PT1140993E - Derivados de glicopeptidos e composicoes farmaceuticas contendo os mesmos - Google Patents

Derivados de glicopeptidos e composicoes farmaceuticas contendo os mesmos

Info

Publication number
PT1140993E
PT1140993E PT99965331T PT99965331T PT1140993E PT 1140993 E PT1140993 E PT 1140993E PT 99965331 T PT99965331 T PT 99965331T PT 99965331 T PT99965331 T PT 99965331T PT 1140993 E PT1140993 E PT 1140993E
Authority
PT
Portugal
Prior art keywords
pharmaceutical compositions
compositions containing
same
derivatives
glycopeptide derivatives
Prior art date
Application number
PT99965331T
Other languages
English (en)
Inventor
Paul Ross Fatheree
J Kevin Judice
Yongqi Mu
Bernice M T Lam
Michael Leadbetter
Martin Sheringham Linsell
Sean Gary Trapp
Guang Yang
Yan Zhu
Original Assignee
Theravance Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Theravance Inc filed Critical Theravance Inc
Publication of PT1140993E publication Critical patent/PT1140993E/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
PT99965331T 1998-12-23 1999-12-22 Derivados de glicopeptidos e composicoes farmaceuticas contendo os mesmos PT1140993E (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US11372898P 1998-12-23 1998-12-23
US12931399P 1999-04-14 1999-04-14
US16402499P 1999-11-04 1999-11-04
US16997899P 1999-12-10 1999-12-10

Publications (1)

Publication Number Publication Date
PT1140993E true PT1140993E (pt) 2003-10-31

Family

ID=27493926

Family Applications (1)

Application Number Title Priority Date Filing Date
PT99965331T PT1140993E (pt) 1998-12-23 1999-12-22 Derivados de glicopeptidos e composicoes farmaceuticas contendo os mesmos

Country Status (23)

Country Link
US (9) US6392012B1 (pt)
EP (1) EP1140993B1 (pt)
JP (1) JP4362017B2 (pt)
KR (1) KR100665204B1 (pt)
CN (1) CN1249081C (pt)
AT (1) ATE242783T1 (pt)
AU (1) AU768204B2 (pt)
BR (1) BRPI9914221B8 (pt)
CA (1) CA2336445C (pt)
CZ (1) CZ301184B6 (pt)
DE (1) DE69908819T2 (pt)
DK (1) DK1140993T3 (pt)
ES (1) ES2201825T3 (pt)
HK (1) HK1040721B (pt)
HU (1) HU230190B1 (pt)
IL (2) IL140093A0 (pt)
NO (1) NO326066B1 (pt)
NZ (1) NZ508594A (pt)
PL (1) PL198311B1 (pt)
PT (1) PT1140993E (pt)
SI (1) SI1140993T1 (pt)
WO (1) WO2000039156A1 (pt)
ZA (1) ZA200007222B (pt)

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DE60136926D1 (de) 2000-05-02 2009-01-22 Theravance Inc Zusammensetzung die eine zyklodextrin und ein glykopeptid-antibiotikum enthält
AU2001259298A1 (en) 2000-05-02 2001-11-12 Advanced Medicine, Inc. Polyacid glycopeptide derivatives
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TWI275594B (en) * 2001-08-24 2007-03-11 Theravance Inc Process for preparing vancomycin phosphonate derivatives
TWI312785B (en) * 2001-08-24 2009-08-01 Theravance Inc Process for preparing vancomycin derivatives
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TWI335332B (en) 2001-10-12 2011-01-01 Theravance Inc Cross-linked vancomycin-cephalosporin antibiotics
US20040033986A1 (en) * 2002-05-17 2004-02-19 Protopopova Marina Nikolaevna Anti tubercular drug: compositions and methods
CN101404986B (zh) 2002-05-17 2011-09-28 赛奎拉公司 用于诊断和治疗感染性疾病的组合物和制药方法
US6878686B2 (en) 2002-05-24 2005-04-12 Theravance, Inc. Cross-linked glycopeptide-cephalosporin antibiotics
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US20060074014A1 (en) * 2002-11-18 2006-04-06 Vicuron Pharmaceuticals Inc. Dalbavancin compositions for treatment of bacterial infections
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US8304597B2 (en) 2004-12-15 2012-11-06 The Procter And Gamble Company Method of using an absorbent article having a functional enhancement indicator
US7368422B2 (en) * 2005-02-28 2008-05-06 Novartis Vaccines And Diagnostics Inc. Semi-synthetic rearranged vancomycin/desmethyl-vancomycin-based glycopeptides with antibiotic activity
US7632918B2 (en) * 2005-02-28 2009-12-15 Novartis Vaccines And Diagnostics, Inc. Semi-synthetic glycopeptides with antibiotic activity
US20070185015A1 (en) * 2005-02-28 2007-08-09 Chiron Corporation and North China Pharmaceutical Corporation Semi-synthetic desmethyl-vancomycin-based glycopeptides with antibiotic activity
CA2623239C (en) 2005-09-22 2016-07-12 Medivas, Llc Solid polymer delivery compositions and methods for use thereof
US8445007B2 (en) 2005-09-22 2013-05-21 Medivas, Llc Bis-(α-amino)-diol-diester-containing poly (ester amide) and poly (ester urethane) compositions and methods of use
WO2007084507A2 (en) * 2006-01-13 2007-07-26 The Scripps Research Institute [ψ[CH2NH]PG4] GLYCOPEPTIDE ANTIBIOTIC ANALOGS
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JP5517153B2 (ja) 2007-12-26 2014-06-11 塩野義製薬株式会社 グリコペプチド抗生物質配糖化誘導体
WO2009123713A1 (en) 2008-04-01 2009-10-08 Cornell University Organo-soluble chitosan salts and chitosan-derived biomaterials prepared thereof
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CN101928330B (zh) * 2009-06-26 2013-10-16 上海来益生物药物研究开发中心有限责任公司 一种新的化合物及其应用
US20140171357A1 (en) * 2011-03-24 2014-06-19 Seachaid Pharmaceuticals, Inc. Vancomycin derivatives
IN2013CH04314A (pt) * 2013-09-23 2015-08-28 Jawaharlal Nehru Ct For Advanced Scient Res Jncasr
EP3240574A1 (en) * 2014-12-25 2017-11-08 Jawaharlal Nehru Centre For Advanced Scientific Research Glycopeptides and uses thereof
WO2017121863A1 (en) * 2016-01-15 2017-07-20 Universität Hamburg Methods for the production of rhamnosylated flavonoids
CA3012176A1 (en) * 2016-01-28 2017-08-03 ACatechol, Inc. Photo-cleavable primer compositions and methods of use
CN107325159A (zh) 2016-04-29 2017-11-07 中国科学院上海药物研究所 一类万古霉素衍生物、其制备方法、药物组合物和用途
AU2018273887B2 (en) * 2017-05-22 2022-09-08 Insmed Incorporated Lipo-glycopeptide cleavable derivatives and uses thereof
CN107987131B (zh) * 2017-11-16 2021-03-09 上海来益生物药物研究开发中心有限责任公司 一组具有抗耐药性细菌活性的化合物、其制备方法和应用
CN108409837B (zh) 2018-03-06 2021-09-24 上海来益生物药物研究开发中心有限责任公司 一组具有抗耐药性细菌活性的糖肽类化合物、其制备方法和应用
NL2023883B1 (en) * 2019-09-24 2021-04-26 Univ Leiden Antibiotic compounds
CN111620931B (zh) * 2020-06-12 2021-12-17 苏州博源医疗科技有限公司 万古霉素衍生物及其制备方法和应用
CN114213284B (zh) * 2022-01-04 2023-08-01 丽珠集团福州福兴医药有限公司 (9h-芴-9-基)-癸基(2-氧代乙基)氨基甲酸甲酯及其合成方法

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UA75083C2 (uk) 2000-06-22 2006-03-15 Тераванс, Інк. Похідні глікопептидфосфонатів
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Also Published As

Publication number Publication date
CZ301184B6 (cs) 2009-12-02
CN1315961A (zh) 2001-10-03
US6949681B2 (en) 2005-09-27
CN1249081C (zh) 2006-04-05
CZ200122A3 (en) 2001-06-13
HUP0400887A2 (hu) 2004-08-30
HUP0400887A3 (en) 2012-09-28
CA2336445C (en) 2011-07-19
NO326066B1 (no) 2008-09-08
ATE242783T1 (de) 2003-06-15
US6455669B1 (en) 2002-09-24
KR20010085857A (ko) 2001-09-07
SI1140993T1 (en) 2003-12-31
IL140093A (en) 2006-06-11
US7101964B2 (en) 2006-09-05
HK1040721A1 (en) 2002-06-21
HK1040721B (zh) 2003-10-17
US7351791B2 (en) 2008-04-01
US20030060598A1 (en) 2003-03-27
AU3127300A (en) 2000-07-31
WO2000039156A1 (en) 2000-07-06
DE69908819D1 (de) 2003-07-17
IL140093A0 (en) 2002-02-10
BR9914221A (pt) 2001-06-26
US7723470B2 (en) 2010-05-25
DE69908819T2 (de) 2004-05-06
NZ508594A (en) 2003-05-30
JP2002533472A (ja) 2002-10-08
AU768204B2 (en) 2003-12-04
CA2336445A1 (en) 2000-07-06
US6444786B1 (en) 2002-09-03
BR9914221B1 (pt) 2013-12-31
US8030445B2 (en) 2011-10-04
US20060241024A1 (en) 2006-10-26
US20090215982A1 (en) 2009-08-27
US6962970B2 (en) 2005-11-08
NO20006323D0 (no) 2000-12-12
EP1140993B1 (en) 2003-06-11
US20080103292A1 (en) 2008-05-01
DK1140993T3 (da) 2003-10-06
US6392012B1 (en) 2002-05-21
PL198311B1 (pl) 2008-06-30
JP4362017B2 (ja) 2009-11-11
HU230190B1 (hu) 2015-09-28
ZA200007222B (en) 2002-03-06
NO20006323L (no) 2001-02-12
KR100665204B1 (ko) 2007-01-04
PL348451A1 (en) 2002-05-20
ES2201825T3 (es) 2004-03-16
EP1140993A1 (en) 2001-10-10
BRPI9914221B8 (pt) 2021-05-25
US20050239690A1 (en) 2005-10-27
US20040204346A1 (en) 2004-10-14

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