NZ566010A - 3, 11b-cis-dihydrotetrabenazine for the treatment of an inflammatory disease - Google Patents
3, 11b-cis-dihydrotetrabenazine for the treatment of an inflammatory diseaseInfo
- Publication number
- NZ566010A NZ566010A NZ566010A NZ56601006A NZ566010A NZ 566010 A NZ566010 A NZ 566010A NZ 566010 A NZ566010 A NZ 566010A NZ 56601006 A NZ56601006 A NZ 56601006A NZ 566010 A NZ566010 A NZ 566010A
- Authority
- NZ
- New Zealand
- Prior art keywords
- dihydrotetrabenazine
- isomer
- pct
- isomers
- cells
- Prior art date
Links
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- A61K31/47—Quinolines; Isoquinolines
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Landscapes
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- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
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Applications Claiming Priority (2)
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| GBGB0516168.2A GB0516168D0 (en) | 2005-08-05 | 2005-08-05 | Pharmaceutical compounds |
| PCT/GB2006/002909 WO2007017643A1 (en) | 2005-08-05 | 2006-08-04 | 3 , llB-CIS-DIHYDROTETRABENAZINE FOR THE TREATMENT OF A PROLIFERATIVE DISEASE OR AN INFLAMMATION |
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| NZ566010A true NZ566010A (en) | 2010-05-28 |
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| NZ566010A NZ566010A (en) | 2005-08-05 | 2006-08-04 | 3, 11b-cis-dihydrotetrabenazine for the treatment of an inflammatory disease |
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| EP (2) | EP1861100B1 (enExample) |
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| MX (1) | MX2008001546A (enExample) |
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| PL (1) | PL1861100T3 (enExample) |
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| SI (1) | SI1861100T1 (enExample) |
| WO (1) | WO2007017643A1 (enExample) |
| ZA (2) | ZA200801171B (enExample) |
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| GB0514501D0 (en) * | 2005-07-14 | 2005-08-24 | Cambridge Lab Ireland Ltd | Pharmaceutical compounds |
| AU2007317242B2 (en) | 2006-11-08 | 2013-08-01 | Neurocrine Biosciences, Inc. | Substituted 3-isobutyl-9, 10-dimethoxy-1,3,4,6,7,11B-hexahydro-2H-pyrido[2,1-a] isoquinolin-2-ol compounds and methods relating thereto |
| GB0721669D0 (en) * | 2007-11-02 | 2007-12-12 | Cambridge Lab Ireland Ltd | Pharmaceutical compounds |
| GB0810857D0 (en) * | 2008-06-13 | 2008-07-23 | Cambridge Lab Ireland Ltd | Pharmaceutical compounds |
| GB2462611A (en) * | 2008-08-12 | 2010-02-17 | Cambridge Lab | Pharmaceutical composition comprising tetrabenazine |
| US20110053866A1 (en) * | 2008-08-12 | 2011-03-03 | Biovail Laboratories International (Barbados) S.R.L. | Pharmaceutical compositions |
| GB2463452A (en) * | 2008-09-08 | 2010-03-17 | Cambridge Lab | Desmethyl derivatives of tetrabenazine and pharmaceutical compositions thereof |
| GB2463451A (en) | 2008-09-08 | 2010-03-17 | Cambridge Lab | 3, 11b cis-dihydrotetrabenazine compounds for use in the treatment of dementia |
| GB2463283A (en) * | 2008-09-08 | 2010-03-10 | Cambridge Lab | 3,11b-cis-dihydrotetrabenazine for use in treating asthma |
| WO2011153157A2 (en) | 2010-06-01 | 2011-12-08 | Auspex Pharmaceutical, Inc. | Benzoquinolone inhibitors of vmat2 |
| CN102285984B (zh) * | 2010-11-25 | 2012-10-10 | 江苏威凯尔医药科技有限公司 | (2R,3R,11bR)-二氢丁苯那嗪及相关化合物的制备方法 |
| MX2016009817A (es) | 2014-01-27 | 2017-02-28 | Auspex Pharmaceuticals Inc | Inhibidores de benzoquinolina del transportador vesicular de monoaminas 2. |
| MA41177A (fr) * | 2014-12-15 | 2017-10-24 | Esteve Labor Dr | Utilisation de ligands des récepteurs sigma dans l'arthrose |
| US10550120B2 (en) | 2016-03-25 | 2020-02-04 | Tohoku University | Indole alkaloid compound having immune checkpoint inhibitory action |
| CN109283279B (zh) * | 2017-07-21 | 2019-11-01 | 南京正大天晴制药有限公司 | 通过高效液相色谱法分离测定雷替曲塞及其对映异构体的方法 |
| CN109283263B (zh) * | 2017-07-21 | 2019-06-25 | 南京正大天晴制药有限公司 | 用于雷替曲塞合成质量控制的检测分析方法 |
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-
2005
- 2005-08-05 GB GBGB0516168.2A patent/GB0516168D0/en not_active Ceased
-
2006
- 2006-08-04 EP EP06765213A patent/EP1861100B1/en active Active
- 2006-08-04 CA CA002620952A patent/CA2620952A1/en not_active Abandoned
- 2006-08-04 ZA ZA200801171A patent/ZA200801171B/xx unknown
- 2006-08-04 JP JP2008524588A patent/JP2009503045A/ja active Pending
- 2006-08-04 MX MX2008001546A patent/MX2008001546A/es active IP Right Grant
- 2006-08-04 US US11/997,675 patent/US20090275605A1/en not_active Abandoned
- 2006-08-04 HR HR20090017T patent/HRP20090017T3/xx unknown
- 2006-08-04 EP EP08104275A patent/EP1964565A1/en not_active Withdrawn
- 2006-08-04 AU AU2006277836A patent/AU2006277836B8/en not_active Expired - Fee Related
- 2006-08-04 ZA ZA200801170A patent/ZA200801170B/xx unknown
- 2006-08-04 NZ NZ566010A patent/NZ566010A/en not_active IP Right Cessation
- 2006-08-04 SI SI200630187T patent/SI1861100T1/sl unknown
- 2006-08-04 KR KR1020087005309A patent/KR20080033501A/ko not_active Withdrawn
- 2006-08-04 DE DE602006003415T patent/DE602006003415D1/de active Active
- 2006-08-04 PL PL06765213T patent/PL1861100T3/pl unknown
- 2006-08-04 PT PT06765213T patent/PT1861100E/pt unknown
- 2006-08-04 WO PCT/GB2006/002909 patent/WO2007017643A1/en not_active Ceased
- 2006-08-04 CN CN2006800366007A patent/CN101321528B/zh not_active Expired - Fee Related
- 2006-08-04 DK DK06765213T patent/DK1861100T3/da active
- 2006-08-04 RU RU2008108516/15A patent/RU2409364C2/ru not_active IP Right Cessation
- 2006-08-04 ES ES06765213T patent/ES2317564T3/es active Active
- 2006-08-04 RS RSP-2009/0015A patent/RS50720B/sr unknown
- 2006-08-04 AT AT06765213T patent/ATE412414T1/de active
-
2009
- 2009-01-27 CY CY20091100100T patent/CY1108729T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| PT1861100E (pt) | 2008-12-26 |
| ZA200801170B (en) | 2009-12-30 |
| RU2409364C2 (ru) | 2011-01-20 |
| PL1861100T3 (pl) | 2009-06-30 |
| CN101321528A (zh) | 2008-12-10 |
| AU2006277836A1 (en) | 2007-02-15 |
| KR20080033501A (ko) | 2008-04-16 |
| EP1861100B1 (en) | 2008-10-29 |
| CY1108729T1 (el) | 2014-04-09 |
| CA2620952A1 (en) | 2007-02-15 |
| CN101321528B (zh) | 2011-05-25 |
| GB0516168D0 (en) | 2005-09-14 |
| RS50720B (sr) | 2010-08-31 |
| DE602006003415D1 (de) | 2008-12-11 |
| MX2008001546A (es) | 2008-04-04 |
| EP1964565A1 (en) | 2008-09-03 |
| DK1861100T3 (da) | 2008-12-15 |
| WO2007017643A1 (en) | 2007-02-15 |
| EP1861100A1 (en) | 2007-12-05 |
| JP2009503045A (ja) | 2009-01-29 |
| US20090275605A1 (en) | 2009-11-05 |
| HK1111084A1 (en) | 2008-08-01 |
| RU2008108516A (ru) | 2009-09-10 |
| AU2006277836B8 (en) | 2011-12-08 |
| ZA200801171B (en) | 2009-08-26 |
| ATE412414T1 (de) | 2008-11-15 |
| HRP20090017T3 (hr) | 2009-03-31 |
| SI1861100T1 (sl) | 2009-04-30 |
| AU2006277836B2 (en) | 2011-11-10 |
| ES2317564T3 (es) | 2009-04-16 |
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Owner name: BIOVAIL LABORATORIES INTERNATIONAL (BARBADOS) , BB Free format text: OLD OWNER(S): CAMBRIDGE LABORATORIES (IRELAND) LIMITED |
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| PSEA | Patent sealed | ||
| RENW | Renewal (renewal fees accepted) | ||
| LAPS | Patent lapsed |