PT96139A - Processo para a preparacao de novos derivados de glicopeptido - Google Patents

Processo para a preparacao de novos derivados de glicopeptido

Info

Publication number
PT96139A
PT96139A PT96139A PT9613990A PT96139A PT 96139 A PT96139 A PT 96139A PT 96139 A PT96139 A PT 96139A PT 9613990 A PT9613990 A PT 9613990A PT 96139 A PT96139 A PT 96139A
Authority
PT
Portugal
Prior art keywords
preparing new
glycopeptide derivatives
new glycopeptide
derivatives
preparing
Prior art date
Application number
PT96139A
Other languages
English (en)
Other versions
PT96139B (pt
Inventor
Ramakrishnan Nagarajan
Amelia Apolinaria Schabel
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of PT96139A publication Critical patent/PT96139A/pt
Publication of PT96139B publication Critical patent/PT96139B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
PT96139A 1989-12-13 1990-12-10 Processo para a preparacao de novos derivados de glicopeptido PT96139B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US44917189A 1989-12-13 1989-12-13

Publications (2)

Publication Number Publication Date
PT96139A true PT96139A (pt) 1991-09-30
PT96139B PT96139B (pt) 1998-04-30

Family

ID=23783157

Family Applications (1)

Application Number Title Priority Date Filing Date
PT96139A PT96139B (pt) 1989-12-13 1990-12-10 Processo para a preparacao de novos derivados de glicopeptido

Country Status (20)

Country Link
US (1) US5591714A (pt)
EP (1) EP0435503B1 (pt)
JP (1) JP3590638B2 (pt)
KR (1) KR910011896A (pt)
CN (1) CN1034506C (pt)
CA (1) CA2031803C (pt)
DE (1) DE69033087T2 (pt)
ES (1) ES2131496T3 (pt)
FI (1) FI906083A (pt)
HU (1) HUT55802A (pt)
IE (1) IE904485A1 (pt)
IL (1) IL96603A (pt)
MX (1) MX23672A (pt)
NO (1) NO303692B1 (pt)
NZ (1) NZ236393A (pt)
PH (1) PH27373A (pt)
PT (1) PT96139B (pt)
RU (2) RU2053240C1 (pt)
YU (1) YU234790A (pt)
ZA (1) ZA909847B (pt)

Families Citing this family (43)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5721208A (en) * 1991-06-29 1998-02-24 Hoechst Aktiengesellschaft Glycopeptides a process for their preparation and their use
TW213468B (pt) * 1991-06-29 1993-09-21 Hoechst Ag
PE40996A1 (es) * 1994-01-28 1996-10-14 Lilly Co Eli Derivado de antibiotico de glucopeptido
US5840684A (en) * 1994-01-28 1998-11-24 Eli Lilly And Company Glycopeptide antibiotic derivatives
US5919756A (en) * 1996-06-28 1999-07-06 Eli Lilly And Company Amides
ID18900A (id) * 1996-11-21 1998-05-20 Lilly Co Eli Alkilasi menurun dari gliko peptida anti biotik
US5952466A (en) * 1997-11-12 1999-09-14 Eli Lilly And Company Reductive alkylation of glycopeptide antibiotics
US5939382A (en) * 1996-11-21 1999-08-17 Eli Lilly And Company Reducing agent for reductive alkylation of glycopeptide antibiotics
US5919771A (en) * 1997-05-20 1999-07-06 Eli Lilly And Company Urea and thiourea derivatives of glycopeptides
US5952310A (en) * 1997-05-20 1999-09-14 Eli Lilly And Company Glycopeptide hexapeptides
US5977063A (en) * 1997-05-20 1999-11-02 Eli Lilly And Company Alkylated hexapeptides
US5972933A (en) * 1998-01-08 1999-10-26 Ed. Geistlich Sohne Ag Fur Chemische Industrie Method of treating microbial infections
CA2330619A1 (en) 1998-05-01 1999-11-11 Eli Lilly And Company N1-modified glycopeptides
BR9910481A (pt) 1998-06-11 2001-01-09 Upjohn Co Composição farmacêutica para comprimido de liberação não-contìnua
DK1140993T3 (da) * 1998-12-23 2003-10-06 Theravance Inc Glycopeptidderivater og farmaceutiske præparater indeholdende dem
GB9925127D0 (en) * 1999-10-22 1999-12-22 Pharmacia & Upjohn Spa Oral formulations for anti-tumor compounds
US20020004502A1 (en) * 2000-01-05 2002-01-10 Redmond H. Paul Treatment of inflammatory bowel disease
AU3818001A (en) * 2000-02-11 2001-08-20 Lilly Co Eli Selective n-acylation of a82846 glycopeptide analogs
JP4870314B2 (ja) * 2000-05-02 2012-02-08 セラヴァンス, インコーポレーテッド シクロデキストリンを含むグリコペプチド抗生物質組成物
AU2001259298A1 (en) * 2000-05-02 2001-11-12 Advanced Medicine, Inc. Polyacid glycopeptide derivatives
ATE402951T1 (de) * 2000-05-02 2008-08-15 Theravance Inc Verfahren zur reduktiven alkylierung von glykopeptiden
EP1154663B1 (en) * 2000-05-09 2008-09-24 Lucent Technologies Inc. Improved quality of service control in a mobile telecommunications network
ES2302733T3 (es) * 2000-06-22 2008-08-01 Theravance, Inc. Derivados carboxi-sacaridos de glucopeptido.
AU2001259816A1 (en) 2000-06-22 2002-01-02 Advanced Medecine, Inc. Polyhydroxy glycopeptide derivatives
UA75083C2 (uk) * 2000-06-22 2006-03-15 Тераванс, Інк. Похідні глікопептидфосфонатів
US6872804B2 (en) * 2000-06-22 2005-03-29 Theravance, Inc. Glycopeptide disulfide and thioester derivatives
TWI312785B (en) * 2001-08-24 2009-08-01 Theravance Inc Process for preparing vancomycin derivatives
TWI275594B (en) * 2001-08-24 2007-03-11 Theravance Inc Process for preparing vancomycin phosphonate derivatives
WO2004091578A2 (en) 2003-04-09 2004-10-28 Biodelivery Sciences International, Inc. Novel encochleation methods, cochleates and methods of use
MX2007006319A (es) * 2004-11-29 2007-07-25 Univ Nagoya Nat Univ Corp Derivados de monomeros de glicopeptico antibioticos.
UA90707C2 (en) 2005-04-06 2010-05-25 Астразенека Аб Novel 5-substituted 7-amino-[1,3]thiazolo[4,5-d]pyrimidine derivatives
AR053347A1 (es) 2005-04-06 2007-05-02 Astrazeneca Ab Derivados de [1,3]tiazolo[4,5-d]pirimidin-2(3h)-ona 5,7-sustituidos
WO2007038246A2 (en) 2005-09-22 2007-04-05 Medivas, Llc Solid polymer delivery compositions and methods for use thereof
EP1926780B1 (en) 2005-09-22 2013-08-14 Medivas, LLC Bis-( -amino)-diol-diester-containing poly(ester amide) and poly(ester urethane) compositions and methods of use
TW200808818A (en) 2006-05-26 2008-02-16 Shionogi & Co Glycopeptide antibiotic derivatives
US8481696B2 (en) 2007-12-26 2013-07-09 Shionogi & Co., Ltd. Glycosylated glycopeptide antibiotic derivatives
CN102083862A (zh) 2008-04-01 2011-06-01 康奈尔大学 有机-可溶性壳聚糖盐和由其制备的壳聚糖衍生生物材料
CN101928331B (zh) * 2009-06-26 2014-05-28 上海来益生物药物研究开发中心有限责任公司 一种化合物及其应用
ES2741282T3 (es) 2011-05-05 2020-02-10 Matinas Biopharma Nanotechnologies Inc Composiciones de cocleato y métodos de elaboración y uso de las mismas
CN104418941B (zh) * 2013-08-19 2017-11-07 爱斯医药科技(南京)有限公司 万古霉素衍生物、制备方法及其应用
CA2925005A1 (en) 2013-09-23 2015-03-26 Jawaharlal Nehru Centre for Advanced Scientific Research (JNCASR) Vancomycin-sugar conjugates and uses thereof
JP6712991B2 (ja) * 2014-07-17 2020-06-24 ザ メディシンズ カンパニー 高純度のオリタバンシン及びその製造方法
CN108409837B (zh) 2018-03-06 2021-09-24 上海来益生物药物研究开发中心有限责任公司 一组具有抗耐药性细菌活性的糖肽类化合物、其制备方法和应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4552701A (en) * 1984-04-16 1985-11-12 Eli Lilly And Company Glycopeptide antibiotics and process of preparation
US4698327A (en) * 1985-04-25 1987-10-06 Eli Lilly And Company Novel glycopeptide derivatives
US4639433A (en) * 1985-08-14 1987-01-27 Eli Lilly And Company Glycopeptide derivatives
US4643987A (en) * 1985-08-14 1987-02-17 Eli Lilly And Company Modified glycopeptides
US4946941A (en) * 1986-01-24 1990-08-07 Shionogi & Co., Ltd. Novel glycopeptide antibiotics
EG18377A (en) * 1986-09-19 1993-04-30 Lilly Co Eli Process for preparing glycopeptide antibiotics
GB8701872D0 (en) * 1987-01-28 1987-03-04 Lepetit Spa N15-alkyl & n15,n15-dialkyl derivatives
US5071749A (en) * 1987-04-16 1991-12-10 Shionogi & Co., Ltd. Glycopetide antibiotic pa-45052-b

Also Published As

Publication number Publication date
MX23672A (es) 1993-11-01
AU633165B2 (en) 1993-01-21
HUT55802A (en) 1991-06-28
NO905354D0 (no) 1990-12-11
NO303692B1 (no) 1998-08-17
FI906083A (fi) 1991-06-14
RU2041237C1 (ru) 1995-08-09
IL96603A0 (en) 1991-09-16
CN1034506C (zh) 1997-04-09
NO905354L (no) 1991-06-14
KR910011896A (ko) 1991-08-07
PT96139B (pt) 1998-04-30
ES2131496T3 (es) 1999-08-01
YU234790A (sh) 1992-12-21
RU2053240C1 (ru) 1996-01-27
DE69033087T2 (de) 1999-10-14
AU6796490A (en) 1991-06-20
PH27373A (en) 1993-06-21
EP0435503A1 (en) 1991-07-03
CA2031803A1 (en) 1991-06-14
JP3590638B2 (ja) 2004-11-17
NZ236393A (en) 1992-05-26
CA2031803C (en) 2001-05-29
EP0435503B1 (en) 1999-05-06
DE69033087D1 (de) 1999-06-10
ZA909847B (en) 1992-08-26
US5591714A (en) 1997-01-07
IE904485A1 (en) 1991-06-19
CN1052483A (zh) 1991-06-26
FI906083A0 (fi) 1990-12-11
JPH04108800A (ja) 1992-04-09
IL96603A (en) 1998-02-08

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Legal Events

Date Code Title Description
BB1A Laying open of patent application

Effective date: 19910430

FG3A Patent granted, date of granting

Effective date: 19980123

MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 19990731