OA11592A - Substituted imidazo!1,2aÜazines as selective inhibitors of cox-2. - Google Patents

Substituted imidazo!1,2aÜazines as selective inhibitors of cox-2. Download PDF

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Publication number
OA11592A
OA11592A OA1200100033A OA1200100033A OA11592A OA 11592 A OA11592 A OA 11592A OA 1200100033 A OA1200100033 A OA 1200100033A OA 1200100033 A OA1200100033 A OA 1200100033A OA 11592 A OA11592 A OA 11592A
Authority
OA
OAPI
Prior art keywords
imidazo
methylsulfonylphenyl
pyridine
pyrimidine
aminosulfonylphenyl
Prior art date
Application number
OA1200100033A
Other languages
English (en)
Inventor
Gallemi Carles Farrerons
Ignacio-Jose Miquel Bono
Ana Maria Fernandez Serrat
Carlos Monserrat Vidal
Carmen Lagunas Arnal
Ferran Gimenez Guasch
Andres Fernandez Garcia
Original Assignee
Salvat Lab Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Salvat Lab Sa filed Critical Salvat Lab Sa
Publication of OA11592A publication Critical patent/OA11592A/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
OA1200100033A 1998-08-03 1999-07-23 Substituted imidazo!1,2aÜazines as selective inhibitors of cox-2. OA11592A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES009801652A ES2140354B1 (es) 1998-08-03 1998-08-03 Imidazo (1,2a) azinas sustituidas como inhibidores selectivos de la cox-2.

Publications (1)

Publication Number Publication Date
OA11592A true OA11592A (en) 2004-07-30

Family

ID=8304755

Family Applications (1)

Application Number Title Priority Date Filing Date
OA1200100033A OA11592A (en) 1998-08-03 1999-07-23 Substituted imidazo!1,2aÜazines as selective inhibitors of cox-2.

Country Status (31)

Country Link
US (1) US6670365B1 (da)
EP (1) EP1104762B1 (da)
JP (1) JP2002522438A (da)
KR (1) KR20010079602A (da)
CN (1) CN1131865C (da)
AP (1) AP2001002082A0 (da)
AT (1) ATE224391T1 (da)
AU (1) AU749770B2 (da)
BG (1) BG105299A (da)
BR (1) BR9912968A (da)
CA (1) CA2339187A1 (da)
CZ (1) CZ291783B6 (da)
DE (1) DE69903046T2 (da)
DK (1) DK1104762T3 (da)
EA (1) EA003399B1 (da)
ES (2) ES2140354B1 (da)
HK (1) HK1037629A1 (da)
HU (1) HUP0103004A3 (da)
ID (1) ID28539A (da)
IL (1) IL141242A0 (da)
MX (1) MXPA01001332A (da)
NO (1) NO20010568L (da)
NZ (1) NZ510196A (da)
OA (1) OA11592A (da)
PL (1) PL345804A1 (da)
PT (1) PT1104762E (da)
SK (1) SK1662001A3 (da)
TR (1) TR200100359T2 (da)
WO (1) WO2000008024A1 (da)
YU (1) YU7401A (da)
ZA (1) ZA200101632B (da)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8241622B2 (en) * 2001-07-13 2012-08-14 University Of Iowa Research Foundation Adeno-associated virus vectors with intravector heterologous terminal palindromic sequences
US20030100594A1 (en) * 2001-08-10 2003-05-29 Pharmacia Corporation Carbonic anhydrase inhibitor
DE10247271A1 (de) * 2002-10-10 2004-08-26 Grünenthal GmbH Substituierte C-Imidazo[1,2-a]pyridin-3-yle
DE10256881A1 (de) * 2002-12-05 2004-06-24 Beiersdorf Ag Neue topische Verwendung von Bis-Arylimidazo[1,2-a]thiolanderivaten
EP1534305B9 (en) 2003-05-07 2007-03-07 Osteologix A/S Treating cartilage / bone conditions with water-soluble strontium salts
CN1860121A (zh) * 2003-07-30 2006-11-08 S.A.L.V.A.T.实验室有限公司 用于预防和治疗癌症的取代咪唑并嘧啶
WO2007034278A2 (en) * 2005-09-19 2007-03-29 Pfizer Products Inc. Fused imidazole derivatives as c3a receptor antagonists
US20070265350A1 (en) * 2005-12-30 2007-11-15 University Of Iowa Research Foundation Method of identifying compounds useful to treat neuronal degenerative diseases
WO2007096764A2 (en) * 2006-02-27 2007-08-30 Glenmark Pharmaceuticals S.A. Bicyclic heteroaryl derivatives as cannabinoid receptor modulators
US8785486B2 (en) * 2007-11-14 2014-07-22 Janssen Pharmaceuticals, Inc. Imidazo[1,2-A]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors
CA2739303A1 (en) * 2008-10-01 2010-04-08 Synta Pharmaceuticals Corp. Compounds for inflammation and immune-related uses
GB201321732D0 (en) * 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents
US11702672B2 (en) 2016-02-08 2023-07-18 University Of Iowa Research Foundation Methods to produce chimeric adeno-associated virus/bocavirus parvovirus
US11684679B2 (en) 2016-03-07 2023-06-27 University Of Iowa Research Foundation AAV-mediated expression using a synthetic promoter and enhancer
CA3209491A1 (en) 2021-03-15 2022-09-22 Saul Yedgar Hyaluronic acid-conjugated dipalmitoyl phosphatidyl ethanolamine in combination with non-steroidal anti-inflammatory drugs (nsaids) for treating or alleviating inflammatory disease

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2785133A (en) * 1954-03-26 1957-03-12 Gen Aniline & Film Corp Compositions for a method of whitening fine fabrics
US3455924A (en) * 1967-02-08 1969-07-15 Upjohn Co Dianisylimidazoles
JPH06504779A (ja) * 1990-12-13 1994-06-02 スミスクライン・ビーチャム・コーポレイション 新規csaids
WO1993019066A1 (en) * 1992-03-17 1993-09-30 Nippon Shinyaku Co., Ltd. Imidazopyridine derivative and medicine
US5620999A (en) 1994-07-28 1997-04-15 Weier; Richard M. Benzenesulfonamide subtituted imidazolyl compounds for the treatment of inflammation
CN1186492A (zh) * 1995-04-04 1998-07-01 葛兰素集团有限公司 咪唑并[1,2-α]吡啶衍生物
UA57002C2 (uk) * 1995-10-13 2003-06-16 Мерк Фросст Кенада Енд Ко./Мерк Фросст Кенада Енд Сі. Похідне (метилсульфоніл)феніл-2-(5н)-фуранону, фармацевтична композиція та спосіб лікування

Also Published As

Publication number Publication date
AU749770B2 (en) 2002-07-04
DK1104762T3 (da) 2002-10-21
AP2001002082A0 (en) 2001-03-31
KR20010079602A (ko) 2001-08-22
SK1662001A3 (en) 2001-08-06
PL345804A1 (en) 2002-01-02
CN1131865C (zh) 2003-12-24
BG105299A (en) 2001-11-30
ZA200101632B (en) 2001-08-30
YU7401A (sh) 2003-10-31
ATE224391T1 (de) 2002-10-15
CZ291783B6 (cs) 2003-05-14
MXPA01001332A (es) 2002-11-29
BR9912968A (pt) 2001-05-08
HUP0103004A3 (en) 2003-03-28
ES2140354B1 (es) 2000-11-01
JP2002522438A (ja) 2002-07-23
US6670365B1 (en) 2003-12-30
EA003399B1 (ru) 2003-04-24
DE69903046T2 (de) 2003-05-22
HUP0103004A2 (hu) 2002-01-28
NO20010568D0 (no) 2001-02-02
EA200100212A1 (ru) 2001-08-27
CZ2001433A3 (cs) 2001-08-15
CA2339187A1 (en) 2000-02-17
TR200100359T2 (tr) 2001-06-21
EP1104762B1 (en) 2002-09-18
ES2182546T3 (es) 2003-03-01
ID28539A (id) 2001-05-31
EP1104762A1 (en) 2001-06-06
WO2000008024A1 (es) 2000-02-17
ES2140354A1 (es) 2000-02-16
NZ510196A (en) 2002-09-27
CN1321157A (zh) 2001-11-07
NO20010568L (no) 2001-04-02
HK1037629A1 (en) 2002-02-15
AU4782499A (en) 2000-02-28
IL141242A0 (en) 2002-03-10
DE69903046D1 (de) 2002-10-24
PT1104762E (pt) 2002-11-29

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