RU2573392C3 - Композиция, содержащая тетрациклические соединения - Google Patents

Композиция, содержащая тетрациклические соединения

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Publication number
RU2573392C3
RU2573392C3 RU2013112011A RU2013112011A RU2573392C3 RU 2573392 C3 RU2573392 C3 RU 2573392C3 RU 2013112011 A RU2013112011 A RU 2013112011A RU 2013112011 A RU2013112011 A RU 2013112011A RU 2573392 C3 RU2573392 C3 RU 2573392C3
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RU
Russia
Prior art keywords
composition containing
tetracyclic compounds
containing tetracyclic
dissolution aid
compounds
Prior art date
Application number
RU2013112011A
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English (en)
Other versions
RU2013112011A (ru
RU2573392C2 (ru
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Чугаи Сейяку Кабусики Кайся
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45605249&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=RU2573392(C3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Чугаи Сейяку Кабусики Кайся filed Critical Чугаи Сейяку Кабусики Кайся
Publication of RU2013112011A publication Critical patent/RU2013112011A/ru
Application granted granted Critical
Publication of RU2573392C2 publication Critical patent/RU2573392C2/ru
Publication of RU2573392C3 publication Critical patent/RU2573392C3/ru

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A—HUMAN NECESSITIES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
    • A—HUMAN NECESSITIES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/381—Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
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    • A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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    • A61K47/20—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing sulfur, e.g. dimethyl sulfoxide [DMSO], docusate, sodium lauryl sulfate or aminosulfonic acids
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    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
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    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Claims (1)

  1. Фармацевтическая композиция, предназначенная для предотвращения и/или лечения рака, содержащая 9-этил-6,6-диметил-8-(4-морфолин-4-илпиперидин-1-ил)-11-оксо-6,11-дигидро-5Н-бензо[b]карбазол-3-карбонитрил или его соль, фармацевтически приемлемый носитель и средство, способствующее растворению, где указанное средство, способствующее растворению, представляет собой гидроксипропилцеллюлозу.
RU2013112011A 2010-08-20 2011-08-19 Композиция, содержащая тетрациклические соединения RU2573392C3 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2010185385 2010-08-20
JP2010-185385 2010-08-20
PCT/JP2011/068735 WO2012023597A1 (ja) 2010-08-20 2011-08-19 ４環性化合物を含む組成物

Publications (3)

Publication Number Publication Date
RU2013112011A RU2013112011A (ru) 2014-09-27
RU2573392C2 RU2573392C2 (ru) 2016-01-20
RU2573392C3 true RU2573392C3 (ru) 2021-06-24

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US (4) US9365514B2 (ru)
EP (2) EP3698788A1 (ru)
JP (1) JP4918630B1 (ru)
KR (1) KR101362589B1 (ru)
CN (1) CN103052386B (ru)
AR (2) AR083246A1 (ru)
AU (1) AU2011291708B2 (ru)
BR (1) BR112013003879B1 (ru)
CA (1) CA2808210C (ru)
ES (1) ES2769550T3 (ru)
HK (1) HK1179878A1 (ru)
IL (1) IL223892B (ru)
MX (1) MX355836B (ru)
MY (1) MY160110A (ru)
NZ (1) NZ608312A (ru)
PL (1) PL2606886T3 (ru)
RU (1) RU2573392C3 (ru)
SG (1) SG187614A1 (ru)
TW (1) TWI526441B (ru)
WO (1) WO2012023597A1 (ru)
ZA (1) ZA201300020B (ru)

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LT2975024T (lt) * 2009-06-10 2018-06-11 Chugai Seiyaku Kabushiki Kaisha Tetraciklininiai junginiai
SG187614A1 (en) 2010-08-20 2013-03-28 Chugai Pharmaceutical Co Ltd Composition containing tetracyclic compound
EP2902029B1 (en) 2012-09-25 2018-08-08 Chugai Seiyaku Kabushiki Kaisha Ret inhibitor
CN104109168B (zh) * 2013-04-20 2017-02-15 山东轩竹医药科技有限公司 四并环激酶抑制剂
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