RU2007124069A - Способы приготовления аминоэтоксибензиловых спиртов - Google Patents
Способы приготовления аминоэтоксибензиловых спиртов Download PDFInfo
- Publication number
- RU2007124069A RU2007124069A RU2007124069/04A RU2007124069A RU2007124069A RU 2007124069 A RU2007124069 A RU 2007124069A RU 2007124069/04 A RU2007124069/04 A RU 2007124069/04A RU 2007124069 A RU2007124069 A RU 2007124069A RU 2007124069 A RU2007124069 A RU 2007124069A
- Authority
- RU
- Russia
- Prior art keywords
- heteroaryl
- aryl
- formula
- alkyl
- group
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C217/00—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
- C07C217/02—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C217/04—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
- C07C217/06—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted
- C07C217/14—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted the oxygen atom of the etherified hydroxy group being further bound to a carbon atom of a six-membered aromatic ring
- C07C217/18—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted the oxygen atom of the etherified hydroxy group being further bound to a carbon atom of a six-membered aromatic ring the six-membered aromatic ring or condensed ring system containing that ring being further substituted
- C07C217/20—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted the oxygen atom of the etherified hydroxy group being further bound to a carbon atom of a six-membered aromatic ring the six-membered aromatic ring or condensed ring system containing that ring being further substituted by halogen atoms, by trihalomethyl, nitro or nitroso groups, or by singly-bound oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
- C07D295/084—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
- C07D295/088—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
- C07C213/02—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reactions involving the formation of amino groups from compounds containing hydroxy groups or etherified or esterified hydroxy groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
- C07C213/08—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reactions not involving the formation of amino groups, hydroxy groups or etherified or esterified hydroxy groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C217/00—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
- C07C217/02—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C217/04—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
- C07C217/06—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted
- C07C217/14—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted the oxygen atom of the etherified hydroxy group being further bound to a carbon atom of a six-membered aromatic ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US64350505P | 2005-01-13 | 2005-01-13 | |
US60/643,505 | 2005-01-13 |
Publications (1)
Publication Number | Publication Date |
---|---|
RU2007124069A true RU2007124069A (ru) | 2009-02-20 |
Family
ID=36570630
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RU2007124069/04A RU2007124069A (ru) | 2005-01-13 | 2006-01-11 | Способы приготовления аминоэтоксибензиловых спиртов |
Country Status (21)
Country | Link |
---|---|
US (2) | US7375251B2 (es) |
EP (1) | EP1836155A2 (es) |
JP (1) | JP2008526969A (es) |
KR (1) | KR20070097502A (es) |
CN (1) | CN101107217A (es) |
AR (1) | AR055837A1 (es) |
AU (1) | AU2006205099A1 (es) |
BR (1) | BRPI0606659A2 (es) |
CA (1) | CA2593965A1 (es) |
CR (1) | CR9208A (es) |
GT (1) | GT200600010A (es) |
IL (1) | IL184193A0 (es) |
MX (1) | MX2007008450A (es) |
NI (1) | NI200700175A (es) |
NO (1) | NO20073276L (es) |
PA (1) | PA8659601A1 (es) |
PE (1) | PE20060874A1 (es) |
RU (1) | RU2007124069A (es) |
SG (1) | SG158860A1 (es) |
TW (1) | TW200637803A (es) |
WO (1) | WO2006076350A2 (es) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2010118997A1 (en) | 2009-04-13 | 2010-10-21 | Sandoz Ag | Processes for the synthesis of bazedoxifene acetate and intermediates thereof |
EP2794580A1 (en) * | 2011-12-23 | 2014-10-29 | Basf Se | Process for manufacturing benzoxazinones |
MX360806B (es) * | 2012-08-17 | 2018-11-16 | Basf Se | Benzoxazinonas de carbamato. |
WO2017004485A1 (en) | 2015-07-02 | 2017-01-05 | Raptor Pharmaceuticals Inc. | Ado-resistant cysteamine analogs and uses thereof |
CN107793344B (zh) * | 2017-10-24 | 2021-01-12 | 扬子江药业集团有限公司 | 一种醋酸巴多昔芬的工业化生产方法 |
CN113816892A (zh) * | 2021-08-27 | 2021-12-21 | 安徽鼎旺医药有限公司 | 一种醋酸巴多昔芬的合成方法 |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CH543472A (fr) | 1969-01-31 | 1973-10-31 | Orchimed Sa | Procédé pour la préparation d'acides phénoxyalcoyl-carboxyliques |
DE2003430C3 (de) * | 1969-01-31 | 1978-12-07 | Laboratorien Fournier Gmbh, 6600 Saarbruecken | p-Benzoylphenoxyisobuttersäureester, ihre Herstellung und diese enthaltende Arzneimittel |
US3772356A (en) * | 1970-03-26 | 1973-11-13 | Lab Bruneau & Cie | Phenoxy-acetamides |
GB8919434D0 (en) * | 1989-08-25 | 1989-10-11 | Beecham Group Plc | Novel compounds |
DE4438028A1 (de) | 1994-10-25 | 1996-05-02 | Thomae Gmbh Dr K | Basisch substituierte N-Phenylalkyl- und N-Phenoxyalkylamide, deren Salze, diese Verbindungen enthaltende Arzneimittel und deren Verwendung sowie Verfahren zu ihrer Herstellung |
US5998402A (en) | 1996-04-19 | 1999-12-07 | American Home Products Corporation | 2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents |
US5929097A (en) | 1996-10-16 | 1999-07-27 | American Cyanamid Company | Preparation and use of ortho-sulfonamido aryl hydroxamic acids as matrix metalloproteinase and tace inhibitors |
EA003937B1 (ru) * | 1997-10-15 | 2003-10-30 | Уайт | Новые арилоксиалкилдиалкиламины |
US6005102A (en) | 1997-10-15 | 1999-12-21 | American Home Products Corporation | Aryloxy-alkyl-dialkylamines |
DE10146867A1 (de) * | 2001-09-24 | 2003-04-24 | Bayer Ag | Tetrahydroisochinoline |
MXPA05008878A (es) * | 2003-02-21 | 2005-10-05 | Pfizer | Derivados de aminotiazol sustituidos con cicloalquilo que contiene n y composiciones farmaceuticas para inhibir la proliferacion celular, y metodos para su uso. |
-
2006
- 2006-01-11 BR BRPI0606659-3A patent/BRPI0606659A2/pt not_active IP Right Cessation
- 2006-01-11 MX MX2007008450A patent/MX2007008450A/es active IP Right Grant
- 2006-01-11 GT GT200600010A patent/GT200600010A/es unknown
- 2006-01-11 TW TW095100972A patent/TW200637803A/zh unknown
- 2006-01-11 EP EP06717938A patent/EP1836155A2/en not_active Withdrawn
- 2006-01-11 SG SG201000069-3A patent/SG158860A1/en unknown
- 2006-01-11 PE PE2006000056A patent/PE20060874A1/es not_active Application Discontinuation
- 2006-01-11 US US11/329,503 patent/US7375251B2/en not_active Expired - Fee Related
- 2006-01-11 JP JP2007551320A patent/JP2008526969A/ja active Pending
- 2006-01-11 WO PCT/US2006/000801 patent/WO2006076350A2/en active Application Filing
- 2006-01-11 AU AU2006205099A patent/AU2006205099A1/en not_active Abandoned
- 2006-01-11 AR ARP060100114A patent/AR055837A1/es unknown
- 2006-01-11 KR KR1020077016099A patent/KR20070097502A/ko not_active Application Discontinuation
- 2006-01-11 PA PA20068659601A patent/PA8659601A1/es unknown
- 2006-01-11 CA CA002593965A patent/CA2593965A1/en not_active Abandoned
- 2006-01-11 RU RU2007124069/04A patent/RU2007124069A/ru not_active Application Discontinuation
- 2006-01-11 CN CNA2006800022748A patent/CN101107217A/zh active Pending
-
2007
- 2007-06-25 CR CR9208A patent/CR9208A/es not_active Application Discontinuation
- 2007-06-25 IL IL184193A patent/IL184193A0/en unknown
- 2007-06-27 NO NO20073276A patent/NO20073276L/no not_active Application Discontinuation
- 2007-07-11 NI NI200700175A patent/NI200700175A/es unknown
-
2008
- 2008-04-17 US US12/104,960 patent/US20080207898A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
US20060155147A1 (en) | 2006-07-13 |
AR055837A1 (es) | 2007-09-12 |
AU2006205099A1 (en) | 2006-07-20 |
IL184193A0 (en) | 2007-10-31 |
PA8659601A1 (es) | 2007-01-17 |
SG158860A1 (en) | 2010-02-26 |
CR9208A (es) | 2007-10-23 |
CA2593965A1 (en) | 2006-07-20 |
NI200700175A (es) | 2008-05-09 |
JP2008526969A (ja) | 2008-07-24 |
PE20060874A1 (es) | 2006-10-16 |
CN101107217A (zh) | 2008-01-16 |
BRPI0606659A2 (pt) | 2009-07-07 |
EP1836155A2 (en) | 2007-09-26 |
WO2006076350A2 (en) | 2006-07-20 |
NO20073276L (no) | 2007-09-04 |
KR20070097502A (ko) | 2007-10-04 |
MX2007008450A (es) | 2007-08-06 |
US20080207898A1 (en) | 2008-08-28 |
WO2006076350A3 (en) | 2007-03-01 |
US7375251B2 (en) | 2008-05-20 |
TW200637803A (en) | 2006-11-01 |
GT200600010A (es) | 2006-08-16 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
RU2007124069A (ru) | Способы приготовления аминоэтоксибензиловых спиртов | |
CN101470349B (zh) | 抗蚀剂组合物、抗蚀剂图案的形成方法、新型化合物以及产酸剂 | |
RU2406722C2 (ru) | Соли бис-(тиогидразидамида) для лечения рака | |
TWI525071B (zh) | 新穎化合物 | |
RU2011121785A (ru) | Синтез карбамоилпиридоновых ингибиторов интегразы вич и промежуточных соединений | |
Katritzky et al. | Benzotriazole-mediated arylalkylation and heteroarylalkylation | |
JP2008517965A5 (es) | ||
RU2008118067A (ru) | Способ получения делмопинола и его производных | |
RU2006129650A (ru) | Способы приготовления арил- и гетероарилалкилсульфонилгалогенидов | |
EP2215063B1 (en) | Facile n-alkylation of acridine compounds in ionic liquids | |
CN105688987A (zh) | 一种新型的手性磷酸催化剂及其合成方法与应用 | |
US20050203317A1 (en) | Method of removing allyl series protecting group using novel ruthenium complex and method of synthesizing allyl ethers | |
JP2022523160A (ja) | 方法および化合物 | |
CN111548269B (zh) | 一种二芳基甲烷结构化合物的制备方法 | |
JP5046213B2 (ja) | 光学活性アルコール化合物の製法 | |
RU2211837C2 (ru) | Трехъядерные конденсированные гетероциклические соединения, способ их получения (варианты) и фармацевтическая композиция | |
CN113185469A (zh) | 一种光调节二芳基二氢吩嗪修饰的方法 | |
EP3484842B1 (en) | Halogen-containing metathesis catalysts and methods thereof | |
Liu et al. | A general and efficient method for synthesis of enaminones and enamino esters catalyzed by NbCl 5 under solvent-free conditions | |
SK20297A3 (en) | Process for producing (3-alkoxyphenyl) magnesium chlorides and their use | |
CN103153936B (zh) | 改进的培瑞维a酸的合成 | |
Lam | Sodium arylsulfinates as a versatile sulfur surrogate for the synthesis of diaryl thioethers and n-aryl sulfonamides | |
KR102132339B1 (ko) | 플라보노이드 유도체의 제조방법 및 그 중간체 | |
JP3822510B2 (ja) | (チオ)エーテルの製造方法および(チオ)アセタールの製造方法 | |
RU2005119155A (ru) | Способ получения имидазолильных соединений |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA92 | Acknowledgement of application withdrawn (lack of supplementary materials submitted) |
Effective date: 20110112 |