BRPI0409009A - compostos cristalinos de n-formila hidroxilamina - Google Patents
compostos cristalinos de n-formila hidroxilaminaInfo
- Publication number
- BRPI0409009A BRPI0409009A BRPI0409009-8A BRPI0409009A BRPI0409009A BR PI0409009 A BRPI0409009 A BR PI0409009A BR PI0409009 A BRPI0409009 A BR PI0409009A BR PI0409009 A BRPI0409009 A BR PI0409009A
- Authority
- BR
- Brazil
- Prior art keywords
- formyl hydroxylamine
- compounds
- alkanes
- crystalline compounds
- crystalline
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C259/00—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups
- C07C259/04—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids
- C07C259/06—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids having carbon atoms of hydroxamic groups bound to hydrogen atoms or to acyclic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Tropical Medicine & Parasitology (AREA)
- Engineering & Computer Science (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
"COMPOSTOS CRISTALINOS DE N-FORMILA HIDROXILAMINA". A presente invenção refere-se a determinados compostos de N-formil hidroxilamina, tal como N-¢1-oxo-2-alquil-3-(N-hidróxiformamido)-propil!-(carbonilamino-aril ou -heteroaril)-azaciclo~ 4-7~alcanos ou tiazaciclo~ 4-7~ alcanos ou imidazaciclo~ 4-7~alcanos que são úteis no tratamento de infecções bacterianas. São descritos sais cristalinos desses compostos da fórmula (I), nos quais M é um metal mono- ou divalente; a é 1/2 ou 1.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US45972603P | 2003-04-02 | 2003-04-02 | |
PCT/EP2004/003478 WO2004087133A1 (en) | 2003-04-02 | 2004-04-01 | Crystalline n-formyl hydroxylamine compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0409009A true BRPI0409009A (pt) | 2006-03-28 |
Family
ID=33131903
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0409009-8A BRPI0409009A (pt) | 2003-04-02 | 2004-04-01 | compostos cristalinos de n-formila hidroxilamina |
Country Status (25)
Country | Link |
---|---|
US (1) | US20070135353A1 (pt) |
EP (1) | EP1613305A1 (pt) |
JP (1) | JP2006522054A (pt) |
KR (1) | KR20060002915A (pt) |
CN (1) | CN1764450A (pt) |
AR (1) | AR043804A1 (pt) |
AU (1) | AU2004226815B2 (pt) |
BR (1) | BRPI0409009A (pt) |
CA (1) | CA2520682A1 (pt) |
CL (1) | CL2004000705A1 (pt) |
CO (1) | CO5630028A2 (pt) |
EC (1) | ECSP056043A (pt) |
IS (1) | IS8093A (pt) |
MA (1) | MA27763A1 (pt) |
MX (1) | MXPA05010610A (pt) |
MY (1) | MY136854A (pt) |
NO (1) | NO20055097L (pt) |
NZ (1) | NZ542432A (pt) |
PE (1) | PE20050392A1 (pt) |
RU (1) | RU2005133660A (pt) |
SG (1) | SG166681A1 (pt) |
TN (1) | TNSN05248A1 (pt) |
TW (1) | TW200427458A (pt) |
WO (1) | WO2004087133A1 (pt) |
ZA (1) | ZA200507179B (pt) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6987104B2 (en) | 2001-06-15 | 2006-01-17 | Vicuron Pharmaceuticals Inc. | Pyrrolidine bicyclic compounds and its derivatives, compositions and methods of use |
KR20050057429A (ko) | 2002-09-19 | 2005-06-16 | 노파르티스 아게 | 중간체의 제조 방법 |
EP1599440A2 (en) | 2003-02-21 | 2005-11-30 | Novartis AG | Chemical process for the preparation of intermediates to obtain n-formyl hydroxylamine compounds |
GT200600196A (es) * | 2005-05-23 | 2007-01-15 | Compuestos n-formil de hidroxilamina | |
ES2930814T3 (es) * | 2016-05-11 | 2022-12-22 | Guangdong Hebo Pharmaceutical Co Ltd | Inhibidor de péptido deformilasa de anillo espiro de tres miembros o anillo espiro de cinco miembros y uso del mismo como agente antitumoral |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3282986A (en) * | 1960-10-06 | 1966-11-01 | Merck & Co Inc | N-acylated hydroxamic acids and derivatives thereof |
GB2349884A (en) * | 1998-02-07 | 2000-11-15 | British Biotech Pharm | Antibacterial agents |
AR036053A1 (es) * | 2001-06-15 | 2004-08-04 | Versicor Inc | Compuestos de n-formil-hidroxilamina, un proceso para su preparacion y composiciones farmaceuticas |
-
2004
- 2004-03-29 TW TW093108548A patent/TW200427458A/zh unknown
- 2004-03-31 PE PE2004000339A patent/PE20050392A1/es not_active Application Discontinuation
- 2004-03-31 AR ARP040101079A patent/AR043804A1/es not_active Application Discontinuation
- 2004-04-01 CL CL200400705A patent/CL2004000705A1/es unknown
- 2004-04-01 AU AU2004226815A patent/AU2004226815B2/en not_active Ceased
- 2004-04-01 MX MXPA05010610A patent/MXPA05010610A/es unknown
- 2004-04-01 NZ NZ542432A patent/NZ542432A/en unknown
- 2004-04-01 CN CNA2004800078725A patent/CN1764450A/zh active Pending
- 2004-04-01 RU RU2005133660/04A patent/RU2005133660A/ru not_active Application Discontinuation
- 2004-04-01 CA CA002520682A patent/CA2520682A1/en not_active Abandoned
- 2004-04-01 US US10/550,631 patent/US20070135353A1/en not_active Abandoned
- 2004-04-01 WO PCT/EP2004/003478 patent/WO2004087133A1/en active IP Right Grant
- 2004-04-01 EP EP04725014A patent/EP1613305A1/en not_active Ceased
- 2004-04-01 BR BRPI0409009-8A patent/BRPI0409009A/pt not_active IP Right Cessation
- 2004-04-01 MY MYPI20041200A patent/MY136854A/en unknown
- 2004-04-01 JP JP2006504952A patent/JP2006522054A/ja active Pending
- 2004-04-01 KR KR1020057018676A patent/KR20060002915A/ko not_active Application Discontinuation
- 2004-04-01 SG SG200801365-8A patent/SG166681A1/en unknown
-
2005
- 2005-09-07 ZA ZA200507179A patent/ZA200507179B/en unknown
- 2005-09-28 EC EC2005006043A patent/ECSP056043A/es unknown
- 2005-09-30 TN TNP2005000248A patent/TNSN05248A1/en unknown
- 2005-10-04 CO CO05100510A patent/CO5630028A2/es not_active Application Discontinuation
- 2005-10-11 MA MA28547A patent/MA27763A1/fr unknown
- 2005-10-27 IS IS8093A patent/IS8093A/is unknown
- 2005-11-01 NO NO20055097A patent/NO20055097L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
AU2004226815B2 (en) | 2007-07-19 |
NO20055097D0 (no) | 2005-11-01 |
AU2004226815A1 (en) | 2004-10-14 |
WO2004087133A1 (en) | 2004-10-14 |
PE20050392A1 (es) | 2005-06-19 |
ZA200507179B (en) | 2006-04-26 |
EP1613305A1 (en) | 2006-01-11 |
MY136854A (en) | 2008-11-28 |
KR20060002915A (ko) | 2006-01-09 |
CA2520682A1 (en) | 2004-10-14 |
MA27763A1 (fr) | 2006-02-01 |
RU2005133660A (ru) | 2006-06-10 |
CL2004000705A1 (es) | 2005-01-14 |
CN1764450A (zh) | 2006-04-26 |
US20070135353A1 (en) | 2007-06-14 |
AR043804A1 (es) | 2005-08-10 |
SG166681A1 (en) | 2010-12-29 |
TNSN05248A1 (en) | 2007-06-11 |
ECSP056043A (es) | 2006-01-27 |
JP2006522054A (ja) | 2006-09-28 |
CO5630028A2 (es) | 2006-04-28 |
IS8093A (is) | 2005-10-27 |
NZ542432A (en) | 2009-04-30 |
TW200427458A (en) | 2004-12-16 |
NO20055097L (no) | 2005-12-22 |
MXPA05010610A (es) | 2005-11-23 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 7A E 8A ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2159 DE 22/05/2012. |