RU2005133660A - Кристаллические n-формилгидроксиламиновые соединения - Google Patents

Кристаллические n-формилгидроксиламиновые соединения Download PDF

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Publication number
RU2005133660A
RU2005133660A RU2005133660/04A RU2005133660A RU2005133660A RU 2005133660 A RU2005133660 A RU 2005133660A RU 2005133660/04 A RU2005133660/04 A RU 2005133660/04A RU 2005133660 A RU2005133660 A RU 2005133660A RU 2005133660 A RU2005133660 A RU 2005133660A
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RU
Russia
Prior art keywords
alkyl
hydrogen
aryl
denotes
crystalline salt
Prior art date
Application number
RU2005133660/04A
Other languages
English (en)
Russian (ru)
Inventor
Джоэл СЛЕЙД (US)
Джоэл СЛЕЙД
Мартин МЮЛЛЕР (CH)
Мартин Мюллер
Сюй ЛЮ (US)
Сюй ЛЮ
Джоджиндер Сингх БАЙВА (US)
Джоджиндер Сингх БАЙВА
Original Assignee
Новартис АГ (CH)
Новартис Аг
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=33131903&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=RU2005133660(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Новартис АГ (CH), Новартис Аг filed Critical Новартис АГ (CH)
Publication of RU2005133660A publication Critical patent/RU2005133660A/ru

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C259/00Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups
    • C07C259/04Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids
    • C07C259/06Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids having carbon atoms of hydroxamic groups bound to hydrogen atoms or to acyclic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/06Antimalarials
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
RU2005133660/04A 2003-04-02 2004-04-01 Кристаллические n-формилгидроксиламиновые соединения RU2005133660A (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US45972603P 2003-04-02 2003-04-02
US60/459,726 2003-04-02

Publications (1)

Publication Number Publication Date
RU2005133660A true RU2005133660A (ru) 2006-06-10

Family

ID=33131903

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2005133660/04A RU2005133660A (ru) 2003-04-02 2004-04-01 Кристаллические n-формилгидроксиламиновые соединения

Country Status (25)

Country Link
US (1) US20070135353A1 (https=)
EP (1) EP1613305A1 (https=)
JP (1) JP2006522054A (https=)
KR (1) KR20060002915A (https=)
CN (1) CN1764450A (https=)
AR (1) AR043804A1 (https=)
AU (1) AU2004226815B2 (https=)
BR (1) BRPI0409009A (https=)
CA (1) CA2520682A1 (https=)
CL (1) CL2004000705A1 (https=)
CO (1) CO5630028A2 (https=)
EC (1) ECSP056043A (https=)
IS (1) IS8093A (https=)
MA (1) MA27763A1 (https=)
MX (1) MXPA05010610A (https=)
MY (1) MY136854A (https=)
NO (1) NO20055097L (https=)
NZ (1) NZ542432A (https=)
PE (1) PE20050392A1 (https=)
RU (1) RU2005133660A (https=)
SG (1) SG166681A1 (https=)
TN (1) TNSN05248A1 (https=)
TW (1) TW200427458A (https=)
WO (1) WO2004087133A1 (https=)
ZA (1) ZA200507179B (https=)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1406893B1 (en) 2001-06-15 2007-04-18 Vicuron Pharmaceuticals, Inc. Pyrrolidine bicyclic compounds
ATE417826T1 (de) 2002-09-19 2009-01-15 Novartis Pharma Gmbh Verfahren zur herstellung von zwischenprodukten
MXPA05008842A (es) 2003-02-21 2005-10-05 Novartis Ag Proceso quimico.
GT200600196A (es) * 2005-05-23 2007-01-15 Compuestos n-formil de hidroxilamina
JP7001898B2 (ja) * 2016-05-11 2022-01-20 グアンドン・ヘボ・ファーマシューティカル・カンパニー・リミテッド スピロ3員環、スピロ5員環系ペプチドデホルミラーゼ阻害剤および抗菌と抗腫瘍におけるその使用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3282986A (en) * 1960-10-06 1966-11-01 Merck & Co Inc N-acylated hydroxamic acids and derivatives thereof
DK1052984T3 (da) * 1998-02-07 2004-09-20 Vernalis Oxford Ltd Antibakterielle midler
AR036053A1 (es) * 2001-06-15 2004-08-04 Versicor Inc Compuestos de n-formil-hidroxilamina, un proceso para su preparacion y composiciones farmaceuticas

Also Published As

Publication number Publication date
NO20055097L (no) 2005-12-22
CA2520682A1 (en) 2004-10-14
US20070135353A1 (en) 2007-06-14
AU2004226815B2 (en) 2007-07-19
NZ542432A (en) 2009-04-30
PE20050392A1 (es) 2005-06-19
TNSN05248A1 (en) 2007-06-11
MXPA05010610A (es) 2005-11-23
BRPI0409009A (pt) 2006-03-28
IS8093A (is) 2005-10-27
AU2004226815A1 (en) 2004-10-14
CO5630028A2 (es) 2006-04-28
SG166681A1 (en) 2010-12-29
CL2004000705A1 (es) 2005-01-14
WO2004087133A1 (en) 2004-10-14
MA27763A1 (fr) 2006-02-01
MY136854A (en) 2008-11-28
ZA200507179B (en) 2006-04-26
NO20055097D0 (no) 2005-11-01
KR20060002915A (ko) 2006-01-09
ECSP056043A (es) 2006-01-27
JP2006522054A (ja) 2006-09-28
TW200427458A (en) 2004-12-16
EP1613305A1 (en) 2006-01-11
AR043804A1 (es) 2005-08-10
CN1764450A (zh) 2006-04-26

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FA94 Acknowledgement of application withdrawn (non-payment of fees)

Effective date: 20101209