RU2011103475A - Новая возможность борьбы с гиардиазом - Google Patents
Новая возможность борьбы с гиардиазом Download PDFInfo
- Publication number
- RU2011103475A RU2011103475A RU2011103475/15A RU2011103475A RU2011103475A RU 2011103475 A RU2011103475 A RU 2011103475A RU 2011103475/15 A RU2011103475/15 A RU 2011103475/15A RU 2011103475 A RU2011103475 A RU 2011103475A RU 2011103475 A RU2011103475 A RU 2011103475A
- Authority
- RU
- Russia
- Prior art keywords
- giardiasis
- combat
- nifurtimox
- new possibility
- anthelmintic
- Prior art date
Links
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/541—Non-condensed thiazines containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/15—Depsipeptides; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Abstract
1. Применение нифуртимокса для получения лекарственных средств для лечения болезней, вызванных гиардиями. !2. Применение по п.1 для лечения болезней, вызванных Giardia lamblia. ! 3. Средство, содержащее нифуртимокс и противоглистный препарат. ! 4. Средство, содержащее нифуртимокс и противоглистный циклооктадепсипептид.
Claims (4)
1. Применение нифуртимокса для получения лекарственных средств для лечения болезней, вызванных гиардиями.
2. Применение по п.1 для лечения болезней, вызванных Giardia lamblia.
3. Средство, содержащее нифуртимокс и противоглистный препарат.
4. Средство, содержащее нифуртимокс и противоглистный циклооктадепсипептид.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE102008031284.3 | 2008-07-02 | ||
DE102008031284A DE102008031284A1 (de) | 2008-07-02 | 2008-07-02 | Neue Bekämpfungsmöglichkeit der Giardiose |
PCT/EP2009/004475 WO2010000399A1 (de) | 2008-07-02 | 2009-06-20 | Verwendung von nifurtimox zur behandlung der giardiose |
Publications (3)
Publication Number | Publication Date |
---|---|
RU2011103475A true RU2011103475A (ru) | 2012-08-10 |
RU2538713C2 RU2538713C2 (ru) | 2015-01-10 |
RU2538713C9 RU2538713C9 (ru) | 2015-08-20 |
Family
ID=41077987
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RU2011103475/15A RU2538713C9 (ru) | 2008-07-02 | 2009-06-20 | Новая возможность борьбы с гиардиазом |
Country Status (30)
Country | Link |
---|---|
US (1) | US8440612B2 (ru) |
EP (1) | EP2310018B1 (ru) |
JP (1) | JP5627579B2 (ru) |
KR (1) | KR101720805B1 (ru) |
CN (1) | CN102083441B (ru) |
AR (1) | AR072425A1 (ru) |
AU (1) | AU2009266125B2 (ru) |
BR (1) | BRPI0913889B1 (ru) |
CA (1) | CA2729730C (ru) |
CL (2) | CL2010001577A1 (ru) |
CO (1) | CO6321270A2 (ru) |
CR (1) | CR20110022A (ru) |
DE (1) | DE102008031284A1 (ru) |
DK (1) | DK2310018T3 (ru) |
DO (1) | DOP2010000405A (ru) |
EC (1) | ECSP10010720A (ru) |
ES (1) | ES2444581T3 (ru) |
HK (1) | HK1158113A1 (ru) |
IL (1) | IL209698A (ru) |
MX (1) | MX2010014446A (ru) |
MY (1) | MY157007A (ru) |
NI (1) | NI201100008A (ru) |
NZ (1) | NZ590276A (ru) |
PE (1) | PE20110283A1 (ru) |
PL (1) | PL2310018T3 (ru) |
RU (1) | RU2538713C9 (ru) |
SV (1) | SV2011003785A (ru) |
UA (1) | UA103328C2 (ru) |
WO (1) | WO2010000399A1 (ru) |
ZA (1) | ZA201009225B (ru) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2814694C (en) * | 2010-10-12 | 2019-01-29 | The United States Of America, As Represented By The Secretary, Department Of Health And Human Services | Methods of treating giardiasis |
SG10202103403SA (en) | 2015-05-20 | 2021-05-28 | Boehringer Ingelheim Animal Health Usa Inc | Anthelmintic depsipeptide compounds |
CN108699052B (zh) | 2015-12-28 | 2022-04-29 | 勃林格殷格翰动物保健美国公司 | 驱虫缩酚酸肽化合物 |
CA3044038A1 (en) | 2016-11-16 | 2018-05-24 | Boehringer Ingelheim Animal Health USA Inc. | Anthelmintic depsipeptide compounds |
EP3750527A1 (en) * | 2019-06-13 | 2020-12-16 | Bayer AG | Stable tablet formulation of nifurtimox and process for producing the same |
CN114377018B (zh) * | 2020-10-21 | 2024-02-06 | 中国医学科学院药物研究所 | 硝呋莫司在制备抗流感病毒药物中的应用 |
Family Cites Families (22)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1170957B (de) * | 1962-11-23 | 1964-05-27 | Bayer Ag | Verfahren zur Herstellung von 5-Nitro-furfuryliden-(2)-iminoderivaten |
JPH081908B2 (ja) * | 1987-07-22 | 1996-01-10 | 三菱電機株式会社 | 超格子半導体素子 |
NO176766C (no) | 1989-02-07 | 1995-05-24 | Meiji Seika Kaisha | Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet |
ATE211466T1 (de) | 1992-03-17 | 2002-01-15 | Fujisawa Pharmaceutical Co | Depsipeptide, herstellung und anwendung |
DE4317458A1 (de) | 1992-06-11 | 1993-12-16 | Bayer Ag | Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung |
AU695021B2 (en) | 1993-02-19 | 1998-08-06 | Meiji Seika Kaisha Ltd. | PF1022 derivative cyclic depsipeptide |
DE4317457A1 (de) | 1993-05-26 | 1994-12-01 | Bayer Ag | Octacyclodepsipeptide mit endoparasitizider Wirkung |
DE4317432A1 (de) | 1993-05-26 | 1994-12-01 | Bayer Ag | Octacyclodepsipeptide mit endoparasitizider Wirkung |
CA2171088A1 (en) | 1993-09-06 | 1995-03-16 | Hitoshi Nishiyama | Cyclodepsipeptide compound |
DE4401389A1 (de) | 1994-01-19 | 1995-07-20 | Bayer Ag | Verwendung von cyclischen Depsipeptiden mit 12 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 12 Ringatomen und Verfahren zu ihrer Herstellung |
DE4406025A1 (de) | 1994-02-24 | 1995-08-31 | Bayer Ag | Milchsäure-haltige cyclische Depsipeptide mit 18 Ringatomen als endoparasitizide Mittel und Verfahren zu ihrer Herstellung |
RU2074038C1 (ru) * | 1994-06-16 | 1997-02-27 | Товарищество с ограниченной ответственностью Предприятие "ТЕПАРК" | Способ изготовления полых металлических емкостей |
DE4437198A1 (de) | 1994-10-18 | 1996-04-25 | Bayer Ag | Verfahren zur Sulfonylierung, Sulfenylierung und Phosphorylierung von cyclischen Depsipeptiden |
ATE425973T1 (de) | 1995-06-30 | 2009-04-15 | Astellas Pharma Inc | Depsipeptid-derivat, verfahren zu dessen herstellung und zwischenprodukt dafur |
CZ295705B6 (cs) | 1995-09-22 | 2005-10-12 | Bayer Aktiengesellschaft | Cyklodepsipeptidové deriváty sloučeniny PF1022 a farmaceutický prostředek s jejich obsahem |
DE19545639A1 (de) | 1995-12-07 | 1997-06-12 | Bayer Ag | Verfahren zur Herstellung von substituierten Arylmilchsäure-haltigen Cyclodepsipeptiden mit 24 Ringatomen |
US6503881B2 (en) * | 1996-08-21 | 2003-01-07 | Micrologix Biotech Inc. | Compositions and methods for treating infections using cationic peptides alone or in combination with antibiotics |
US5874630A (en) * | 1998-01-06 | 1999-02-23 | Occidental Chemical Corporation | Synthesis of mercaptans from alcohols |
US6133228A (en) * | 1998-05-28 | 2000-10-17 | Firmenich Sa | Slow release of fragrant compounds in perfumery using 2-benzoyl benzoates, 2-alkanoyl benzoates or α-keto esters |
DE19828047A1 (de) * | 1998-06-24 | 1999-12-30 | Bayer Ag | Substituierte Cyclooctadepsipeptide |
CA2586950A1 (en) * | 2004-11-12 | 2006-05-18 | Celgene Corporation | Methods and compositions using immunomodulatory compounds for treatment and management of parasitic diseases |
DE102005033496A1 (de) | 2005-07-19 | 2007-01-25 | Bayer Healthcare Ag | Desinfektionsmittel |
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2008
- 2008-07-02 DE DE102008031284A patent/DE102008031284A1/de not_active Withdrawn
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2009
- 2009-06-20 US US13/000,715 patent/US8440612B2/en not_active Expired - Fee Related
- 2009-06-20 CN CN2009801255081A patent/CN102083441B/zh not_active Expired - Fee Related
- 2009-06-20 ES ES09772099.9T patent/ES2444581T3/es active Active
- 2009-06-20 WO PCT/EP2009/004475 patent/WO2010000399A1/de active Application Filing
- 2009-06-20 CA CA2729730A patent/CA2729730C/en not_active Expired - Fee Related
- 2009-06-20 RU RU2011103475/15A patent/RU2538713C9/ru not_active IP Right Cessation
- 2009-06-20 EP EP09772099.9A patent/EP2310018B1/de not_active Not-in-force
- 2009-06-20 MX MX2010014446A patent/MX2010014446A/es active IP Right Grant
- 2009-06-20 BR BRPI0913889A patent/BRPI0913889B1/pt not_active IP Right Cessation
- 2009-06-20 NZ NZ590276A patent/NZ590276A/xx not_active IP Right Cessation
- 2009-06-20 MY MYPI2010006319A patent/MY157007A/en unknown
- 2009-06-20 JP JP2011515179A patent/JP5627579B2/ja not_active Expired - Fee Related
- 2009-06-20 AU AU2009266125A patent/AU2009266125B2/en not_active Ceased
- 2009-06-20 UA UAA201101135A patent/UA103328C2/ru unknown
- 2009-06-20 DK DK09772099.9T patent/DK2310018T3/da active
- 2009-06-20 PE PE2010001201A patent/PE20110283A1/es not_active Application Discontinuation
- 2009-06-20 PL PL09772099T patent/PL2310018T3/pl unknown
- 2009-06-20 KR KR1020117002111A patent/KR101720805B1/ko active IP Right Grant
- 2009-06-30 AR ARP090102439A patent/AR072425A1/es not_active Application Discontinuation
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2010
- 2010-12-01 IL IL209698A patent/IL209698A/en active IP Right Grant
- 2010-12-22 ZA ZA2010/09225A patent/ZA201009225B/en unknown
- 2010-12-27 CL CL2010001577A patent/CL2010001577A1/es unknown
- 2010-12-27 EC EC2010010720A patent/ECSP10010720A/es unknown
- 2010-12-27 CO CO10162857A patent/CO6321270A2/es active IP Right Grant
- 2010-12-27 DO DO2010000405A patent/DOP2010000405A/es unknown
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2011
- 2011-01-03 SV SV2011003785A patent/SV2011003785A/es active IP Right Grant
- 2011-01-05 NI NI201100008A patent/NI201100008A/es unknown
- 2011-01-11 CR CR20110022A patent/CR20110022A/es unknown
- 2011-11-25 HK HK11112838.8A patent/HK1158113A1/xx not_active IP Right Cessation
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2013
- 2013-03-15 CL CL2013000709A patent/CL2013000709A1/es unknown
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TH4A | Reissue of patent specification | ||
MM4A | The patent is invalid due to non-payment of fees |
Effective date: 20200621 |