SA04250351B1 - مشتقات الأميد او أملاحها المقبولة صيدليا مفيدة كمثبطات لأمراض يسببها السيكتون - Google Patents

مشتقات الأميد او أملاحها المقبولة صيدليا مفيدة كمثبطات لأمراض يسببها السيكتون Download PDF

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Publication number
SA04250351B1
SA04250351B1 SA04250351A SA04250351A SA04250351B1 SA 04250351 B1 SA04250351 B1 SA 04250351B1 SA 04250351 A SA04250351 A SA 04250351A SA 04250351 A SA04250351 A SA 04250351A SA 04250351 B1 SA04250351 B1 SA 04250351B1
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SA
Saudi Arabia
Prior art keywords
cyclopropyl
alkyl
oxoquinazolin
methyl
methylbenzamide
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SA04250351A
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Arabic (ar)
English (en)
Other versions
SA04250351A (ar
Inventor
ديرج سوذرلاند براون
ايان الون ناش
Original Assignee
استرازينيكا ايه بي
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Application filed by استرازينيكا ايه بي filed Critical استرازينيكا ايه بي
Publication of SA04250351A publication Critical patent/SA04250351A/ar
Publication of SA04250351B1 publication Critical patent/SA04250351B1/ar

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms
    • C07D239/91—Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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SA04250351A 2003-10-24 2004-10-23 مشتقات الأميد او أملاحها المقبولة صيدليا مفيدة كمثبطات لأمراض يسببها السيكتون SA04250351B1 (ar)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0324790.5A GB0324790D0 (en) 2003-10-24 2003-10-24 Amide derivatives

Publications (2)

Publication Number Publication Date
SA04250351A SA04250351A (ar) 2005-12-03
SA04250351B1 true SA04250351B1 (ar) 2009-06-01

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SA04250351A SA04250351B1 (ar) 2003-10-24 2004-10-23 مشتقات الأميد او أملاحها المقبولة صيدليا مفيدة كمثبطات لأمراض يسببها السيكتون

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Country Link
US (1) US7750154B2 (enExample)
EP (1) EP1682520B1 (enExample)
JP (1) JP4987478B2 (enExample)
KR (1) KR101127697B1 (enExample)
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UA83867C2 (ru) 2008-08-26
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CA2543351C (en) 2012-09-11
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DE602004031543D1 (de) 2011-04-07
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ATE499347T1 (de) 2011-03-15
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