NO980211L - Opplösning av 1-azabicyklo£2,2,2|oktan-3-amin, 2-(difenylmetyl)-N-££2-metoksy-5-(1-metyletyl)fenyl|metyl| - Google Patents

Opplösning av 1-azabicyklo£2,2,2|oktan-3-amin, 2-(difenylmetyl)-N-££2-metoksy-5-(1-metyletyl)fenyl|metyl|

Info

Publication number
NO980211L
NO980211L NO980211A NO980211A NO980211L NO 980211 L NO980211 L NO 980211L NO 980211 A NO980211 A NO 980211A NO 980211 A NO980211 A NO 980211A NO 980211 L NO980211 L NO 980211L
Authority
NO
Norway
Prior art keywords
methyl
diphenylmethyl
azabicyclo
methoxy
amine
Prior art date
Application number
NO980211A
Other languages
English (en)
Norwegian (no)
Other versions
NO980211D0 (no
Inventor
Derek L Tickner
Morgan Meltz
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NO980211D0 publication Critical patent/NO980211D0/no
Publication of NO980211L publication Critical patent/NO980211L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Indole Compounds (AREA)
NO980211A 1995-07-17 1998-01-16 Opplösning av 1-azabicyklo£2,2,2|oktan-3-amin, 2-(difenylmetyl)-N-££2-metoksy-5-(1-metyletyl)fenyl|metyl| NO980211L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US119195P 1995-07-17 1995-07-17
PCT/IB1996/000648 WO1997003984A1 (en) 1995-07-17 1996-07-04 Resolution of 1-azabicyclo[2.2.2]octan-3-amine, 2-(diphenylmethyl)-n-[[2-methoxy-5-(1-methylethyl)phenyl]methyl]

Publications (2)

Publication Number Publication Date
NO980211D0 NO980211D0 (no) 1998-01-16
NO980211L true NO980211L (no) 1998-03-16

Family

ID=21694832

Family Applications (1)

Application Number Title Priority Date Filing Date
NO980211A NO980211L (no) 1995-07-17 1998-01-16 Opplösning av 1-azabicyklo£2,2,2|oktan-3-amin, 2-(difenylmetyl)-N-££2-metoksy-5-(1-metyletyl)fenyl|metyl|

Country Status (26)

Country Link
US (1) US6008357A (zh)
EP (1) EP0840735B1 (zh)
JP (1) JP3043074B2 (zh)
KR (1) KR100276989B1 (zh)
CN (1) CN1068598C (zh)
AR (1) AR002772A1 (zh)
AT (1) ATE250600T1 (zh)
AU (1) AU697553B2 (zh)
CA (1) CA2227194C (zh)
CO (1) CO4480720A1 (zh)
CZ (1) CZ15098A3 (zh)
DE (1) DE69630123T2 (zh)
DK (1) DK0840735T3 (zh)
ES (1) ES2205039T3 (zh)
HK (1) HK1010195A1 (zh)
HU (1) HUP9900238A3 (zh)
IL (1) IL122655A0 (zh)
MY (1) MY115734A (zh)
NO (1) NO980211L (zh)
NZ (1) NZ310539A (zh)
PE (1) PE8798A1 (zh)
PL (1) PL184261B1 (zh)
PT (1) PT840735E (zh)
RU (1) RU2136681C1 (zh)
WO (1) WO1997003984A1 (zh)
ZA (1) ZA966026B (zh)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6861526B2 (en) 2002-10-16 2005-03-01 Pfizer Inc. Process for the preparation of (S,S)-cis-2-benzhydryl-3-benzylaminoquinuclidine
AU2005210259A1 (en) * 2004-02-02 2005-08-18 Pfizer Products Inc. Process for preparation of 1-(2S,3S)-2-benzhydr yl-N-(5-tert-butyl-2-methoxybenzyl)quinuclidin-3-amine
WO2006055321A2 (en) * 2004-11-10 2006-05-26 Boehringer Ingelheim Chemicals, Inc. Process of making fentanyl intermediates
CN102395557A (zh) * 2008-12-09 2012-03-28 佛罗里达大学研究基金会公司 激酶抑制剂化合物
US20160332962A1 (en) 2015-05-13 2016-11-17 Janssen Pharmaceutica Nv (s)-csa salt of s-ketamine, (r)-csa salt of s-ketamine and processes for the preparation of s-ketamine
CN108341812A (zh) * 2017-01-23 2018-07-31 科贝源(北京)生物医药科技有限公司 一种含奎宁环化合物的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1990005525A1 (en) * 1988-11-23 1990-05-31 Pfizer Inc. Quinuclidine derivatives as substance p antagonists
NO168529C (no) * 1989-09-15 1992-03-04 Chiron Lab As Fremgangsmaate for fremstilling av s-(-) og r-(+)-n-(quinuclidinyl-3)-amider.
CA2109415C (en) * 1991-05-22 1998-12-29 Fumitaka Ito Substituted 3-aminoquinuclidines
PL171379B1 (en) * 1991-05-31 1997-04-30 Pfizer Method of obtaining novel derivatives of quinuclidine
US5604241A (en) * 1992-10-21 1997-02-18 Pfizer Inc. Substituted benzylaminoquinuclidines as substance P antagonists

Also Published As

Publication number Publication date
JPH10511102A (ja) 1998-10-27
DK0840735T3 (da) 2004-02-09
AU697553B2 (en) 1998-10-08
US6008357A (en) 1999-12-28
CN1068598C (zh) 2001-07-18
EP0840735A1 (en) 1998-05-13
PL184261B1 (pl) 2002-09-30
NZ310539A (en) 1998-11-25
CA2227194C (en) 2002-02-12
AR002772A1 (es) 1998-04-29
PT840735E (pt) 2004-02-27
HUP9900238A2 (hu) 1999-05-28
JP3043074B2 (ja) 2000-05-22
WO1997003984A1 (en) 1997-02-06
HUP9900238A3 (en) 2001-08-28
CA2227194A1 (en) 1997-02-06
AU6134896A (en) 1997-02-18
NO980211D0 (no) 1998-01-16
KR19990029058A (ko) 1999-04-15
ATE250600T1 (de) 2003-10-15
PE8798A1 (es) 1998-03-02
MY115734A (en) 2003-08-30
CO4480720A1 (es) 1997-07-09
KR100276989B1 (ko) 2001-01-15
EP0840735B1 (en) 2003-09-24
RU2136681C1 (ru) 1999-09-10
DE69630123D1 (en) 2003-10-30
CN1190970A (zh) 1998-08-19
IL122655A0 (en) 1998-08-16
DE69630123T2 (de) 2004-04-08
CZ15098A3 (cs) 1999-02-17
ZA966026B (en) 1998-01-16
MX9800538A (es) 1998-05-31
ES2205039T3 (es) 2004-05-01
HK1010195A1 (en) 1999-06-17
PL324610A1 (en) 1998-06-08

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