MX23672A - Derivados de glicopeptidos y procedimiento para su preparacion. - Google Patents

Derivados de glicopeptidos y procedimiento para su preparacion.

Info

Publication number
MX23672A
MX23672A MX2367290A MX2367290A MX23672A MX 23672 A MX23672 A MX 23672A MX 2367290 A MX2367290 A MX 2367290A MX 2367290 A MX2367290 A MX 2367290A MX 23672 A MX23672 A MX 23672A
Authority
MX
Mexico
Prior art keywords
glycopeptides
derivatives
procedure
preparation
Prior art date
Application number
MX2367290A
Other languages
English (en)
Inventor
Ramakrishnan Nagarajan
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of MX23672A publication Critical patent/MX23672A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
MX2367290A 1989-12-13 1990-12-10 Derivados de glicopeptidos y procedimiento para su preparacion. MX23672A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US44917189A 1989-12-13 1989-12-13

Publications (1)

Publication Number Publication Date
MX23672A true MX23672A (es) 1993-11-01

Family

ID=23783157

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2367290A MX23672A (es) 1989-12-13 1990-12-10 Derivados de glicopeptidos y procedimiento para su preparacion.

Country Status (20)

Country Link
US (1) US5591714A (es)
EP (1) EP0435503B1 (es)
JP (1) JP3590638B2 (es)
KR (1) KR910011896A (es)
CN (1) CN1034506C (es)
CA (1) CA2031803C (es)
DE (1) DE69033087T2 (es)
ES (1) ES2131496T3 (es)
FI (1) FI906083A7 (es)
HU (1) HUT55802A (es)
IE (1) IE904485A1 (es)
IL (1) IL96603A (es)
MX (1) MX23672A (es)
NO (1) NO303692B1 (es)
NZ (1) NZ236393A (es)
PH (1) PH27373A (es)
PT (1) PT96139B (es)
RU (2) RU2041237C1 (es)
YU (1) YU234790A (es)
ZA (1) ZA909847B (es)

Families Citing this family (45)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW213468B (es) * 1991-06-29 1993-09-21 Hoechst Ag
US5721208A (en) * 1991-06-29 1998-02-24 Hoechst Aktiengesellschaft Glycopeptides a process for their preparation and their use
AU703106B2 (en) * 1994-01-28 1999-03-18 Eli Lilly And Company Glycopeptide antibiotic derivatives
US5840684A (en) * 1994-01-28 1998-11-24 Eli Lilly And Company Glycopeptide antibiotic derivatives
DE19512484A1 (de) * 1995-04-04 1996-10-17 Bayer Ag Kohlenhydratmodifizierte Cytostatika
US5919756A (en) * 1996-06-28 1999-07-06 Eli Lilly And Company Amides
US5939382A (en) * 1996-11-21 1999-08-17 Eli Lilly And Company Reducing agent for reductive alkylation of glycopeptide antibiotics
ID18900A (id) * 1996-11-21 1998-05-20 Lilly Co Eli Alkilasi menurun dari gliko peptida anti biotik
US5952466A (en) * 1997-11-12 1999-09-14 Eli Lilly And Company Reductive alkylation of glycopeptide antibiotics
RU2124022C1 (ru) * 1997-04-10 1998-12-27 Институт биоорганической химии им.М.М.Шемякина и Ю.А.Овчинникова РАН Фуллереновое производное гликопептида, обладающее адъювантной активностью
US5952310A (en) * 1997-05-20 1999-09-14 Eli Lilly And Company Glycopeptide hexapeptides
US5977063A (en) * 1997-05-20 1999-11-02 Eli Lilly And Company Alkylated hexapeptides
US5919771A (en) * 1997-05-20 1999-07-06 Eli Lilly And Company Urea and thiourea derivatives of glycopeptides
US5972933A (en) * 1998-01-08 1999-10-26 Ed. Geistlich Sohne Ag Fur Chemische Industrie Method of treating microbial infections
ATE361931T1 (de) * 1998-05-01 2007-06-15 Lilly Co Eli N1 modifizierte glycopeptide
AU753241C (en) 1998-06-11 2003-05-08 Pharmacia & Upjohn Company Tablet formation
ATE242783T1 (de) * 1998-12-23 2003-06-15 Theravance Inc Glycopeptid-derivate und pharmazeutische zusammensetzungen, die sie enthalten
GB9925127D0 (en) * 1999-10-22 1999-12-22 Pharmacia & Upjohn Spa Oral formulations for anti-tumor compounds
US20020004502A1 (en) * 2000-01-05 2002-01-10 Redmond H. Paul Treatment of inflammatory bowel disease
AU3818001A (en) * 2000-02-11 2001-08-20 Lilly Co Eli Selective n-acylation of a82846 glycopeptide analogs
JP4713810B2 (ja) * 2000-05-02 2011-06-29 セラヴァンス, インコーポレーテッド グリコペプチドに対する還元的アルキル化プロセス
EP1278549B1 (en) * 2000-05-02 2008-12-10 Theravance, Inc. Composition containing a cyclodextrin and a glycopeptide antibiotic
US6770621B2 (en) 2000-05-02 2004-08-03 Theravance, Inc. Polyacid glycopeptide derivatives
EP1154663B1 (en) * 2000-05-09 2008-09-24 Lucent Technologies Inc. Improved quality of service control in a mobile telecommunications network
UA75083C2 (uk) * 2000-06-22 2006-03-15 Тераванс, Інк. Похідні глікопептидфосфонатів
US6828299B2 (en) 2000-06-22 2004-12-07 Theravance, Inc. Polyhydroxy glycopeptide derivatives
US6872804B2 (en) * 2000-06-22 2005-03-29 Theravance, Inc. Glycopeptide disulfide and thioester derivatives
ATE388960T1 (de) 2000-06-22 2008-03-15 Theravance Inc Glykopeptidderivate mit carboxysacchariden
TWI312785B (en) * 2001-08-24 2009-08-01 Theravance Inc Process for preparing vancomycin derivatives
TWI275594B (en) 2001-08-24 2007-03-11 Theravance Inc Process for preparing vancomycin phosphonate derivatives
US20050013854A1 (en) 2003-04-09 2005-01-20 Mannino Raphael J. Novel encochleation methods, cochleates and methods of use
US8778874B2 (en) 2004-11-29 2014-07-15 National University Corporation Nagoya University Glycopeptide antibiotic monomer derivatives
AR053347A1 (es) 2005-04-06 2007-05-02 Astrazeneca Ab Derivados de [1,3]tiazolo[4,5-d]pirimidin-2(3h)-ona 5,7-sustituidos
UA90707C2 (en) 2005-04-06 2010-05-25 Астразенека Аб Novel 5-substituted 7-amino-[1,3]thiazolo[4,5-d]pyrimidine derivatives
EP1926780B1 (en) 2005-09-22 2013-08-14 Medivas, LLC Bis-( -amino)-diol-diester-containing poly(ester amide) and poly(ester urethane) compositions and methods of use
JP5178520B2 (ja) 2005-09-22 2013-04-10 メディバス エルエルシー 固体ポリマー送達組成物およびその使用法
TW200808818A (en) 2006-05-26 2008-02-16 Shionogi & Co Glycopeptide antibiotic derivatives
KR20100109934A (ko) 2007-12-26 2010-10-11 시오노기세야쿠 가부시키가이샤 글리코펩티드 항생 물질 배당화 유도체
US8841440B2 (en) 2008-04-01 2014-09-23 Cornell University Organo-soluble chitosan salts and chitosan-derived biomaterials prepared thereof
CN101928331B (zh) * 2009-06-26 2014-05-28 上海来益生物药物研究开发中心有限责任公司 一种化合物及其应用
JP6347743B2 (ja) 2011-05-05 2018-06-27 マティナス バイオファーマ ナノテクノロジーズ,インコーポレーテッド コクリエート組成物およびその製造および使用方法
CN104418941B (zh) * 2013-08-19 2017-11-07 爱斯医药科技(南京)有限公司 万古霉素衍生物、制备方法及其应用
CA2925005A1 (en) 2013-09-23 2015-03-26 Jawaharlal Nehru Centre for Advanced Scientific Research (JNCASR) Vancomycin-sugar conjugates and uses thereof
HUE070928T2 (hu) * 2014-07-17 2025-07-28 Melinta Therapeutics Llc Nagy tisztaságú oritavancin és eljárás annak elõállítására
CN108409837B (zh) 2018-03-06 2021-09-24 上海来益生物药物研究开发中心有限责任公司 一组具有抗耐药性细菌活性的糖肽类化合物、其制备方法和应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4552701A (en) * 1984-04-16 1985-11-12 Eli Lilly And Company Glycopeptide antibiotics and process of preparation
US4698327A (en) * 1985-04-25 1987-10-06 Eli Lilly And Company Novel glycopeptide derivatives
US4643987A (en) * 1985-08-14 1987-02-17 Eli Lilly And Company Modified glycopeptides
US4639433A (en) * 1985-08-14 1987-01-27 Eli Lilly And Company Glycopeptide derivatives
US4946941A (en) * 1986-01-24 1990-08-07 Shionogi & Co., Ltd. Novel glycopeptide antibiotics
EG18377A (en) * 1986-09-19 1993-04-30 Lilly Co Eli Process for preparing glycopeptide antibiotics
GB8701872D0 (en) * 1987-01-28 1987-03-04 Lepetit Spa N15-alkyl & n15,n15-dialkyl derivatives
US5071749A (en) * 1987-04-16 1991-12-10 Shionogi & Co., Ltd. Glycopetide antibiotic pa-45052-b

Also Published As

Publication number Publication date
KR910011896A (ko) 1991-08-07
EP0435503B1 (en) 1999-05-06
FI906083A0 (fi) 1990-12-11
DE69033087T2 (de) 1999-10-14
IL96603A0 (en) 1991-09-16
US5591714A (en) 1997-01-07
ES2131496T3 (es) 1999-08-01
CA2031803C (en) 2001-05-29
JPH04108800A (ja) 1992-04-09
IL96603A (en) 1998-02-08
NO905354L (no) 1991-06-14
AU633165B2 (en) 1993-01-21
JP3590638B2 (ja) 2004-11-17
CN1052483A (zh) 1991-06-26
DE69033087D1 (de) 1999-06-10
FI906083A7 (fi) 1991-06-14
AU6796490A (en) 1991-06-20
PH27373A (en) 1993-06-21
CN1034506C (zh) 1997-04-09
NO303692B1 (no) 1998-08-17
NO905354D0 (no) 1990-12-11
RU2053240C1 (ru) 1996-01-27
NZ236393A (en) 1992-05-26
HUT55802A (en) 1991-06-28
EP0435503A1 (en) 1991-07-03
YU234790A (sh) 1992-12-21
CA2031803A1 (en) 1991-06-14
PT96139B (pt) 1998-04-30
IE904485A1 (en) 1991-06-19
RU2041237C1 (ru) 1995-08-09
PT96139A (pt) 1991-09-30
ZA909847B (en) 1992-08-26

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