ATE361931T1 - N1 modifizierte glycopeptide - Google Patents

N1 modifizierte glycopeptide

Info

Publication number
ATE361931T1
ATE361931T1 AT99909654T AT99909654T ATE361931T1 AT E361931 T1 ATE361931 T1 AT E361931T1 AT 99909654 T AT99909654 T AT 99909654T AT 99909654 T AT99909654 T AT 99909654T AT E361931 T1 ATE361931 T1 AT E361931T1
Authority
AT
Austria
Prior art keywords
modified glycopeptides
glycopeptides
modified
compounds
useful
Prior art date
Application number
AT99909654T
Other languages
English (en)
Inventor
Richard Thompson
Stephen Wilkie
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Application granted granted Critical
Publication of ATE361931T1 publication Critical patent/ATE361931T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
AT99909654T 1998-05-01 1999-02-26 N1 modifizierte glycopeptide ATE361931T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US8387998P 1998-05-01 1998-05-01

Publications (1)

Publication Number Publication Date
ATE361931T1 true ATE361931T1 (de) 2007-06-15

Family

ID=22181253

Family Applications (1)

Application Number Title Priority Date Filing Date
AT99909654T ATE361931T1 (de) 1998-05-01 1999-02-26 N1 modifizierte glycopeptide

Country Status (10)

Country Link
US (3) US6670446B1 (de)
EP (1) EP1073447B1 (de)
JP (1) JP4307723B2 (de)
AT (1) ATE361931T1 (de)
AU (1) AU2881399A (de)
CA (1) CA2330619A1 (de)
DE (1) DE69936052T2 (de)
DK (1) DK1073447T3 (de)
ES (1) ES2283107T3 (de)
WO (1) WO1999056760A1 (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4307723B2 (ja) * 1998-05-01 2009-08-05 イーライ リリー アンド カンパニー N1−修飾グリコペプチド
WO2000039156A1 (en) 1998-12-23 2000-07-06 Advanced Medicine, Inc. Glycopeptide derivatives and pharmaceutical compositions containing the same
US6518243B1 (en) 1999-04-02 2003-02-11 Trustees Of Princeton University Desleucyl glycopeptide antibiotics and methods of making same
US6699836B2 (en) 1999-04-02 2004-03-02 The Trustees Of Princeton University Vancomycin analogs
PL356966A1 (en) * 2000-02-11 2004-07-12 Eli Lilly And Company Selective n-acylation of a82846 glycopeptide analogs
AR053347A1 (es) 2005-04-06 2007-05-02 Astrazeneca Ab Derivados de [1,3]tiazolo[4,5-d]pirimidin-2(3h)-ona 5,7-sustituidos
UA90707C2 (en) 2005-04-06 2010-05-25 Астразенека Аб Novel 5-substituted 7-amino-[1,3]thiazolo[4,5-d]pyrimidine derivatives
CA2623239C (en) 2005-09-22 2016-07-12 Medivas, Llc Solid polymer delivery compositions and methods for use thereof
CA2623198C (en) 2005-09-22 2014-08-05 Medivas, Llc Bis-(a-amino)-diol-diester-containing poly(ester amide) and poly(ester urethane) compositions and methods of use
US8841440B2 (en) 2008-04-01 2014-09-23 Cornell University Organo-soluble chitosan salts and chitosan-derived biomaterials prepared thereof

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4698327A (en) 1985-04-25 1987-10-06 Eli Lilly And Company Novel glycopeptide derivatives
US4639433A (en) 1985-08-14 1987-01-27 Eli Lilly And Company Glycopeptide derivatives
US4643987A (en) 1985-08-14 1987-02-17 Eli Lilly And Company Modified glycopeptides
EG18377A (en) 1986-09-19 1993-04-30 Lilly Co Eli Process for preparing glycopeptide antibiotics
US5534420A (en) 1988-07-28 1996-07-09 Eli Lilly And Company Biotransformation of glycopeptide antibiotics
IL96603A (en) 1989-12-13 1998-02-08 Lilly Co Eli Antibacterial glycopeptide derivativesProcess for their preparation and pharmaceutical preparations containing the same
RU2145609C1 (ru) 1994-01-28 2000-02-20 Эли Лилли Энд Компани Производные гликопептида или их соли, способ получения, фармацевтическая композиция
US5952310A (en) * 1997-05-20 1999-09-14 Eli Lilly And Company Glycopeptide hexapeptides
JP4307723B2 (ja) 1998-05-01 2009-08-05 イーライ リリー アンド カンパニー N1−修飾グリコペプチド

Also Published As

Publication number Publication date
CA2330619A1 (en) 1999-11-11
DE69936052T2 (de) 2008-01-17
JP2002513764A (ja) 2002-05-14
US6670446B1 (en) 2003-12-30
DK1073447T3 (da) 2007-09-03
US6939947B2 (en) 2005-09-06
EP1073447A4 (de) 2001-10-04
ES2283107T3 (es) 2007-10-16
EP1073447B1 (de) 2007-05-09
US20050037950A1 (en) 2005-02-17
EP1073447A1 (de) 2001-02-07
US20060128609A1 (en) 2006-06-15
AU2881399A (en) 1999-11-23
JP4307723B2 (ja) 2009-08-05
DE69936052D1 (de) 2007-06-21
WO1999056760A1 (en) 1999-11-11

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Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties