PA8513301A1 - Inhibidor del intercambiador de sodio-hidrògeno de tipo 1 - Google Patents

Inhibidor del intercambiador de sodio-hidrògeno de tipo 1

Info

Publication number
PA8513301A1
PA8513301A1 PA20018513301A PA8513301A PA8513301A1 PA 8513301 A1 PA8513301 A1 PA 8513301A1 PA 20018513301 A PA20018513301 A PA 20018513301A PA 8513301 A PA8513301 A PA 8513301A PA 8513301 A1 PA8513301 A1 PA 8513301A1
Authority
PA
Panama
Prior art keywords
inhibitor
sodium
type
hydrogen exchanger
nhe
Prior art date
Application number
PA20018513301A
Other languages
English (en)
Spanish (es)
Inventor
Weichao George Chen
Eric David Cox
Angel Guzman-Perez
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of PA8513301A1 publication Critical patent/PA8513301A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Epidemiology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Treatment Of Water By Ion Exchange (AREA)
  • Preventing Corrosion Or Incrustation Of Metals (AREA)
  • Plural Heterocyclic Compounds (AREA)
PA20018513301A 2000-04-28 2001-03-12 Inhibidor del intercambiador de sodio-hidrògeno de tipo 1 PA8513301A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US20043200P 2000-04-28 2000-04-28

Publications (1)

Publication Number Publication Date
PA8513301A1 true PA8513301A1 (es) 2003-09-05

Family

ID=22741697

Family Applications (1)

Application Number Title Priority Date Filing Date
PA20018513301A PA8513301A1 (es) 2000-04-28 2001-03-12 Inhibidor del intercambiador de sodio-hidrògeno de tipo 1

Country Status (40)

Country Link
EP (1) EP1276737A1 (is)
JP (1) JP2003531900A (is)
KR (1) KR20020093079A (is)
CN (1) CN1225466C (is)
AP (1) AP2002002651A0 (is)
AR (1) AR028375A1 (is)
AU (1) AU2001235896A1 (is)
BG (1) BG107139A (is)
BR (1) BR0110268A (is)
CA (1) CA2407535A1 (is)
CO (1) CO5221125A1 (is)
CR (1) CR6797A (is)
CZ (1) CZ20023408A3 (is)
DZ (1) DZ3310A1 (is)
EA (1) EA004882B1 (is)
EE (1) EE200200615A (is)
GT (1) GT200100064A (is)
HN (1) HN2001000042A (is)
HR (1) HRP20020851A2 (is)
HU (1) HUP0300651A2 (is)
IL (1) IL152075A0 (is)
IS (2) IS6567A (is)
MA (1) MA26897A1 (is)
MX (1) MXPA02010600A (is)
MY (1) MY133842A (is)
NO (1) NO20025132L (is)
NZ (1) NZ521348A (is)
OA (1) OA12256A (is)
PA (1) PA8513301A1 (is)
PE (1) PE20011270A1 (is)
PL (1) PL357765A1 (is)
SK (1) SK14872002A3 (is)
SV (1) SV2002000418A (is)
TN (1) TNSN01065A1 (is)
TR (1) TR200202439T2 (is)
UA (1) UA73348C2 (is)
UY (1) UY26680A1 (is)
WO (1) WO2001083470A1 (is)
YU (1) YU79602A (is)
ZA (1) ZA200208605B (is)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR0116841A (pt) * 2001-01-31 2004-02-25 Pfizer Producs Inc Etanolatos de inibidor de permutador sódio-hidrogênio do tipo-1
MXPA04004685A (es) * 2001-12-19 2004-08-12 Pfizer Prod Inc Procedimientos para preparar inhibidores de tipo-1 de intercambiador sodio-hidrogeno.
MXPA04008646A (es) * 2002-05-02 2004-12-06 Pfizer Prod Inc Tratamiento para la diabetes y complicaciones diabeticas con inhibidores del nhe-1.
FR2840302B1 (fr) * 2002-06-03 2004-07-16 Aventis Pharma Sa Derives d'isoindolones, procede de preparation et intermediaire de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant
ES2220185B1 (es) * 2002-07-16 2006-04-01 Consejo Sup. De Investig. Cientificas Nuevo peptido inhibidor del intercambiador na+/h+ (pinhe), y sus aplicaciones.
EP1596860A4 (en) * 2003-02-14 2009-05-27 Smithkline Beecham Corp NEW CONNECTIONS
RU2518741C1 (ru) * 2013-03-22 2014-06-10 Федеральное государственное автономное образовательное учреждение высшего профессионального образования "ЮЖНЫЙ ФЕДЕРАЛЬНЫЙ УНИВЕРСИТЕТ" СРЕДСТВО, ИНГИБИРУЮЩЕЕ Na+/H+-ОБМЕН, И ГАЛОГЕНИДЫ 1-ДИАЛКИЛАМИНОЭТИЛ-3-[ЗАМЕЩЕННЫЙ(ДИЗАМЕЩЕННЫЙ) ФЕНАЦИЛ]-2-АМИНОБЕНЗИМИДАЗОЛИЯ

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2237080T3 (es) * 1998-02-27 2005-07-16 Pfizer Products Inc. Derivados de n-((anillo di- o triaza dinsaturado de cinco miembros sustituido)carbonil)guanidina para el tratamiento de isquemia.

Also Published As

Publication number Publication date
NZ521348A (en) 2004-09-24
HN2001000042A (es) 2001-07-09
HRP20020851A2 (en) 2005-02-28
MA26897A1 (fr) 2004-12-20
YU79602A (en) 2006-05-25
SV2002000418A (es) 2002-07-03
DZ3310A1 (fr) 2001-11-07
MY133842A (en) 2007-11-30
EA200201023A1 (ru) 2003-02-27
EE200200615A (et) 2004-04-15
CA2407535A1 (en) 2001-11-08
IL152075A0 (en) 2003-05-29
CZ20023408A3 (cs) 2004-01-14
IS6567A (is) 2002-09-24
KR20020093079A (ko) 2002-12-12
CN1225466C (zh) 2005-11-02
SK14872002A3 (sk) 2004-03-02
GT200100064A (es) 2002-03-22
OA12256A (en) 2003-11-06
PE20011270A1 (es) 2001-12-12
ZA200208605B (en) 2003-10-24
BG107139A (bg) 2003-07-31
UA73348C2 (en) 2005-07-15
EA004882B1 (ru) 2004-08-26
WO2001083470A1 (en) 2001-11-08
NO20025132L (no) 2002-12-12
JP2003531900A (ja) 2003-10-28
TR200202439T2 (tr) 2003-02-21
CR6797A (es) 2004-05-17
HUP0300651A2 (hu) 2003-07-28
MXPA02010600A (es) 2003-03-10
PL357765A1 (en) 2004-07-26
AP2002002651A0 (en) 2002-12-31
NO20025132D0 (no) 2002-10-25
BR0110268A (pt) 2003-12-30
UY26680A1 (es) 2001-12-28
CO5221125A1 (es) 2002-11-28
AU2001235896A1 (en) 2001-11-12
EP1276737A1 (en) 2003-01-22
IS6588A (is) 2002-10-21
TNSN01065A1 (fr) 2005-11-10
CN1426404A (zh) 2003-06-25
AR028375A1 (es) 2003-05-07

Similar Documents

Publication Publication Date Title
PA8468401A1 (es) Compuestos para el tratamiento de la isquemia
ES2195970T3 (es) L-ribavirina y usos de la misma.
ES2145638T3 (es) Nuevos compuestos azoicos, utilizacion para tincion, composiciones que los contienen y procedimientos de tincion.
GT199900150A (es) 1,2,3,4-tetrahidroquinolinas 2-sustituidas 4-carboxiamino sustituidas.
ES2157027T3 (es) Oxazolidinonas sustituidas y su uso como farmacos antibacterianos.
BR9913745A (pt) Cetonas de piridina úteis como herbicidas
ES2191183T3 (es) Derivados 6,6- o 6,7-biciclicos que contienen pirido o pirimido sustituidos.
ECSP055747A (es) Antagonistas de cgrp elegidos, procedimiento para su preparación, así como su empleo como medicamentos
GT199900067A (es) Nuevas 4-fenilpiperidinas para el tratamiento dedermatosis prurìtica.
ES2179337T3 (es) Disulfuros de triazolilo.
MX9307232A (es) Arilcicloalquilaminas n,n-disustituidas, sus sales, medicamentos que contiene estos compuestos y su empleo, asi como procedimientos para su preparacion.
PA8586801A1 (es) Inhibidores de hiv-integrasa, composiciones farmaceuticas y metodos para su uso
AR018162A1 (es) Pirroles substituidos, composicion farmaceutica y el uso de los mismos para la preparacion de dicha composicion farmaceutica
UY27203A1 (es) Bencimidazoles útiles en el tratamiento de la disfunción sexual
AR020563A1 (es) Compuestos (poli)tia-alquinoicos y sus derivados, composiciones que los incluyen y su utilizacion
PA8513301A1 (es) Inhibidor del intercambiador de sodio-hidrògeno de tipo 1
AR030537A1 (es) Acidos quinolincarboxilicos y naftiridincarboxilico antibacterianos
CU23269A3 (es) Bromhidrato de eletriptan monohidratado
GT199900113A (es) Inhibidores de las fkbp.
ES2189072T3 (es) Nuevo benzo-cicloalquenos heterociclicos, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen.
AR006675A1 (es) 4-benzoilisotiazoles herbicidas, procedimiento para obtenerlas, las composiciones herbicidas que las contienen y el procedimiento de aplicacionde dichos compuestos.
AR025797A1 (es) Quinazolinonas
TR200201167T2 (tr) Sodyum-hidrojen değiştirici tip 1 önleyici kristalleri.
UY26417A1 (es) Cristales de inhibidor del intercambiador de sodio-hidrógeno tipo 1
BR0005122A (pt) Método para a preparação de inibidor de permutador de sódio-hidrogênio do tipo 1