RU2007143383A - Клейкие лекарственные формы - Google Patents

Клейкие лекарственные формы Download PDF

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Publication number
RU2007143383A
RU2007143383A RU2007143383/15A RU2007143383A RU2007143383A RU 2007143383 A RU2007143383 A RU 2007143383A RU 2007143383/15 A RU2007143383/15 A RU 2007143383/15A RU 2007143383 A RU2007143383 A RU 2007143383A RU 2007143383 A RU2007143383 A RU 2007143383A
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Russia
Prior art keywords
adhesive
dosage form
form according
film
backing
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RU2007143383/15A
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English (en)
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RU2446790C2 (ru
Inventor
Йосихиро ИВАО (JP)
Йосихиро ИВАО
Кацуюки ОКУБО (JP)
Кацуюки ОКУБО
Кацухиро ОКАДА (JP)
Кацухиро ОКАДА
Кенсуке МАЦУОКА (JP)
Кенсуке МАЦУОКА
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Нитто Денко Корпорейшн (Jp)
Нитто Денко Корпорейшн
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Publication of RU2007143383A publication Critical patent/RU2007143383A/ru
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7053Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7053Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
    • A61K9/7061Polyacrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7069Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained otherwise than by reactions only involving carbon to carbon unsaturated bonds, e.g. polysiloxane, polyesters, polyurethane, polyethylene oxide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61LMETHODS OR APPARATUS FOR STERILISING MATERIALS OR OBJECTS IN GENERAL; DISINFECTION, STERILISATION OR DEODORISATION OF AIR; CHEMICAL ASPECTS OF BANDAGES, DRESSINGS, ABSORBENT PADS OR SURGICAL ARTICLES; MATERIALS FOR BANDAGES, DRESSINGS, ABSORBENT PADS OR SURGICAL ARTICLES
    • A61L15/00Chemical aspects of, or use of materials for, bandages, dressings or absorbent pads
    • A61L15/16Bandages, dressings or absorbent pads for physiological fluids such as urine or blood, e.g. sanitary towels, tampons
    • A61L15/22Bandages, dressings or absorbent pads for physiological fluids such as urine or blood, e.g. sanitary towels, tampons containing macromolecular materials
    • A61L15/26Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61LMETHODS OR APPARATUS FOR STERILISING MATERIALS OR OBJECTS IN GENERAL; DISINFECTION, STERILISATION OR DEODORISATION OF AIR; CHEMICAL ASPECTS OF BANDAGES, DRESSINGS, ABSORBENT PADS OR SURGICAL ARTICLES; MATERIALS FOR BANDAGES, DRESSINGS, ABSORBENT PADS OR SURGICAL ARTICLES
    • A61L15/00Chemical aspects of, or use of materials for, bandages, dressings or absorbent pads
    • A61L15/16Bandages, dressings or absorbent pads for physiological fluids such as urine or blood, e.g. sanitary towels, tampons
    • A61L15/42Use of materials characterised by their function or physical properties
    • A61L15/58Adhesives
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B32LAYERED PRODUCTS
    • B32BLAYERED PRODUCTS, i.e. PRODUCTS BUILT-UP OF STRATA OF FLAT OR NON-FLAT, e.g. CELLULAR OR HONEYCOMB, FORM
    • B32B27/00Layered products comprising a layer of synthetic resin
    • B32B27/12Layered products comprising a layer of synthetic resin next to a fibrous or filamentary layer
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B32LAYERED PRODUCTS
    • B32BLAYERED PRODUCTS, i.e. PRODUCTS BUILT-UP OF STRATA OF FLAT OR NON-FLAT, e.g. CELLULAR OR HONEYCOMB, FORM
    • B32B7/00Layered products characterised by the relation between layers; Layered products characterised by the relative orientation of features between layers, or by the relative values of a measurable parameter between layers, i.e. products comprising layers having different physical, chemical or physicochemical properties; Layered products characterised by the interconnection of layers
    • B32B7/04Interconnection of layers
    • B32B7/12Interconnection of layers using interposed adhesives or interposed materials with bonding properties
    • CCHEMISTRY; METALLURGY
    • C09DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
    • C09JADHESIVES; NON-MECHANICAL ASPECTS OF ADHESIVE PROCESSES IN GENERAL; ADHESIVE PROCESSES NOT PROVIDED FOR ELSEWHERE; USE OF MATERIALS AS ADHESIVES
    • C09J7/00Adhesives in the form of films or foils
    • C09J7/20Adhesives in the form of films or foils characterised by their carriers
    • C09J7/29Laminated material
    • CCHEMISTRY; METALLURGY
    • C09DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
    • C09JADHESIVES; NON-MECHANICAL ASPECTS OF ADHESIVE PROCESSES IN GENERAL; ADHESIVE PROCESSES NOT PROVIDED FOR ELSEWHERE; USE OF MATERIALS AS ADHESIVES
    • C09J2400/00Presence of inorganic and organic materials
    • C09J2400/20Presence of organic materials
    • C09J2400/26Presence of textile or fabric
    • C09J2400/263Presence of textile or fabric in the substrate
    • CCHEMISTRY; METALLURGY
    • C09DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
    • C09JADHESIVES; NON-MECHANICAL ASPECTS OF ADHESIVE PROCESSES IN GENERAL; ADHESIVE PROCESSES NOT PROVIDED FOR ELSEWHERE; USE OF MATERIALS AS ADHESIVES
    • C09J2467/00Presence of polyester
    • C09J2467/006Presence of polyester in the substrate
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10TTECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
    • Y10T156/00Adhesive bonding and miscellaneous chemical manufacture
    • Y10T156/10Methods of surface bonding and/or assembly therefor
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10TTECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
    • Y10T428/00Stock material or miscellaneous articles
    • Y10T428/24Structurally defined web or sheet [e.g., overall dimension, etc.]
    • Y10T428/24942Structurally defined web or sheet [e.g., overall dimension, etc.] including components having same physical characteristic in differing degree
    • Y10T428/2495Thickness [relative or absolute]
    • Y10T428/24959Thickness [relative or absolute] of adhesive layers

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Dermatology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Hematology (AREA)
  • Materials Engineering (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Materials For Medical Uses (AREA)
  • Laminated Bodies (AREA)

Abstract

1. Клейкая лекарственная форма, состоящая из ! подложки и ! самоклеящегося клейкого слоя, который содержит лекарственное средство и нанесен, по меньшей мере, на одну сторону подложки, ! где подложка состоит из полиэфирной пленки, имеющей толщину от 0,5 до 6,0 мкм, и полиэфирного нетканого материала, непосредственно связанного с указанной пленкой. ! 2. Клейкая лекарственная форма по п.1, где самоклеящийся клейкий слой непосредственно или через промежуточный слой нанесен на подложку со стороны нетканого материала. ! 3. Клейкая лекарственная форма по п.1, где полиэфирное волокно указанного нетканого материала непосредственно связано с частью полиэфирной пленки, к которой прикреплен указанный нетканый материал. ! 4. Клейкая лекарственная форма по п.1, где указанный нетканый материал имеет плотность от 5 до 40 г/м2. ! 5. Клейкая лекарственная форма по п.1, где в молекулу лекарственного средства входит, по меньшей мере, одна первичная, вторичная или третичная аминогруппа. ! 6. Клейкая лекарственная форма по п.1, где указанная пленка и указанный нетканый материал сплавлены друг с другом. ! 7. Клейкая лекарственная форма по п.1, где самоклеящийся клейкий слой нанесен на подложку со стороны указанной пленки.

Claims (7)

1. Клейкая лекарственная форма, состоящая из
подложки и
самоклеящегося клейкого слоя, который содержит лекарственное средство и нанесен, по меньшей мере, на одну сторону подложки,
где подложка состоит из полиэфирной пленки, имеющей толщину от 0,5 до 6,0 мкм, и полиэфирного нетканого материала, непосредственно связанного с указанной пленкой.
2. Клейкая лекарственная форма по п.1, где самоклеящийся клейкий слой непосредственно или через промежуточный слой нанесен на подложку со стороны нетканого материала.
3. Клейкая лекарственная форма по п.1, где полиэфирное волокно указанного нетканого материала непосредственно связано с частью полиэфирной пленки, к которой прикреплен указанный нетканый материал.
4. Клейкая лекарственная форма по п.1, где указанный нетканый материал имеет плотность от 5 до 40 г/м2.
5. Клейкая лекарственная форма по п.1, где в молекулу лекарственного средства входит, по меньшей мере, одна первичная, вторичная или третичная аминогруппа.
6. Клейкая лекарственная форма по п.1, где указанная пленка и указанный нетканый материал сплавлены друг с другом.
7. Клейкая лекарственная форма по п.1, где самоклеящийся клейкий слой нанесен на подложку со стороны указанной пленки.
RU2007143383/15A 2006-11-22 2007-11-22 Клейкие лекарственные формы RU2446790C2 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2006-315751 2006-11-22
JP2006315751A JP4392016B2 (ja) 2006-11-22 2006-11-22 貼付製剤

Publications (2)

Publication Number Publication Date
RU2007143383A true RU2007143383A (ru) 2009-05-27
RU2446790C2 RU2446790C2 (ru) 2012-04-10

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RU2007143383/15A RU2446790C2 (ru) 2006-11-22 2007-11-22 Клейкие лекарственные формы

Country Status (9)

Country Link
US (2) US20080118725A1 (ru)
EP (1) EP1925300B1 (ru)
JP (1) JP4392016B2 (ru)
KR (1) KR101093396B1 (ru)
CN (1) CN101194898B (ru)
AT (1) ATE488228T1 (ru)
CA (1) CA2611727C (ru)
DE (1) DE602007010570D1 (ru)
RU (1) RU2446790C2 (ru)

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JP5193674B2 (ja) * 2007-06-01 2013-05-08 日東電工株式会社 貼付剤および貼付製剤
JP5432613B2 (ja) * 2008-07-17 2014-03-05 日東電工株式会社 貼付剤および貼付製剤
JP5432614B2 (ja) * 2008-07-17 2014-03-05 日東電工株式会社 貼付剤および貼付製剤
JP2010126450A (ja) * 2008-11-25 2010-06-10 Lintec Corp 経皮吸収貼付剤
JP2010241746A (ja) * 2009-04-07 2010-10-28 Nitto Denko Corp 貼付剤および貼付製剤
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Also Published As

Publication number Publication date
CN101194898B (zh) 2012-09-26
ATE488228T1 (de) 2010-12-15
US20080118725A1 (en) 2008-05-22
RU2446790C2 (ru) 2012-04-10
CA2611727C (en) 2013-04-02
KR101093396B1 (ko) 2011-12-14
JP4392016B2 (ja) 2009-12-24
EP1925300A3 (en) 2008-09-17
JP2008127351A (ja) 2008-06-05
CA2611727A1 (en) 2008-05-22
US20110056609A1 (en) 2011-03-10
EP1925300B1 (en) 2010-11-17
EP1925300A2 (en) 2008-05-28
KR20080046578A (ko) 2008-05-27
DE602007010570D1 (de) 2010-12-30
CN101194898A (zh) 2008-06-11

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