NO984084L - 4-Amino-pyrimidin-derivater, medikamenter inneholdende disse forbindelser, deres anvendelse og fremgangsmÕte ved fremstilling derav - Google Patents

4-Amino-pyrimidin-derivater, medikamenter inneholdende disse forbindelser, deres anvendelse og fremgangsmÕte ved fremstilling derav

Info

Publication number
NO984084L
NO984084L NO984084A NO984084A NO984084L NO 984084 L NO984084 L NO 984084L NO 984084 A NO984084 A NO 984084A NO 984084 A NO984084 A NO 984084A NO 984084 L NO984084 L NO 984084L
Authority
NO
Norway
Prior art keywords
amino
preparation
pyrimidine derivatives
compounds
medicaments containing
Prior art date
Application number
NO984084A
Other languages
English (en)
Other versions
NO984084D0 (no
Inventor
Frank Himmelsbach
Georg Dahmann
Den Thomas Von R
Thomas Metz
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE1996108631 external-priority patent/DE19608631A1/de
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of NO984084L publication Critical patent/NO984084L/no
Publication of NO984084D0 publication Critical patent/NO984084D0/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Den foreliggende oppfinnelse vedrører 4-amino-pyrimidin-derivater med den generelle formel hvor Ra. Rb- A og B er som definert i krav 1, deres tautomerer, deres stereoisomerer og deres salter, spesielt deres fysiologisk akseptable salter med uorganiske eller organiske syrer eller baser, og som har verdifulle farmakologiske egenskaper, særlig en hemmende virkning på signaltransduksjonen formidlet gjennom tyrosin- kinaser, deres anvendelse for behandling av sykdommer, særlig tumorsykdom- mer, og deres fremstilling.
NO984084A 1996-03-06 1998-09-04 4-Amino-pyrimidin-derivater, medikamenter inneholdende disse forbindelser, deres anvendelse og fremgangsmÕte ved fremstilling derav NO984084D0 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE1996108631 DE19608631A1 (de) 1996-03-06 1996-03-06 4-Amino-pyrimidin-Derivate, diese Verbindungen enthaltende Arnzeimittel, deren Verwendung und Verfahren zu ihrer Herstellung
DE19629652A DE19629652A1 (de) 1996-03-06 1996-07-23 4-Amino-pyrimidin-Derivate, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung
PCT/EP1997/001057 WO1997032881A1 (de) 1996-03-06 1997-03-03 4-amino-pyrimidin-derivate, diese verbindungen enthaltende arzneimittel, deren verwendung und verfahren zu ihrer herstellung

Publications (2)

Publication Number Publication Date
NO984084L true NO984084L (no) 1998-09-04
NO984084D0 NO984084D0 (no) 1998-09-04

Family

ID=26023531

Family Applications (1)

Application Number Title Priority Date Filing Date
NO984084A NO984084D0 (no) 1996-03-06 1998-09-04 4-Amino-pyrimidin-derivater, medikamenter inneholdende disse forbindelser, deres anvendelse og fremgangsmÕte ved fremstilling derav

Country Status (19)

Country Link
EP (1) EP0885226A1 (no)
JP (1) JP2000506847A (no)
KR (1) KR19990087550A (no)
CN (1) CN1212695A (no)
AU (1) AU710274B2 (no)
BG (1) BG102708A (no)
BR (1) BR9708312A (no)
CA (1) CA2243994A1 (no)
CZ (1) CZ281798A3 (no)
DE (1) DE19629652A1 (no)
EE (1) EE9800277A (no)
HU (1) HUP9901820A3 (no)
IL (1) IL125404A0 (no)
NO (1) NO984084D0 (no)
NZ (1) NZ331546A (no)
PL (1) PL328771A1 (no)
SK (1) SK120598A3 (no)
TR (1) TR199801749T2 (no)
WO (1) WO1997032881A1 (no)

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JP4471404B2 (ja) 1996-02-13 2010-06-02 アストラゼネカ ユーケイ リミテッド Ｖｅｇｆインヒビターとしてのキナゾリン誘導体
ATE211134T1 (de) 1996-03-05 2002-01-15 4-anilinochinazolin derivate
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DE4431867A1 (de) * 1994-09-07 1996-03-14 Thomae Gmbh Dr K Pyrimido[5,4-d]pyrimidine, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung

Also Published As

Publication number Publication date
SK120598A3 (en) 1999-06-11
HUP9901820A2 (hu) 1999-09-28
BR9708312A (pt) 1999-08-03
BG102708A (en) 1999-09-30
AU710274B2 (en) 1999-09-16
EE9800277A (et) 1999-02-15
JP2000506847A (ja) 2000-06-06
KR19990087550A (ko) 1999-12-27
PL328771A1 (en) 1999-02-15
TR199801749T2 (xx) 1998-12-21
AU1925197A (en) 1997-09-22
DE19629652A1 (de) 1998-01-29
NZ331546A (en) 2000-03-27
IL125404A0 (en) 1999-03-12
CA2243994A1 (en) 1997-09-12
CN1212695A (zh) 1999-03-31
NO984084D0 (no) 1998-09-04
WO1997032881A1 (de) 1997-09-12
CZ281798A3 (cs) 1999-02-17
EP0885226A1 (de) 1998-12-23
HUP9901820A3 (en) 2001-10-29

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