RU2625800C2 - Способы получения сложных эфиров пинакола и 4-хлор-2 фтор-3- замещенной фенилбороновой кислоты и способы их применения - Google Patents
Способы получения сложных эфиров пинакола и 4-хлор-2 фтор-3- замещенной фенилбороновой кислоты и способы их применения Download PDFInfo
- Publication number
- RU2625800C2 RU2625800C2 RU2014131414A RU2014131414A RU2625800C2 RU 2625800 C2 RU2625800 C2 RU 2625800C2 RU 2014131414 A RU2014131414 A RU 2014131414A RU 2014131414 A RU2014131414 A RU 2014131414A RU 2625800 C2 RU2625800 C2 RU 2625800C2
- Authority
- RU
- Russia
- Prior art keywords
- chloro
- fluoro
- acid
- methoxyphenyl
- methoxyphenylboronic acid
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/79—Acids; Esters
- C07D213/803—Processes of preparation
- C07D213/807—Processes of preparation by oxidation of pyridines or condensed pyridines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F1/00—Compounds containing elements of Groups 1 or 11 of the Periodic Table
- C07F1/02—Lithium compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/04—Esters of boric acids
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Materials Engineering (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161582173P | 2011-12-30 | 2011-12-30 | |
| US61/582,173 | 2011-12-30 | ||
| PCT/US2012/070967 WO2013101665A1 (en) | 2011-12-30 | 2012-12-20 | Methods of forming 4-chloro-2-fluoro-3-substituted-phenylboronic acid pinacol esters and methods of using the same |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| RU2014131414A RU2014131414A (ru) | 2016-02-20 |
| RU2625800C2 true RU2625800C2 (ru) | 2017-07-19 |
Family
ID=48695350
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2014131414A RU2625800C2 (ru) | 2011-12-30 | 2012-12-20 | Способы получения сложных эфиров пинакола и 4-хлор-2 фтор-3- замещенной фенилбороновой кислоты и способы их применения |
Country Status (17)
| Country | Link |
|---|---|
| US (2) | US8912339B2 (https=) |
| EP (1) | EP2797933B1 (https=) |
| JP (2) | JP6290788B2 (https=) |
| KR (1) | KR102062343B1 (https=) |
| CN (1) | CN104114562A (https=) |
| AR (1) | AR089539A1 (https=) |
| AU (1) | AU2012362698B2 (https=) |
| BR (1) | BR112014016048B8 (https=) |
| CA (1) | CA2861631C (https=) |
| CO (1) | CO7020930A2 (https=) |
| IL (1) | IL233413A (https=) |
| IN (1) | IN2014DN05647A (https=) |
| MX (1) | MX341834B (https=) |
| NZ (1) | NZ627041A (https=) |
| PL (1) | PL2797933T3 (https=) |
| RU (1) | RU2625800C2 (https=) |
| WO (1) | WO2013101665A1 (https=) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL2797933T3 (pl) * | 2011-12-30 | 2018-01-31 | Dow Agrosciences Llc | Sposoby wytwarzania estrów pinakolowych kwasu 4-chloro-2-fluoro-3-podstawionego-fenyloboronowego oraz sposoby ich stosowania |
| RU2616621C2 (ru) * | 2011-12-30 | 2017-04-18 | ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи | Способы получения метил 4-амино-3-хлор-6-(4-хлор-2-фтор-3-метоксифенил)пиридин-2-карбоксилата |
| BR102014021960A2 (pt) | 2013-09-05 | 2015-09-15 | Univ Michigan State | métodos para a produção de arenos borilados |
| TW201625354A (zh) | 2014-06-16 | 2016-07-16 | 陶氏農業科學公司 | 用於製備氧硼基化芳烴之方法 |
| BR112017019207A2 (pt) * | 2015-05-22 | 2018-04-24 | Dow Agrosciences Llc | recuperação e/ou reutilização de catalisador de paládio após acoplamento de suzuki |
| CN108558925A (zh) * | 2018-04-16 | 2018-09-21 | 南通纺织丝绸产业技术研究院 | 2,6-二异丙基苯胺基锂在催化酮和硼烷硼氢化反应中的应用 |
| CN108329339A (zh) * | 2018-04-16 | 2018-07-27 | 苏州大学张家港工业技术研究院 | 2,6-二甲基苯胺基锂在催化酮和硼烷硼氢化反应中的应用 |
| CN108654692A (zh) * | 2018-04-16 | 2018-10-16 | 苏州大学 | 正丁基锂在催化酮和硼烷硼氢化反应中的应用 |
| CN108503660A (zh) * | 2018-04-16 | 2018-09-07 | 苏州大学 | 苯胺基锂在催化醛和硼烷硼氢化反应中的应用 |
| CN108383863A (zh) * | 2018-04-16 | 2018-08-10 | 苏州大学 | 2,6-二异丙基苯胺基锂在制备硼酸酯中的应用 |
| CN108503659A (zh) * | 2018-04-16 | 2018-09-07 | 苏州大学 | 利用2,6-二异丙基苯胺基锂制备硼酸酯的方法 |
| CN108373480A (zh) * | 2018-04-16 | 2018-08-07 | 苏州大学 | 利用对甲基苯胺基锂制备硼酸酯的方法 |
| CN108409772A (zh) * | 2018-04-16 | 2018-08-17 | 南通纺织丝绸产业技术研究院 | 基于醛制备硼酸酯的方法 |
| CN108404984A (zh) * | 2018-04-16 | 2018-08-17 | 苏州大学 | 正丁基锂在催化醛和硼烷硼氢化反应中的应用 |
| CN108273550A (zh) * | 2018-04-16 | 2018-07-13 | 苏州大学张家港工业技术研究院 | 对甲基苯胺基锂在催化酮和硼烷硼氢化反应中的应用 |
| CN116715689B (zh) * | 2023-06-09 | 2025-12-12 | 珠海市海瑞德生物科技有限公司 | 氟比洛芬及其中间体的合成方法 |
Citations (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20090182168A1 (en) * | 2008-01-11 | 2009-07-16 | Dow Agrosciences Llc | Process for the selective deprotonation and functionalization of 1-fluoro-2-substituted-3-chlorobenzenes |
| EP2181098B1 (en) * | 2007-08-30 | 2011-03-02 | Dow AgroSciences LLC | 2-(substituted phenyl)-6-amino-5-alkoxy, thioalkoxy and aminoalkyl-4-pyrimidinecarboxylates and their use as herbicides |
| US7915200B2 (en) * | 2007-08-13 | 2011-03-29 | Dow Agrosciences Llc | 2-(2-fluoro-substituted phenyl)-6-amino-5-chloro-4-pyrimidinecarboxylates and their use as herbicides |
| EP2332914A1 (en) * | 2007-10-02 | 2011-06-15 | Dow AgroSciences LLC | Substituted 4-amino-picolinic acids and their use as herbicides |
| US7964758B2 (en) * | 2006-02-13 | 2011-06-21 | Nissan Chemical Industries, Ltd. | Process for production of 2-(substituted phenyl)-3,3,3-trifluoropropene compound |
| RU2428416C2 (ru) * | 2006-01-13 | 2011-09-10 | Дау Агросайенсиз Ллс | 6-(полизамещенный арил)-4-аминопиколинаты и их применение в качестве гербицидов |
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|---|---|---|---|---|
| EP0986541A4 (en) * | 1997-04-09 | 2002-08-14 | Commw Scient Ind Res Org | METHOD FOR COVALENT BINDING ORGANIC COMPOUNDS USING DIBORANE DERIVATIVES |
| EA200702614A1 (ru) * | 2005-05-25 | 2008-04-28 | Майкробиа, Инк. | Способы получения 4-(бифенилил)азетидин-2-оналкилфосфиновых кислот |
| WO2008066921A2 (en) * | 2006-11-30 | 2008-06-05 | Sensors For Medicine And Science, Inc. | Oxidation resistant indicator molecules |
| US8349858B2 (en) * | 2007-06-21 | 2013-01-08 | Merck Sharp & Dohme | Polycyclic guanine derivatives and use thereof |
| HK1200458A1 (en) * | 2011-07-26 | 2015-08-07 | Dow Agrosciences Llc | Methods of isolating 4-chloro-2-fluoro-3-substituted-phenylboronic acids |
| PL2797933T3 (pl) * | 2011-12-30 | 2018-01-31 | Dow Agrosciences Llc | Sposoby wytwarzania estrów pinakolowych kwasu 4-chloro-2-fluoro-3-podstawionego-fenyloboronowego oraz sposoby ich stosowania |
| RU2616621C2 (ru) * | 2011-12-30 | 2017-04-18 | ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи | Способы получения метил 4-амино-3-хлор-6-(4-хлор-2-фтор-3-метоксифенил)пиридин-2-карбоксилата |
-
2012
- 2012-12-20 PL PL12862457T patent/PL2797933T3/pl unknown
- 2012-12-20 WO PCT/US2012/070967 patent/WO2013101665A1/en not_active Ceased
- 2012-12-20 CA CA2861631A patent/CA2861631C/en active Active
- 2012-12-20 KR KR1020147020891A patent/KR102062343B1/ko active Active
- 2012-12-20 JP JP2014550379A patent/JP6290788B2/ja active Active
- 2012-12-20 MX MX2014008017A patent/MX341834B/es active IP Right Grant
- 2012-12-20 CN CN201280069312.7A patent/CN104114562A/zh active Pending
- 2012-12-20 AU AU2012362698A patent/AU2012362698B2/en active Active
- 2012-12-20 EP EP12862457.4A patent/EP2797933B1/en active Active
- 2012-12-20 US US13/722,471 patent/US8912339B2/en active Active
- 2012-12-20 NZ NZ627041A patent/NZ627041A/en unknown
- 2012-12-20 RU RU2014131414A patent/RU2625800C2/ru active
- 2012-12-20 BR BR112014016048A patent/BR112014016048B8/pt active IP Right Grant
- 2012-12-28 AR ARP120105068A patent/AR089539A1/es active IP Right Grant
-
2014
- 2014-06-26 IL IL233413A patent/IL233413A/en active IP Right Grant
- 2014-07-08 IN IN5647DEN2014 patent/IN2014DN05647A/en unknown
- 2014-07-22 CO CO14158850A patent/CO7020930A2/es unknown
- 2014-11-06 US US14/535,096 patent/US9422313B2/en active Active
-
2018
- 2018-02-08 JP JP2018021348A patent/JP2018104447A/ja active Pending
Patent Citations (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2428416C2 (ru) * | 2006-01-13 | 2011-09-10 | Дау Агросайенсиз Ллс | 6-(полизамещенный арил)-4-аминопиколинаты и их применение в качестве гербицидов |
| US7964758B2 (en) * | 2006-02-13 | 2011-06-21 | Nissan Chemical Industries, Ltd. | Process for production of 2-(substituted phenyl)-3,3,3-trifluoropropene compound |
| US7915200B2 (en) * | 2007-08-13 | 2011-03-29 | Dow Agrosciences Llc | 2-(2-fluoro-substituted phenyl)-6-amino-5-chloro-4-pyrimidinecarboxylates and their use as herbicides |
| EP2181098B1 (en) * | 2007-08-30 | 2011-03-02 | Dow AgroSciences LLC | 2-(substituted phenyl)-6-amino-5-alkoxy, thioalkoxy and aminoalkyl-4-pyrimidinecarboxylates and their use as herbicides |
| EP2332914A1 (en) * | 2007-10-02 | 2011-06-15 | Dow AgroSciences LLC | Substituted 4-amino-picolinic acids and their use as herbicides |
| US20090182168A1 (en) * | 2008-01-11 | 2009-07-16 | Dow Agrosciences Llc | Process for the selective deprotonation and functionalization of 1-fluoro-2-substituted-3-chlorobenzenes |
Also Published As
| Publication number | Publication date |
|---|---|
| US8912339B2 (en) | 2014-12-16 |
| BR112014016048B8 (pt) | 2022-10-11 |
| CA2861631C (en) | 2021-05-04 |
| JP6290788B2 (ja) | 2018-03-07 |
| CA2861631A1 (en) | 2013-07-04 |
| US20150203514A1 (en) | 2015-07-23 |
| KR20140117442A (ko) | 2014-10-07 |
| MX2014008017A (es) | 2014-12-08 |
| IL233413A (en) | 2017-12-31 |
| IL233413A0 (en) | 2014-08-31 |
| WO2013101665A1 (en) | 2013-07-04 |
| JP2015507631A (ja) | 2015-03-12 |
| CO7020930A2 (es) | 2014-08-11 |
| AR089539A1 (es) | 2014-08-27 |
| US20130172565A1 (en) | 2013-07-04 |
| BR112014016048A2 (pt) | 2017-06-13 |
| EP2797933B1 (en) | 2017-08-16 |
| BR112014016048B1 (pt) | 2019-12-03 |
| CN104114562A (zh) | 2014-10-22 |
| AU2012362698B2 (en) | 2017-08-24 |
| NZ627041A (en) | 2016-07-29 |
| PL2797933T3 (pl) | 2018-01-31 |
| KR102062343B1 (ko) | 2020-01-02 |
| RU2014131414A (ru) | 2016-02-20 |
| EP2797933A1 (en) | 2014-11-05 |
| JP2018104447A (ja) | 2018-07-05 |
| BR112014016048A8 (pt) | 2017-07-04 |
| MX341834B (es) | 2016-09-05 |
| EP2797933A4 (en) | 2015-08-12 |
| AU2012362698A1 (en) | 2014-07-24 |
| US9422313B2 (en) | 2016-08-23 |
| IN2014DN05647A (https=) | 2015-04-03 |
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