RU2016110852A3 - - Google Patents

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RU2016110852A3
RU2016110852A3 RU2016110852A RU2016110852A RU2016110852A3 RU 2016110852 A3 RU2016110852 A3 RU 2016110852A3 RU 2016110852 A RU2016110852 A RU 2016110852A RU 2016110852 A RU2016110852 A RU 2016110852A RU 2016110852 A3 RU2016110852 A3 RU 2016110852A3
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RU2016110852A
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
  • Immunology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Hematology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pulmonology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Cardiology (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Obesity (AREA)
  • Epidemiology (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Oncology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Communicable Diseases (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Child & Adolescent Psychology (AREA)
  • Psychiatry (AREA)
RU2016110852A 2013-09-27 2014-09-25 Ингибиторы irak и их применения RU2016110852A (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361883497P 2013-09-27 2013-09-27
US61/883,497 2013-09-27
PCT/US2014/057444 WO2015048281A1 (en) 2013-09-27 2014-09-25 Irak inhibitors and uses thereof

Publications (2)

Publication Number Publication Date
RU2016110852A RU2016110852A (ru) 2017-10-30
RU2016110852A3 true RU2016110852A3 (enExample) 2018-06-25

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RU2016110852A RU2016110852A (ru) 2013-09-27 2014-09-25 Ингибиторы irak и их применения

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US (2) US9518065B2 (enExample)
EP (1) EP3049086A4 (enExample)
JP (1) JP2016531870A (enExample)
KR (1) KR20160092991A (enExample)
CN (1) CN106232122A (enExample)
BR (1) BR112016006319A2 (enExample)
CA (1) CA2925211A1 (enExample)
MX (1) MX2016003843A (enExample)
RU (1) RU2016110852A (enExample)
TW (1) TW201522349A (enExample)
WO (1) WO2015048281A1 (enExample)

Families Citing this family (40)

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Publication number Priority date Publication date Assignee Title
WO2017004133A1 (en) * 2015-06-29 2017-01-05 Nimbus Iris, Inc. Irak inhibitors and uses thereof
DK3331877T3 (da) 2015-08-04 2022-01-03 Yissum Res Dev Co Of Hebrew Univ Jerusalem Ltd Pyrazolpyrimidinderivat og anvendelser deraf
EP3331879B1 (en) 2015-08-04 2020-05-20 Rigel Pharmaceuticals, Inc. Benzazole compounds and methods for making and using the compounds
JP6541871B2 (ja) 2015-08-13 2019-07-10 北京韓美薬品有限公司 Ｉｒａｋ４阻害剤、及びその応用
CN107531725B (zh) * 2015-08-13 2021-03-19 北京韩美药品有限公司 Irak4抑制剂及其应用
GB201518456D0 (en) * 2015-10-19 2015-12-02 Galapagos Nv Novel compounds and pharmaceutical compositions thereof for the treatment of inflammatory, autoimmune and/or proliferative diseases
SG10201508795XA (en) * 2015-10-23 2017-05-30 Agency Science Tech & Res Method for treating cancer
WO2017205762A1 (en) * 2016-05-27 2017-11-30 Pharmacyclics Llc Inhibitors of interleukin-1 receptor-associated kinase
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BR112016006319A2 (pt) 2017-08-01
US20170035766A1 (en) 2017-02-09
WO2015048281A1 (en) 2015-04-02
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