EA201001330A1 - Соединения и композиции в качестве модуляторов активности gpr119 - Google Patents

Соединения и композиции в качестве модуляторов активности gpr119

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Publication number
EA201001330A1
EA201001330A1 EA201001330A EA201001330A EA201001330A1 EA 201001330 A1 EA201001330 A1 EA 201001330A1 EA 201001330 A EA201001330 A EA 201001330A EA 201001330 A EA201001330 A EA 201001330A EA 201001330 A1 EA201001330 A1 EA 201001330A1
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EA
Eurasian Patent Office
Prior art keywords
compounds
compositions
gpr119 activity
activity modulators
gpr119
Prior art date
Application number
EA201001330A
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English (en)
Inventor
Филлип Алпер
Роберт Эппле
Пьер-Ив Мишелли
Даниел Мутник
Виктор Никулин
Майкл Дж. Петрасси Х.
Original Assignee
Айрм Ллк
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Publication date
Application filed by Айрм Ллк filed Critical Айрм Ллк
Publication of EA201001330A1 publication Critical patent/EA201001330A1/ru

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Abstract

В заявке описаны соединения, фармацевтические композиции, содержащие такие соединения, и способы применения таких соединений для лечения или предупреждения заболеваний или нарушений, связанных с активностью GPR119.
EA201001330A 2008-02-22 2009-02-20 Соединения и композиции в качестве модуляторов активности gpr119 EA201001330A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US3089708P 2008-02-22 2008-02-22
PCT/US2009/034789 WO2009105722A1 (en) 2008-02-22 2009-02-20 Compounds and compositions as modulators of gpr119 activity

Publications (1)

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EA201001330A1 true EA201001330A1 (ru) 2011-04-29

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EA201001330A EA201001330A1 (ru) 2008-02-22 2009-02-20 Соединения и композиции в качестве модуляторов активности gpr119

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Country Link
US (1) US20110172244A1 (ru)
EP (1) EP2252586A1 (ru)
JP (1) JP2011513234A (ru)
CN (1) CN102007100A (ru)
AU (1) AU2009217282A1 (ru)
BR (1) BRPI0908851A2 (ru)
CA (1) CA2716332A1 (ru)
EA (1) EA201001330A1 (ru)
MX (1) MX2010009203A (ru)
WO (1) WO2009105722A1 (ru)

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TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
WO2013045413A1 (en) 2011-09-27 2013-04-04 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
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AU2021405511A1 (en) * 2020-12-22 2023-06-22 Luxembourg Institute Of Health (Lih) Conolidine analogues as selective ackr3 modulators for the treatment of cancer and cardiovascular diseases

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Publication number Publication date
WO2009105722A1 (en) 2009-08-27
CN102007100A (zh) 2011-04-06
BRPI0908851A2 (pt) 2017-05-30
EP2252586A1 (en) 2010-11-24
MX2010009203A (es) 2010-11-10
US20110172244A1 (en) 2011-07-14
AU2009217282A1 (en) 2009-08-27
JP2011513234A (ja) 2011-04-28
CA2716332A1 (en) 2009-08-27

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