herstellung
GB1575009A (en) * 1976-06-21 1980-09-17 Acf Chemiefarma Nv 6,7-benzomorphan derivatives
CN1111900A (zh) * 1993-06-30 1995-11-15 东丽株式会社 止咳药
NZ268969A (en) * 1993-07-23 1997-06-24 Toray Industries Morphinan derivatives and pharmaceutical compositions
US6844438B2 (en) * 2001-08-15 2005-01-18 Mclean Hospital Corporation N-substituted derivatives of morphinan and uses thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE582575A (da) * 1958-09-22
US3647806A (en) * 1966-04-18 1972-03-07 Syntex Corp Tetrahydropyranyl and tetrahydro-furanyl benzomorphan ethers

Also Published As

Publication number Publication date
DK133555C (da) 1976-10-25
US3917606A (en) 1975-11-04
NO137695B (no) 1977-12-27
FI57409C (fi) 1980-08-11
DE2217420C3 (de) 1981-03-12
GB1425347A (en) 1976-02-18
DE2217420B2 (de) 1980-08-07
FI57409B (fi) 1980-04-30
DE2217420A1 (de) 1973-10-31
NO137695C (no) 1978-04-05
DK133555B (da) 1976-06-08

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