PT82445B - Processo para a preparacao de novos derivados glicopeptidicos - Google Patents

Processo para a preparacao de novos derivados glicopeptidicos

Info

Publication number
PT82445B
PT82445B PT82445A PT8244586A PT82445B PT 82445 B PT82445 B PT 82445B PT 82445 A PT82445 A PT 82445A PT 8244586 A PT8244586 A PT 8244586A PT 82445 B PT82445 B PT 82445B
Authority
PT
Portugal
Prior art keywords
glicopeptidic
derivatives
preparing new
preparing
new
Prior art date
Application number
PT82445A
Other languages
English (en)
Other versions
PT82445A (en
Inventor
Ramakrishnan Nagarajan
Amelia Apolinaria Schabel
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of PT82445A publication Critical patent/PT82445A/pt
Publication of PT82445B publication Critical patent/PT82445B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C09DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
    • C09KMATERIALS FOR MISCELLANEOUS APPLICATIONS, NOT PROVIDED FOR ELSEWHERE
    • C09K9/00Tenebrescent materials, i.e. materials for which the range of wavelengths for energy absorption is changed as a result of excitation by some form of energy
PT82445A 1985-04-25 1986-04-23 Processo para a preparacao de novos derivados glicopeptidicos PT82445B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US72673185A 1985-04-25 1985-04-25

Publications (2)

Publication Number Publication Date
PT82445A PT82445A (en) 1986-05-01
PT82445B true PT82445B (pt) 1988-11-30

Family

ID=24919774

Family Applications (1)

Application Number Title Priority Date Filing Date
PT82445A PT82445B (pt) 1985-04-25 1986-04-23 Processo para a preparacao de novos derivados glicopeptidicos

Country Status (15)

Country Link
EP (1) EP0201251A3 (pt)
JP (1) JPS61251699A (pt)
KR (1) KR870001282B1 (pt)
CN (1) CN86103330A (pt)
AU (1) AU587615B2 (pt)
DK (1) DK188486A (pt)
ES (1) ES8706725A1 (pt)
GR (1) GR861071B (pt)
HU (1) HU204854B (pt)
IL (1) IL78597A0 (pt)
NZ (1) NZ215947A (pt)
PH (1) PH23900A (pt)
PT (1) PT82445B (pt)
SU (1) SU1586521A3 (pt)
ZA (1) ZA863091B (pt)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8701872D0 (en) * 1987-01-28 1987-03-04 Lepetit Spa N15-alkyl & n15,n15-dialkyl derivatives
US5071749A (en) * 1987-04-16 1991-12-10 Shionogi & Co., Ltd. Glycopetide antibiotic pa-45052-b
GB8711066D0 (en) * 1987-05-11 1987-06-17 Lepetit Spa Teicoplanin derivatives
GB8817053D0 (en) * 1988-07-18 1988-08-24 Lepetit Spa Process for preparing n15 n15-dialkyl derivatives of teicoplanin compounds
UA43323C2 (uk) * 1994-01-28 2001-12-17 Елі Ліллі Енд Компані Антибіотичні похідні глікопептидів, спосіб отримання та фармацевтична композиція
US5840684A (en) * 1994-01-28 1998-11-24 Eli Lilly And Company Glycopeptide antibiotic derivatives
JP4051421B2 (ja) * 1995-07-05 2008-02-27 サノフイ−アベンテイス・エツセ・ピー・アー 等電点電気泳動によるダルバヘプチド抗生物質の精製
JP4713810B2 (ja) 2000-05-02 2011-06-29 セラヴァンス, インコーポレーテッド グリコペプチドに対する還元的アルキル化プロセス
TWI312785B (en) 2001-08-24 2009-08-01 Theravance Inc Process for preparing vancomycin derivatives
TWI275594B (en) 2001-08-24 2007-03-11 Theravance Inc Process for preparing vancomycin phosphonate derivatives
EP1818340A4 (en) 2004-11-29 2009-02-25 Univ Nagoya Nat Univ Corp MONOMERIC ANTIBIOTIC DERIVATIVES OF GLYCOPEPTIDES
TW200808818A (en) 2006-05-26 2008-02-16 Shionogi & Co Glycopeptide antibiotic derivatives
US8481696B2 (en) 2007-12-26 2013-07-09 Shionogi & Co., Ltd. Glycosylated glycopeptide antibiotic derivatives
US10577395B2 (en) * 2014-07-10 2020-03-03 The Scripps Research Institute N-(hydrophobe-substituted) vancosaminyl [Ψ-[C(=NH) NH] Tpg4] vancomycin and [Ψ-[CH2NH]Tpg4] vancomycin
CN105985412A (zh) * 2015-02-28 2016-10-05 爱斯医药科技(南京)有限公司 万古霉素衍生物、制备方法及其应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4462942A (en) * 1982-07-30 1984-07-31 Eli Lilly And Company A47934 Antibiotic and process for production thereof
IL70441A (en) * 1982-12-20 1986-11-30 Lilly Co Eli Antibiotic a 51568 factors a and b and process for production thereof
DE3572178D1 (en) * 1984-04-16 1989-09-14 Lilly Co Eli Improvements in and relating to antibiotics m43a, m43b, m43c and m43d

Also Published As

Publication number Publication date
SU1586521A3 (ru) 1990-08-15
PH23900A (en) 1989-12-18
HUT40683A (en) 1987-01-28
DK188486D0 (da) 1986-04-24
NZ215947A (en) 1988-10-28
EP0201251A2 (en) 1986-11-12
CN86103330A (zh) 1986-10-29
IL78597A0 (en) 1986-08-31
ZA863091B (en) 1987-12-30
HU204854B (en) 1992-02-28
GR861071B (en) 1986-08-21
ES8706725A1 (es) 1987-07-01
AU587615B2 (en) 1989-08-24
PT82445A (en) 1986-05-01
KR870001282B1 (ko) 1987-06-30
DK188486A (da) 1986-10-26
ES554286A0 (es) 1987-07-01
EP0201251A3 (en) 1987-12-16
JPS61251699A (ja) 1986-11-08
KR860008210A (ko) 1986-11-14
AU5659886A (en) 1986-10-30

Similar Documents

Publication Publication Date Title
PT82890B (pt) Processo para a preparacao de novos derivados de n-aralquil-piperidinametanol
ES547326A0 (es) Un metodo para preparar esterol-liposomas
PT81859B (pt) Processo para a preparacao de derivados de tiazolidinodionas
ES554380A0 (es) Un procedimiento para preparar derivados de 8-fenilxantina
ES554567A0 (es) Un procedimiento para preparar derivados de 8-amino-purina
PT80237B (pt) Processo para a metilacao selectiva de derivados de eritromicina a
PT81463B (pt) Processo para a preparacao de novos derivados 5-amino-4-hidroxivalerilo
PT82710B (pt) Processo para a preparacao de derivados la-7-substituidos de mitomicina
PT83073B (pt) Processo para a preparacao de novos derivados da guanina
PT83835B (pt) Processo para a preparacao de novos derivados de calcitonina
PT82769B (pt) Processo para a preparacao de derivados de acidos tiazolidino-4(s)-caboxilicos
BR8600542A (pt) Processo para a obtencao de eteraminas terciarias
ES557183A0 (es) Un metodo para preparar derivados de cefem
ES557006A0 (es) Un metodo para preparar 6-hidroxi-2-acetilnaftaleno
PT83820B (pt) Processo para a preparacao de derivados de tioxantona
PT82445B (pt) Processo para a preparacao de novos derivados glicopeptidicos
PT88180A (pt) Processo para a preparacao de derivados alquilaminoalcoxifenilo
ES551064A0 (es) Un metodo para preparar derivados de cefem
BR8602643A (pt) Processo para preparar compostos
PT82245B (pt) Processo para a preparacao de 2-amino-6-cloropurina
ES552617A0 (es) Un procedimiento para preparar derivados de bencimidazol
ES554238A0 (es) Un precedimiento para preparar derivados de ciclopentil-eter
PT96322A (pt) Processo para a preparacao de derivados de glicerol
PT94008A (pt) Processo para a preparacao de novos derivados de tieno-triazolo-diazepina
ES550467A0 (es) Un metodo para preparar derivados de 9-bencilpurina

Legal Events

Date Code Title Description
MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 19911029