RU2009105196A - Противовирусные соединения (варианты), фармацевтическая композиция на их основе, названные соединения для изготовления лекарственного средства, способ лечения или профилактики вирусной инфекции с их помощью - Google Patents

Противовирусные соединения (варианты), фармацевтическая композиция на их основе, названные соединения для изготовления лекарственного средства, способ лечения или профилактики вирусной инфекции с их помощью Download PDF

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Publication number
RU2009105196A
RU2009105196A RU2009105196/04A RU2009105196A RU2009105196A RU 2009105196 A RU2009105196 A RU 2009105196A RU 2009105196/04 A RU2009105196/04 A RU 2009105196/04A RU 2009105196 A RU2009105196 A RU 2009105196A RU 2009105196 A RU2009105196 A RU 2009105196A
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RU
Russia
Prior art keywords
substituted
carbonylmethyl
methyl
amino
group
Prior art date
Application number
RU2009105196/04A
Other languages
English (en)
Russian (ru)
Inventor
Януш БОТЯНСКИ (HU)
Януш БОТЯНСКИ
Рональд Конрад ГРИФФИТ (US)
Рональд Конрад Гриффит
Сон Мин ПХАМ (US)
Сон Мин ПХАМ
Кристофер Дон РОБЕРТС (US)
Кристофер Дон Робертс
Фрвнц Ульрих ШМИЦ (DE)
Фрвнц Ульрих ШМИЦ
Original Assignee
СмитКлайн Бичэм Конэрейшн (US)
СмитКлайн Бичэм Конэрейшн
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by СмитКлайн Бичэм Конэрейшн (US), СмитКлайн Бичэм Конэрейшн filed Critical СмитКлайн Бичэм Конэрейшн (US)
Publication of RU2009105196A publication Critical patent/RU2009105196A/ru

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Virology (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
RU2009105196/04A 2006-07-14 2007-07-12 Противовирусные соединения (варианты), фармацевтическая композиция на их основе, названные соединения для изготовления лекарственного средства, способ лечения или профилактики вирусной инфекции с их помощью RU2009105196A (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US83104006P 2006-07-14 2006-07-14
US60/831,040 2006-07-14

Publications (1)

Publication Number Publication Date
RU2009105196A true RU2009105196A (ru) 2010-08-27

Family

ID=38742551

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2009105196/04A RU2009105196A (ru) 2006-07-14 2007-07-12 Противовирусные соединения (варианты), фармацевтическая композиция на их основе, названные соединения для изготовления лекарственного средства, способ лечения или профилактики вирусной инфекции с их помощью

Country Status (13)

Country Link
EP (1) EP2044083A1 (ko)
JP (1) JP2009543807A (ko)
KR (1) KR20090033881A (ko)
CN (1) CN101490058A (ko)
AR (1) AR062258A1 (ko)
AU (1) AU2007272441A1 (ko)
BR (1) BRPI0714346A2 (ko)
CA (1) CA2657651A1 (ko)
MX (1) MX2009000513A (ko)
PE (1) PE20080427A1 (ko)
RU (1) RU2009105196A (ko)
TW (1) TW200813070A (ko)
WO (2) WO2008008907A2 (ko)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9108983B2 (en) 2013-07-23 2015-08-18 Les Laboratoires Servier Pyrrole compounds, a process for their preparation and pharmaceutical compositions containing them

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20070049593A1 (en) 2004-02-24 2007-03-01 Japan Tobacco Inc. Tetracyclic fused heterocyclic compound and use thereof as HCV polymerase inhibitor
US7659263B2 (en) 2004-11-12 2010-02-09 Japan Tobacco Inc. Thienopyrrole compound and use thereof as HCV polymerase inhibitor
ATE548044T1 (de) 2007-05-04 2012-03-15 Vertex Pharma Kombinationstherapie zur behandlung von hiv- infektionen
MX2012006877A (es) 2009-12-18 2012-08-31 Idenix Pharmaceuticals Inc Inhibidores de virus de hepatitis c de arileno o heteroarileno 5, 5 - fusionado.
WO2012087833A1 (en) * 2010-12-22 2012-06-28 Abbott Laboratories Hepatitis c inhibitors and uses thereof
US20120252721A1 (en) * 2011-03-31 2012-10-04 Idenix Pharmaceuticals, Inc. Methods for treating drug-resistant hepatitis c virus infection with a 5,5-fused arylene or heteroarylene hepatitis c virus inhibitor
RU2546006C1 (ru) 2014-03-07 2015-04-10 Римма Ильинична Ашкинази Противовирусное средство
WO2016118043A1 (ru) 2015-01-20 2016-07-28 Виктор Вениаминович ТЕЦ Гемостатическое средство
US10167293B2 (en) * 2016-05-26 2019-01-01 Bayer Pharma Aktiengesellschaft [8-(phenylsulfonyl)-3,8-diazabicyclo[3.2.1]oct-3-yl](1H-1,2,3-triazol-4-yl)methanones
US11285170B2 (en) 2017-05-24 2022-03-29 Viktor Veniaminovich Tets Fractionated antimicrobial compositions and use thereof
MX2023012110A (es) * 2021-04-16 2023-10-24 Gilead Sciences Inc Compuestos de tienopirrol.
CN117957234A (zh) 2021-09-10 2024-04-30 吉利德科学公司 噻吩并吡咯化合物

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1401825E (pt) * 2001-06-11 2009-10-23 Virochem Pharma Inc Compostos e métodos para o tratamento ou para a prevenção de infecções com flavivírus
RU2375350C2 (ru) * 2003-06-04 2009-12-10 Смитклайн Бичам Корпорейшн Азотсодержащие производные гетероарила

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9108983B2 (en) 2013-07-23 2015-08-18 Les Laboratoires Servier Pyrrole compounds, a process for their preparation and pharmaceutical compositions containing them
EA026906B1 (ru) * 2013-07-23 2017-05-31 Ле Лаборатуар Сервье Новые пиррольные соединения, способ их получения и фармацевтические композиции, содержащие их
US10688101B2 (en) 2013-07-23 2020-06-23 Les Laboratories Servier Pyrrole compounds, a process for their preparation and pharmaceutical compositions containing them
US11058689B2 (en) 2013-07-23 2021-07-13 Les Laboratoires Servier Pyrrole compounds, a process for their preparation and pharmaceutical

Also Published As

Publication number Publication date
AU2007272441A1 (en) 2008-01-17
BRPI0714346A2 (pt) 2013-03-19
WO2008008912A1 (en) 2008-01-17
EP2044083A1 (en) 2009-04-08
WO2008008907A2 (en) 2008-01-17
WO2008008907A3 (en) 2008-03-20
AU2007272441A2 (en) 2009-03-19
CA2657651A1 (en) 2008-01-17
AR062258A1 (es) 2008-10-29
MX2009000513A (es) 2009-03-09
TW200813070A (en) 2008-03-16
KR20090033881A (ko) 2009-04-06
CN101490058A (zh) 2009-07-22
JP2009543807A (ja) 2009-12-10
PE20080427A1 (es) 2008-06-11

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Effective date: 20110301