JPS5553262A - Phenylethanolamine derivative - Google Patents

Phenylethanolamine derivative

Info

Publication number
JPS5553262A
JPS5553262A JP12809978A JP12809978A JPS5553262A JP S5553262 A JPS5553262 A JP S5553262A JP 12809978 A JP12809978 A JP 12809978A JP 12809978 A JP12809978 A JP 12809978A JP S5553262 A JPS5553262 A JP S5553262A
Authority
JP
Japan
Prior art keywords
lower alkyl
phenylethanolamine derivative
phenylethanolamine
derivative
acosmia
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP12809978A
Other languages
Japanese (ja)
Other versions
JPS6213344B2 (en
Inventor
Kazuo Imai
Kunihiro Niigata
Takashi Fujikura
Shinichi Hashimoto
Takaichi Takenaka
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Yamanouchi Pharmaceutical Co Ltd
Original Assignee
Yamanouchi Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yamanouchi Pharmaceutical Co Ltd filed Critical Yamanouchi Pharmaceutical Co Ltd
Priority to JP12809978A priority Critical patent/JPS5553262A/en
Publication of JPS5553262A publication Critical patent/JPS5553262A/en
Publication of JPS6213344B2 publication Critical patent/JPS6213344B2/ja
Granted legal-status Critical Current

Links

Abstract

NEW MATERIAL:A phenylethanolamine derivative I [X is H, lower alkyl, lower alkoxy, halogen, OH, sulfamoyl, carbamoyl, cyano, etc.; R1 is H or lower alkyl; n is 0.1 or 3; Y is methylene, O or S; R2 is (substituted) aryl, benzodioxane ring, etc.].
EXAMPLE: 5-[ 1-Hydroxy-2-{ 1-( 1,4-benzodioxan-2-yl )ethylamino }propyl ]-2- methoxybenzenesulfonamide.
USE: An agent having both β-and α-adrenalin-blocking activities, useful as a hypotensor having reduced side effects, and as a remedy for peripheral acosmia, e.g. Raynaud's disease, etc., or angina pectoris.
PROCESS: A compound I is prepared by aminolysis of a halohydrin II1 or an epoxide II2 with an amine III1.
COPYRIGHT: (C)1980,JPO&Japio
JP12809978A 1978-10-17 1978-10-17 Phenylethanolamine derivative Granted JPS5553262A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP12809978A JPS5553262A (en) 1978-10-17 1978-10-17 Phenylethanolamine derivative

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP12809978A JPS5553262A (en) 1978-10-17 1978-10-17 Phenylethanolamine derivative

Publications (2)

Publication Number Publication Date
JPS5553262A true JPS5553262A (en) 1980-04-18
JPS6213344B2 JPS6213344B2 (en) 1987-03-25

Family

ID=14976361

Family Applications (1)

Application Number Title Priority Date Filing Date
JP12809978A Granted JPS5553262A (en) 1978-10-17 1978-10-17 Phenylethanolamine derivative

Country Status (1)

Country Link
JP (1) JPS5553262A (en)

Cited By (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0034432A2 (en) * 1980-02-08 1981-08-26 Yamanouchi Pharmaceutical Co., Ltd. Sulfamoyl-substituted phenethylamine derivatives, their preparation, and pharmaceutical compositions, containing them
US6037362A (en) * 1996-01-10 2000-03-14 Asahi Kasei Kogyo Kabushiki Kaisha Tricyclic compounds and drug compositions containing the same
US6172099B1 (en) 1997-07-03 2001-01-09 Asahi Kasei Kogyo Kabushiki Kaisha Tricyclic compounds having saturated rings and medicinal compositions containing the same
US6861444B2 (en) 2000-04-28 2005-03-01 Asahi Kasei Pharma Corporation Bicyclic compounds
US7271190B2 (en) 2001-10-25 2007-09-18 Asahi Kasei Pharma Corporation Indazole compounds as β3 adrenoceptor agonist
US8008506B2 (en) 2008-10-09 2011-08-30 Asahi Kasei Pharma Corporation Indazole compounds
US8304443B2 (en) 2008-10-09 2012-11-06 Asahi Kasei Pharma Corporation Indazole derivatives

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS53111029A (en) * 1977-02-03 1978-09-28 Allen & Hanburys Ltd New derivative of benzensulfonamido and benzencarboxyamido * method of its production and drug composition containing these
JPS5950671A (en) * 1982-09-16 1984-03-23 Olympus Optical Co Ltd Method for displaying focus information of television camera or the like

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS53111029A (en) * 1977-02-03 1978-09-28 Allen & Hanburys Ltd New derivative of benzensulfonamido and benzencarboxyamido * method of its production and drug composition containing these
JPS5950671A (en) * 1982-09-16 1984-03-23 Olympus Optical Co Ltd Method for displaying focus information of television camera or the like

Cited By (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0034432A2 (en) * 1980-02-08 1981-08-26 Yamanouchi Pharmaceutical Co., Ltd. Sulfamoyl-substituted phenethylamine derivatives, their preparation, and pharmaceutical compositions, containing them
US6037362A (en) * 1996-01-10 2000-03-14 Asahi Kasei Kogyo Kabushiki Kaisha Tricyclic compounds and drug compositions containing the same
US6187809B1 (en) * 1996-01-10 2001-02-13 Asahi Kasei Kogyo Kabushiki Kaisha Tricyclic compounds and drug compositions containing the same
US6545053B1 (en) 1996-01-10 2003-04-08 Asahi Kasei Kogyo Kabushiki Kaisha Tricyclic compounds and drug compositions containing same
US6172099B1 (en) 1997-07-03 2001-01-09 Asahi Kasei Kogyo Kabushiki Kaisha Tricyclic compounds having saturated rings and medicinal compositions containing the same
US6861444B2 (en) 2000-04-28 2005-03-01 Asahi Kasei Pharma Corporation Bicyclic compounds
US7271190B2 (en) 2001-10-25 2007-09-18 Asahi Kasei Pharma Corporation Indazole compounds as β3 adrenoceptor agonist
US7511069B2 (en) 2001-10-25 2009-03-31 Asahi Pharma Corporation Indazole compounds as β3 andrenoceptor agonist
US7598284B2 (en) 2001-10-25 2009-10-06 Asahi Kasei Pharma Corporation Indazole compounds as B3 adrenoceptor agonist
US8008506B2 (en) 2008-10-09 2011-08-30 Asahi Kasei Pharma Corporation Indazole compounds
US8304443B2 (en) 2008-10-09 2012-11-06 Asahi Kasei Pharma Corporation Indazole derivatives

Also Published As

Publication number Publication date
JPS6213344B2 (en) 1987-03-25

Similar Documents

Publication Publication Date Title
IE811931L (en) Oxiranes.
JPS5553262A (en) Phenylethanolamine derivative
JPS5629548A (en) Omega-aminoalkoxystilbenes and their acid addition salts
KR830007512A (en) Method for producing short acting β-blocker
JPS55129256A (en) Antifungal compound
JPS5692884A (en) Novel piperidine derivative and its preparation
IT1193608B (en) ARYOXYPROPANOLAMINE DERIVATIVES, PROCEDURE FOR THEIR PREPARATION PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR THERAPEUTIC USE
JPS5756476A (en) Omega-aminoalkoxybenzoylthiophene
JPS5553261A (en) New phenylethanolamine derivative and its preparation
JPS55115877A (en) Novel amidine compound and its preparation
JPS56126833A (en) Forming method for color image
JPS57108064A (en) Perfluoroalkylthio compound
JPS5473751A (en) Phenyl ethanolamine derivatives and their preparation
KR850003407A (en) Process for preparing organophosphate ester derivative
JPS5728040A (en) Phenylethanolamine derivative
JPS55130949A (en) Novel phenylacetamide derivative
JPS5651461A (en) Novel 3-phenyl-4-quinazolone derivative
JPS56142272A (en) Hydrazinopyridazine derivative
JPS5225736A (en) Preparation of benzamide derivatives
JPS5612361A (en) Isopropylamine derivative and its preparation
JPS5515456A (en) 2-substituted-piperazinomethyl-1,4-benzodioxane
JPS5653654A (en) Preparation of novel aniline derivative
JPS5780379A (en) (omega-piperazinylalkoxy)alkylenedioxybenzene and its acid addition salt
JPS5750973A (en) Alkane acid derivative
JPS56169676A (en) Novel substituted benzylidene hydrazinophthalazine derivative