AR089539A1 - Metodos de formacion de esteres pinacolicos de acido 4-cloro-2-fluoro-3-sustituido-fenilboronico y sus metodos de uso - Google Patents
Metodos de formacion de esteres pinacolicos de acido 4-cloro-2-fluoro-3-sustituido-fenilboronico y sus metodos de usoInfo
- Publication number
- AR089539A1 AR089539A1 ARP120105068A ARP120105068A AR089539A1 AR 089539 A1 AR089539 A1 AR 089539A1 AR P120105068 A ARP120105068 A AR P120105068A AR P120105068 A ARP120105068 A AR P120105068A AR 089539 A1 AR089539 A1 AR 089539A1
- Authority
- AR
- Argentina
- Prior art keywords
- substituted
- fluoro
- chloro
- methods
- pinacolic
- Prior art date
Links
- 239000002253 acid Substances 0.000 title abstract 2
- 230000015572 biosynthetic process Effects 0.000 title abstract 2
- -1 4-chloro-2-fluoro-3-substituted-phenylboronic acid Chemical class 0.000 abstract 14
- 150000002148 esters Chemical class 0.000 abstract 3
- IVDFJHOHABJVEH-UHFFFAOYSA-N pinacol Chemical compound CC(C)(O)C(C)(C)O IVDFJHOHABJVEH-UHFFFAOYSA-N 0.000 abstract 2
- QAUCEEIOCLCCFG-UHFFFAOYSA-N trihydroxy borate Chemical compound OOB(OO)OO QAUCEEIOCLCCFG-UHFFFAOYSA-N 0.000 abstract 2
- 150000001642 boronic acid derivatives Chemical class 0.000 abstract 1
- 229910052744 lithium Inorganic materials 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/79—Acids; Esters
- C07D213/803—Processes of preparation
- C07D213/807—Processes of preparation by oxidation of pyridines or condensed pyridines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F1/00—Compounds containing elements of Groups 1 or 11 of the Periodic Table
- C07F1/02—Lithium compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/04—Esters of boric acids
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Materials Engineering (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161582173P | 2011-12-30 | 2011-12-30 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR089539A1 true AR089539A1 (es) | 2014-08-27 |
Family
ID=48695350
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP120105068A AR089539A1 (es) | 2011-12-30 | 2012-12-28 | Metodos de formacion de esteres pinacolicos de acido 4-cloro-2-fluoro-3-sustituido-fenilboronico y sus metodos de uso |
Country Status (17)
| Country | Link |
|---|---|
| US (2) | US8912339B2 (https=) |
| EP (1) | EP2797933B1 (https=) |
| JP (2) | JP6290788B2 (https=) |
| KR (1) | KR102062343B1 (https=) |
| CN (1) | CN104114562A (https=) |
| AR (1) | AR089539A1 (https=) |
| AU (1) | AU2012362698B2 (https=) |
| BR (1) | BR112014016048B8 (https=) |
| CA (1) | CA2861631C (https=) |
| CO (1) | CO7020930A2 (https=) |
| IL (1) | IL233413A (https=) |
| IN (1) | IN2014DN05647A (https=) |
| MX (1) | MX341834B (https=) |
| NZ (1) | NZ627041A (https=) |
| PL (1) | PL2797933T3 (https=) |
| RU (1) | RU2625800C2 (https=) |
| WO (1) | WO2013101665A1 (https=) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL2797933T3 (pl) * | 2011-12-30 | 2018-01-31 | Dow Agrosciences Llc | Sposoby wytwarzania estrów pinakolowych kwasu 4-chloro-2-fluoro-3-podstawionego-fenyloboronowego oraz sposoby ich stosowania |
| RU2616621C2 (ru) * | 2011-12-30 | 2017-04-18 | ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи | Способы получения метил 4-амино-3-хлор-6-(4-хлор-2-фтор-3-метоксифенил)пиридин-2-карбоксилата |
| BR102014021960A2 (pt) | 2013-09-05 | 2015-09-15 | Univ Michigan State | métodos para a produção de arenos borilados |
| TW201625354A (zh) | 2014-06-16 | 2016-07-16 | 陶氏農業科學公司 | 用於製備氧硼基化芳烴之方法 |
| BR112017019207A2 (pt) * | 2015-05-22 | 2018-04-24 | Dow Agrosciences Llc | recuperação e/ou reutilização de catalisador de paládio após acoplamento de suzuki |
| CN108558925A (zh) * | 2018-04-16 | 2018-09-21 | 南通纺织丝绸产业技术研究院 | 2,6-二异丙基苯胺基锂在催化酮和硼烷硼氢化反应中的应用 |
| CN108329339A (zh) * | 2018-04-16 | 2018-07-27 | 苏州大学张家港工业技术研究院 | 2,6-二甲基苯胺基锂在催化酮和硼烷硼氢化反应中的应用 |
| CN108654692A (zh) * | 2018-04-16 | 2018-10-16 | 苏州大学 | 正丁基锂在催化酮和硼烷硼氢化反应中的应用 |
| CN108503660A (zh) * | 2018-04-16 | 2018-09-07 | 苏州大学 | 苯胺基锂在催化醛和硼烷硼氢化反应中的应用 |
| CN108383863A (zh) * | 2018-04-16 | 2018-08-10 | 苏州大学 | 2,6-二异丙基苯胺基锂在制备硼酸酯中的应用 |
| CN108503659A (zh) * | 2018-04-16 | 2018-09-07 | 苏州大学 | 利用2,6-二异丙基苯胺基锂制备硼酸酯的方法 |
| CN108373480A (zh) * | 2018-04-16 | 2018-08-07 | 苏州大学 | 利用对甲基苯胺基锂制备硼酸酯的方法 |
| CN108409772A (zh) * | 2018-04-16 | 2018-08-17 | 南通纺织丝绸产业技术研究院 | 基于醛制备硼酸酯的方法 |
| CN108404984A (zh) * | 2018-04-16 | 2018-08-17 | 苏州大学 | 正丁基锂在催化醛和硼烷硼氢化反应中的应用 |
| CN108273550A (zh) * | 2018-04-16 | 2018-07-13 | 苏州大学张家港工业技术研究院 | 对甲基苯胺基锂在催化酮和硼烷硼氢化反应中的应用 |
| CN116715689B (zh) * | 2023-06-09 | 2025-12-12 | 珠海市海瑞德生物科技有限公司 | 氟比洛芬及其中间体的合成方法 |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0986541A4 (en) * | 1997-04-09 | 2002-08-14 | Commw Scient Ind Res Org | METHOD FOR COVALENT BINDING ORGANIC COMPOUNDS USING DIBORANE DERIVATIVES |
| EA200702614A1 (ru) * | 2005-05-25 | 2008-04-28 | Майкробиа, Инк. | Способы получения 4-(бифенилил)азетидин-2-оналкилфосфиновых кислот |
| EP2060566B1 (en) * | 2006-01-13 | 2016-06-08 | Dow AgroSciences LLC | Poly-substituted aryls |
| US7964758B2 (en) * | 2006-02-13 | 2011-06-21 | Nissan Chemical Industries, Ltd. | Process for production of 2-(substituted phenyl)-3,3,3-trifluoropropene compound |
| WO2008066921A2 (en) * | 2006-11-30 | 2008-06-05 | Sensors For Medicine And Science, Inc. | Oxidation resistant indicator molecules |
| US8349858B2 (en) * | 2007-06-21 | 2013-01-08 | Merck Sharp & Dohme | Polycyclic guanine derivatives and use thereof |
| ES2400405T3 (es) * | 2007-08-13 | 2013-04-09 | Dow Agrosciences Llc | 2-(Fenil 2-fluoro-substituido)-6-amino-5-cloro-4-pirimidinacarboxilatos y su uso como herbicidas |
| MY150491A (en) | 2007-08-30 | 2014-01-30 | Dow Agrosciences Llc | 2-(substituted phenyl)-6-amino-5-alkoxy, thioalkoxy and aminoalkyl 4- pyrimidinecarboxylates and their use as herbicides |
| CA2699598C (en) * | 2007-10-02 | 2013-05-21 | Dow Agrosciences Llc | 2-substituted-6-amino-5-alkyl, alkenyl or alkynyl-4-pyrimidinecarboxylic acids and 6-substituted-4-amino-3-alkyl, alkenyl or alkynyl picolinic acids and their use as herbicides |
| UA104282C2 (ru) * | 2008-01-11 | 2014-01-27 | ДАУ АГРОСАЙЕНСИЗ ЕлЕлСи | Способ селективного депротонирования и введения заместителя к 1-фтор-2-замещенным-3-хлорбензолам |
| HK1200458A1 (en) * | 2011-07-26 | 2015-08-07 | Dow Agrosciences Llc | Methods of isolating 4-chloro-2-fluoro-3-substituted-phenylboronic acids |
| PL2797933T3 (pl) * | 2011-12-30 | 2018-01-31 | Dow Agrosciences Llc | Sposoby wytwarzania estrów pinakolowych kwasu 4-chloro-2-fluoro-3-podstawionego-fenyloboronowego oraz sposoby ich stosowania |
| RU2616621C2 (ru) * | 2011-12-30 | 2017-04-18 | ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи | Способы получения метил 4-амино-3-хлор-6-(4-хлор-2-фтор-3-метоксифенил)пиридин-2-карбоксилата |
-
2012
- 2012-12-20 PL PL12862457T patent/PL2797933T3/pl unknown
- 2012-12-20 WO PCT/US2012/070967 patent/WO2013101665A1/en not_active Ceased
- 2012-12-20 CA CA2861631A patent/CA2861631C/en active Active
- 2012-12-20 KR KR1020147020891A patent/KR102062343B1/ko active Active
- 2012-12-20 JP JP2014550379A patent/JP6290788B2/ja active Active
- 2012-12-20 MX MX2014008017A patent/MX341834B/es active IP Right Grant
- 2012-12-20 CN CN201280069312.7A patent/CN104114562A/zh active Pending
- 2012-12-20 AU AU2012362698A patent/AU2012362698B2/en active Active
- 2012-12-20 EP EP12862457.4A patent/EP2797933B1/en active Active
- 2012-12-20 US US13/722,471 patent/US8912339B2/en active Active
- 2012-12-20 NZ NZ627041A patent/NZ627041A/en unknown
- 2012-12-20 RU RU2014131414A patent/RU2625800C2/ru active
- 2012-12-20 BR BR112014016048A patent/BR112014016048B8/pt active IP Right Grant
- 2012-12-28 AR ARP120105068A patent/AR089539A1/es active IP Right Grant
-
2014
- 2014-06-26 IL IL233413A patent/IL233413A/en active IP Right Grant
- 2014-07-08 IN IN5647DEN2014 patent/IN2014DN05647A/en unknown
- 2014-07-22 CO CO14158850A patent/CO7020930A2/es unknown
- 2014-11-06 US US14/535,096 patent/US9422313B2/en active Active
-
2018
- 2018-02-08 JP JP2018021348A patent/JP2018104447A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| US8912339B2 (en) | 2014-12-16 |
| BR112014016048B8 (pt) | 2022-10-11 |
| CA2861631C (en) | 2021-05-04 |
| JP6290788B2 (ja) | 2018-03-07 |
| CA2861631A1 (en) | 2013-07-04 |
| US20150203514A1 (en) | 2015-07-23 |
| KR20140117442A (ko) | 2014-10-07 |
| MX2014008017A (es) | 2014-12-08 |
| IL233413A (en) | 2017-12-31 |
| IL233413A0 (en) | 2014-08-31 |
| RU2625800C2 (ru) | 2017-07-19 |
| WO2013101665A1 (en) | 2013-07-04 |
| JP2015507631A (ja) | 2015-03-12 |
| CO7020930A2 (es) | 2014-08-11 |
| US20130172565A1 (en) | 2013-07-04 |
| BR112014016048A2 (pt) | 2017-06-13 |
| EP2797933B1 (en) | 2017-08-16 |
| BR112014016048B1 (pt) | 2019-12-03 |
| CN104114562A (zh) | 2014-10-22 |
| AU2012362698B2 (en) | 2017-08-24 |
| NZ627041A (en) | 2016-07-29 |
| PL2797933T3 (pl) | 2018-01-31 |
| KR102062343B1 (ko) | 2020-01-02 |
| RU2014131414A (ru) | 2016-02-20 |
| EP2797933A1 (en) | 2014-11-05 |
| JP2018104447A (ja) | 2018-07-05 |
| BR112014016048A8 (pt) | 2017-07-04 |
| MX341834B (es) | 2016-09-05 |
| EP2797933A4 (en) | 2015-08-12 |
| AU2012362698A1 (en) | 2014-07-24 |
| US9422313B2 (en) | 2016-08-23 |
| IN2014DN05647A (https=) | 2015-04-03 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant, registration |