NO983197L - Nye trisykliske forbindelser og medikamentsammensetninger inneholdende slike - Google Patents

Nye trisykliske forbindelser og medikamentsammensetninger inneholdende slike

Info

Publication number
NO983197L
NO983197L NO983197A NO983197A NO983197L NO 983197 L NO983197 L NO 983197L NO 983197 A NO983197 A NO 983197A NO 983197 A NO983197 A NO 983197A NO 983197 L NO983197 L NO 983197L
Authority
NO
Norway
Prior art keywords
represents hydrogen
amino
compositions containing
tricyclic compounds
drug compositions
Prior art date
Application number
NO983197A
Other languages
English (en)
Other versions
NO312159B1 (no
Inventor
Shiro Miyoshi
Kohei Ogawa
Original Assignee
Asahi Chemical Ind
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Asahi Chemical Ind filed Critical Asahi Chemical Ind
Publication of NO983197L publication Critical patent/NO983197L/no
Publication of NO312159B1 publication Critical patent/NO312159B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/91—Dibenzofurans; Hydrogenated dibenzofurans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C307/00—Amides of sulfuric acids, i.e. compounds having singly-bound oxygen atoms of sulfate groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C307/04—Diamides of sulfuric acids
    • C07C307/10—Diamides of sulfuric acids having nitrogen atoms of the sulfamide groups bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
    • C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C311/08—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/30—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/37—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56—Ring systems containing three or more rings
    • C07D209/80—[b, c]- or [b, d]-condensed
    • C07D209/82—Carbazoles; Hydrogenated carbazoles
    • C07D209/88—Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/76—Dibenzothiophenes
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/02—Ortho- or ortho- and peri-condensed systems
    • C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
    • C07C2603/06—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members
    • C07C2603/10—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings
    • C07C2603/12—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings only one five-membered ring
    • C07C2603/18—Fluorenes; Hydrogenated fluorenes
NO19983197A 1996-01-10 1998-07-10 Nye trisykliske forbindelser og medikamentsammensetninger inneholdende slike NO312159B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP257696 1996-01-10
PCT/JP1996/003689 WO1997025311A1 (fr) 1996-01-10 1996-12-18 Nouveaux composes tricycliques et compositions medicamenteuses contenant ces composes

Publications (2)

Publication Number Publication Date
NO983197L true NO983197L (no) 1998-09-10
NO312159B1 NO312159B1 (no) 2002-04-02

Family

ID=11533209

Family Applications (2)

Application Number Title Priority Date Filing Date
NO19983197A NO312159B1 (no) 1996-01-10 1998-07-10 Nye trisykliske forbindelser og medikamentsammensetninger inneholdende slike
NO20012876A NO20012876D0 (no) 1996-01-10 2001-06-11 Nye trisykliske forbindelser og medikamentsammensetninger inneholdende slike

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO20012876A NO20012876D0 (no) 1996-01-10 2001-06-11 Nye trisykliske forbindelser og medikamentsammensetninger inneholdende slike

Country Status (14)

Country Link
US (4) US6037362A (no)
EP (1) EP0882707B1 (no)
JP (1) JP2000239255A (no)
KR (1) KR100395280B1 (no)
CN (2) CN1083831C (no)
AT (1) ATE251608T1 (no)
AU (1) AU715233B2 (no)
CA (1) CA2242351C (no)
DE (1) DE69630319T2 (no)
ES (1) ES2208772T3 (no)
HK (1) HK1017669A1 (no)
NO (2) NO312159B1 (no)
PT (1) PT882707E (no)
WO (1) WO1997025311A1 (no)

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US20030073644A1 (en) * 1998-11-11 2003-04-17 Smithkline Beecham P.L.C. Combinations comprising a beta-agonist and a further antidiabetic agent
CN1333760A (zh) * 1998-12-15 2002-01-30 旭化成株式会社 新杂环化合物以及含此化合物的药用组合物
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WO2000059885A1 (fr) * 1999-04-01 2000-10-12 Asahi Kasei Kabushiki Kaisha Procede de preparation de derives d'alcools amines tricycliques avec des azides
KR20020031381A (ko) * 1999-07-09 2002-05-01 야마모토 카즈모토 삼환성 아미노 알코올 유도체의 제조법
CA2383757A1 (en) * 1999-09-03 2001-03-15 Masami Ogawa Processes for the preparation of tricyclic amino alcohol derivatives
US20030220329A1 (en) * 1999-09-17 2003-11-27 Duke University Method of improving beta-adrenergic receptor function
BR0014469A (pt) * 1999-10-04 2002-06-11 Asahi Chemical Ind Processo para melhorar a solubilidade de um derivado de amino álcool tricìclico, composição farmacêutica, processo para preparar a mesma, e, derivado de amino álcool tricìclico
CN1423637A (zh) * 1999-12-16 2003-06-11 旭化成株式会社 新的取代的三环化合物
EP1258253A1 (en) * 2000-01-28 2002-11-20 Asahi Kasei Kabushiki Kaisha Novel remedies with the use of beta3 agonist
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AU2001252575A1 (en) * 2000-04-28 2001-11-12 Asahi Kasei Kabushiki Kaisha Novel tricyclic compounds
WO2001083453A1 (fr) * 2000-04-28 2001-11-08 Asahi Kasei Kabushiki Kaisha Nouveaux composes tricycliques substitues
GB0010757D0 (en) * 2000-05-05 2000-06-28 Astrazeneca Ab Chemical compounds
IL156487A0 (en) * 2000-12-22 2004-01-04 Astrazeneca Ab Carbazole derivatives and their use as neuropeptide y5 receptor ligands
WO2002074306A1 (fr) * 2001-03-19 2002-09-26 Asahi Kasei Kabushiki Kaisha Remedes pour la steatose hepatique
GB0121941D0 (en) * 2001-09-11 2001-10-31 Astrazeneca Ab Chemical compounds
KR100816527B1 (ko) * 2001-09-12 2008-04-10 한국화학연구원 페닐테트라졸 유도체로 치환된 β-아미노알코올 화합물
KR100622461B1 (ko) 2001-10-25 2006-09-19 아사히 가세이 파마 가부시키가이샤 2환식 화합물
AU2003209527A1 (en) * 2002-02-27 2003-09-09 Pfizer Products Inc. Crystal forms of (r)-2-(2-(4-oxazol-4-yl-phenoxy)-ethylamino)-1-pyridin-3-yl-ethanol
US6864268B2 (en) 2002-02-27 2005-03-08 Pfizer Inc. β3 adrenergic receptor agonists
AU2003248352A1 (en) 2002-02-27 2003-09-09 Pfizer Products Inc. PROCESSES AND INTERMEDIATES USEFUL IN PREPARING Beta3-ADRENERGIC RECEPTOR AGONISTS
EP1424079A1 (en) * 2002-11-27 2004-06-02 Boehringer Ingelheim International GmbH Combination of a beta-3-receptor agonist and of a reuptake inhibitor of serotonin and/or norepinephrine
WO2004072016A1 (ja) * 2003-02-14 2004-08-26 Kissei Pharmaceutical Co., Ltd. アミノアルコール誘導体、それを含有する医薬組成物およびそれらの用途
JP4644601B2 (ja) * 2003-10-24 2011-03-02 キッセイ薬品工業株式会社 アミノアルコール誘導体、それを含有する医薬組成物およびそれらの用途
US8501994B2 (en) 2007-08-28 2013-08-06 Sunovion Pharmaceuticals Inc. Acetamide stereoisomer
US7718822B2 (en) 2007-08-28 2010-05-18 Sepracor Inc. Carbamate Stereoisomer
CA2740772A1 (en) 2008-10-09 2010-04-15 Asahi Kasei Pharma Corporation Indazole compounds
CN102171191A (zh) 2008-10-09 2011-08-31 旭化成制药株式会社 吲唑衍生物
US20100222404A1 (en) * 2008-11-04 2010-09-02 Asahi Kasei Pharma Corporation Indazole derivative dihydrochloride
WO2011040510A1 (ja) * 2009-09-30 2011-04-07 旭化成ファーマ株式会社 インダゾール類縁体
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Also Published As

Publication number Publication date
EP0882707A1 (en) 1998-12-09
CN1209119A (zh) 1999-02-24
KR100395280B1 (ko) 2004-06-04
AU1170897A (en) 1997-08-01
NO20012876D0 (no) 2001-06-11
CN1083831C (zh) 2002-05-01
HK1017669A1 (en) 1999-11-26
EP0882707A4 (en) 2001-04-11
KR19990077162A (ko) 1999-10-25
US20030139475A1 (en) 2003-07-24
PT882707E (pt) 2004-02-27
US6037362A (en) 2000-03-14
NO312159B1 (no) 2002-04-02
AU715233B2 (en) 2000-01-20
DE69630319T2 (de) 2004-07-29
WO1997025311A1 (fr) 1997-07-17
CA2242351C (en) 2003-03-11
DE69630319D1 (de) 2003-11-13
NO20012876L (no) 1998-09-10
CA2242351A1 (en) 1997-07-17
CN1295064A (zh) 2001-05-16
ATE251608T1 (de) 2003-10-15
ES2208772T3 (es) 2004-06-16
US6545053B1 (en) 2003-04-08
EP0882707B1 (en) 2003-10-08
US6187809B1 (en) 2001-02-13
JP2000239255A (ja) 2000-09-05

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Legal Events

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MM1K Lapsed by not paying the annual fees

Free format text: LAPSED IN JUNE 2003