NZ604018A - Furanyl compounds and the use thereof - Google Patents
Furanyl compounds and the use thereofInfo
- Publication number
- NZ604018A NZ604018A NZ604018A NZ60401811A NZ604018A NZ 604018 A NZ604018 A NZ 604018A NZ 604018 A NZ604018 A NZ 604018A NZ 60401811 A NZ60401811 A NZ 60401811A NZ 604018 A NZ604018 A NZ 604018A
- Authority
- NZ
- New Zealand
- Prior art keywords
- compounds
- amelioration
- prevention
- treatment
- furanyl
- Prior art date
Links
- 125000002541 furyl group Chemical group 0.000 title abstract 3
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 3
- 206010028980 Neoplasm Diseases 0.000 abstract 2
- 201000011510 cancer Diseases 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 230000000694 effects Effects 0.000 abstract 2
- 238000000034 method Methods 0.000 abstract 2
- 230000002265 prevention Effects 0.000 abstract 2
- 230000002062 proliferating effect Effects 0.000 abstract 2
- 101001082110 Acanthamoeba polyphaga mimivirus Eukaryotic translation initiation factor 4E homolog Proteins 0.000 abstract 1
- 101001082109 Danio rerio Eukaryotic translation initiation factor 4E-1B Proteins 0.000 abstract 1
- 241000027355 Ferocactus setispinus Species 0.000 abstract 1
- 239000002246 antineoplastic agent Substances 0.000 abstract 1
- 229940041181 antineoplastic drug Drugs 0.000 abstract 1
- 238000009169 immunotherapy Methods 0.000 abstract 1
- 230000037361 pathway Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 238000001959 radiotherapy Methods 0.000 abstract 1
- 238000001356 surgical procedure Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A61K31/341—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Oncology (AREA)
- Hematology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Furan Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US35230810P | 2010-06-07 | 2010-06-07 | |
| PCT/US2011/039377 WO2011156321A1 (en) | 2010-06-07 | 2011-06-07 | Furanyl compounds and the use thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NZ604018A true NZ604018A (en) | 2015-02-27 |
Family
ID=44210539
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NZ604018A NZ604018A (en) | 2010-06-07 | 2011-06-07 | Furanyl compounds and the use thereof |
Country Status (11)
| Country | Link |
|---|---|
| US (3) | US8722731B2 (cg-RX-API-DMAC7.html) |
| EP (1) | EP2576532B1 (cg-RX-API-DMAC7.html) |
| JP (1) | JP5855095B2 (cg-RX-API-DMAC7.html) |
| CN (2) | CN103108868B (cg-RX-API-DMAC7.html) |
| AU (1) | AU2011265047B2 (cg-RX-API-DMAC7.html) |
| CA (1) | CA2801778C (cg-RX-API-DMAC7.html) |
| MX (2) | MX367469B (cg-RX-API-DMAC7.html) |
| NZ (1) | NZ604018A (cg-RX-API-DMAC7.html) |
| SG (1) | SG186229A1 (cg-RX-API-DMAC7.html) |
| WO (1) | WO2011156321A1 (cg-RX-API-DMAC7.html) |
| ZA (1) | ZA201209237B (cg-RX-API-DMAC7.html) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5855095B2 (ja) | 2010-06-07 | 2016-02-09 | ノボメディックス, エルエルシーNovomedix, Llc | フラニル化合物およびその使用 |
| EP2897607B1 (en) * | 2012-09-21 | 2017-11-22 | Rhode Island Hospital | Inhibitors of beta-hydrolase for treatment of cancer |
| WO2014085633A1 (en) | 2012-11-30 | 2014-06-05 | Novomedix, Llc | Substituted biaryl sulfonamides and the use thereof |
| US10335493B2 (en) * | 2013-12-10 | 2019-07-02 | Emory University | Targeted protease compositions and uses related thereto |
| EP3102703A2 (en) | 2014-02-07 | 2016-12-14 | Effector Therapeutics Inc. | Methods for treating fibrotic disease |
| US10548908B2 (en) * | 2016-09-15 | 2020-02-04 | Nostopharma, LLC | Compositions and methods for preventing and treating heterotopic ossification and pathologic calcification |
| EP4114529A1 (en) * | 2020-03-03 | 2023-01-11 | PIC Therapeutics, Inc. | Eif4e inhibitors and uses thereof |
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- 2011-06-07 CN CN201510161879.2A patent/CN104860907A/zh active Pending
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Also Published As
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|---|---|
| CN103108868A (zh) | 2013-05-15 |
| US20140309297A1 (en) | 2014-10-16 |
| CN103108868B (zh) | 2015-11-25 |
| MX2012014273A (es) | 2013-03-22 |
| AU2011265047B2 (en) | 2014-10-23 |
| CN104860907A (zh) | 2015-08-26 |
| SG186229A1 (en) | 2013-01-30 |
| US9663483B2 (en) | 2017-05-30 |
| WO2011156321A9 (en) | 2012-04-05 |
| CA2801778C (en) | 2018-06-05 |
| JP5855095B2 (ja) | 2016-02-09 |
| US20160024040A1 (en) | 2016-01-28 |
| US8722731B2 (en) | 2014-05-13 |
| EP2576532A1 (en) | 2013-04-10 |
| US20130116317A1 (en) | 2013-05-09 |
| EP2576532B1 (en) | 2018-07-18 |
| WO2011156321A1 (en) | 2011-12-15 |
| ZA201209237B (en) | 2015-05-27 |
| US9149527B2 (en) | 2015-10-06 |
| AU2011265047A1 (en) | 2013-01-10 |
| MX367469B (es) | 2019-08-23 |
| CA2801778A1 (en) | 2011-12-15 |
| JP2013528215A (ja) | 2013-07-08 |
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