NO883146L - Antiinflamatorisk aktive arylderivater og fremgangsmaate for deres fremstilling. - Google Patents
Antiinflamatorisk aktive arylderivater og fremgangsmaate for deres fremstilling.Info
- Publication number
- NO883146L NO883146L NO88883146A NO883146A NO883146L NO 883146 L NO883146 L NO 883146L NO 88883146 A NO88883146 A NO 88883146A NO 883146 A NO883146 A NO 883146A NO 883146 L NO883146 L NO 883146L
- Authority
- NO
- Norway
- Prior art keywords
- formula
- compound
- methyl
- enyl
- prop
- Prior art date
Links
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Classifications
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
- C07C251/32—Oximes
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N37/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids
- A01N37/18—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing the group —CO—N<, e.g. carboxylic acid amides or imides; Thio analogues thereof
- A01N37/28—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing the group —CO—N<, e.g. carboxylic acid amides or imides; Thio analogues thereof containing the group; Thio analogues thereof
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/14—Decongestants or antiallergics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Wood Science & Technology (AREA)
- Pest Control & Pesticides (AREA)
- Epidemiology (AREA)
- Environmental Sciences (AREA)
- Zoology (AREA)
- Pulmonology (AREA)
- Dentistry (AREA)
- Plant Pathology (AREA)
- Pain & Pain Management (AREA)
- Immunology (AREA)
- Ophthalmology & Optometry (AREA)
- Agronomy & Crop Science (AREA)
- Heart & Thoracic Surgery (AREA)
- Neurology (AREA)
- Rheumatology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Biomedical Technology (AREA)
- Cardiology (AREA)
- Neurosurgery (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB878716640A GB8716640D0 (en) | 1987-07-15 | 1987-07-15 | Aryl derivatives |
| GB888802378A GB8802378D0 (en) | 1988-02-03 | 1988-02-03 | New aryl derivatives |
| GB888806278A GB8806278D0 (en) | 1988-03-16 | 1988-03-16 | New aryl derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO883146D0 NO883146D0 (no) | 1988-07-14 |
| NO883146L true NO883146L (no) | 1989-01-16 |
Family
ID=27263507
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO88883146A NO883146L (no) | 1987-07-15 | 1988-07-14 | Antiinflamatorisk aktive arylderivater og fremgangsmaate for deres fremstilling. |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US4988733A (xx) |
| EP (1) | EP0299761B1 (xx) |
| JP (1) | JPS6445344A (xx) |
| KR (1) | KR890001966A (xx) |
| AT (1) | ATE70530T1 (xx) |
| AU (1) | AU603468B2 (xx) |
| DE (1) | DE3866981D1 (xx) |
| DK (1) | DK392788A (xx) |
| ES (1) | ES2051854T3 (xx) |
| FI (1) | FI883355A (xx) |
| GR (1) | GR3003393T3 (xx) |
| HU (1) | HU203076B (xx) |
| IL (1) | IL87105A0 (xx) |
| MC (1) | MC1959A1 (xx) |
| NO (1) | NO883146L (xx) |
| NZ (1) | NZ225408A (xx) |
| PL (1) | PL154186B1 (xx) |
| PT (1) | PT87987B (xx) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH0288553A (ja) * | 1988-07-14 | 1990-03-28 | Wellcome Found Ltd:The | 抗炎症性アリール誘導体 |
| ES2060015T3 (es) * | 1989-02-03 | 1994-11-16 | Wellcome Found | Derivados arilicos anti-inflamatorios. |
| US5476873A (en) * | 1990-07-25 | 1995-12-19 | Abbott Laboratories | Acetylene derivatives having lipoxygenase inhibitory activity |
| JPH0819069B2 (ja) * | 1990-07-25 | 1996-02-28 | アボツト・ラボラトリーズ | リポキシゲナーゼ阻害活性を有するアセチレン誘導体 |
| US5234933A (en) * | 1991-10-31 | 1993-08-10 | Board Of Governors Of Wayne State University And Vanderbilt University | Cyclic hydroxamic acids |
| US5169854A (en) * | 1992-02-26 | 1992-12-08 | Abbott Laboratories | N-substituted-furylalkenyl hydroxamic acid and N-hydroxyurea compounds having lipoxygenase inhibitory activity |
| US5187192A (en) * | 1992-03-13 | 1993-02-16 | Abbott Laboratories | Cyclobutyl derivatives having lipoxygenase inhibitory activity |
| ATE189123T1 (de) * | 1992-06-30 | 2000-02-15 | Us Health | Verfahren zur herstellung einer schutzsperre gegen virus |
| GB9215921D0 (en) * | 1992-07-27 | 1992-09-09 | Wellcome Found | Anti-inflammatory compounds |
| WO1994004537A2 (en) * | 1992-08-20 | 1994-03-03 | Cytomed, Inc. | Dual functional anti-inflammatory and immunosuppressive agents |
| GB9308652D0 (en) * | 1993-04-27 | 1993-06-09 | Wellcome Found | Anti-inflammatory compounds |
| EP0833622B8 (en) * | 1995-06-12 | 2005-10-12 | G.D. Searle & Co. | Compositions comprising a cyclooxygenase-2 inhibitor and a 5-lipoxygenase inhibitor |
| AR029916A1 (es) * | 2000-05-05 | 2003-07-23 | Smithkline Beecham Corp | N-formil-n-hidroxi-ariloxi alquilaminas y metodos para tratar infecciones bacterianas |
| AR028075A1 (es) * | 2000-05-05 | 2003-04-23 | Smithkline Beecham Corp | Inhibidores de la peptido-desformilasa |
| US20040034024A1 (en) * | 2001-05-04 | 2004-02-19 | Aubart Kelly M | Peptide deformylase inhibitors |
| ATE445838T1 (de) | 2001-07-25 | 2009-10-15 | Raptor Pharmaceutical Inc | Zusammensetzungen und verfahren zur modulation des transports durch die blut-hirn-schranke |
| EP2671508B1 (en) | 2005-04-28 | 2020-09-16 | Proteus Digital Health, Inc. | Pharma-informatics system |
| CA2663377A1 (en) | 2006-09-18 | 2008-03-27 | Raptor Pharmaceutical Inc. | Treatment of liver disorders by administration of receptor-associated protein (rap)-conjugates |
| GB0624187D0 (en) * | 2006-12-04 | 2007-01-10 | Jackson William P | HDAC inhibitors |
| HUE059078T2 (hu) | 2009-02-20 | 2022-10-28 | Enhanx Biopharm Inc | Glutation-alapú hatóanyagszállító rendszer |
| JP2012526144A (ja) | 2009-05-06 | 2012-10-25 | ラボラトリー スキン ケア インコーポレイテッド | 活性物質−リン酸カルシウム粒子複合体を含む経皮送達組成物およびその使用方法 |
| US20120077778A1 (en) | 2010-09-29 | 2012-03-29 | Andrea Bourdelais | Ladder-Frame Polyether Conjugates |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0196184B1 (en) * | 1985-03-16 | 1992-09-16 | The Wellcome Foundation Limited | Aryl derivatives |
| IE59397B1 (en) * | 1985-03-16 | 1994-02-23 | Wellcome Found | New aryl derivatives |
| US4608390A (en) * | 1985-04-26 | 1986-08-26 | Abbott Laboratories | Lipoxygenase inhibiting compounds |
| GB8718212D0 (en) * | 1987-07-31 | 1987-09-09 | Angus Fire Armour Ltd | Lining tubular objects |
-
1988
- 1988-07-12 PL PL1988273728A patent/PL154186B1/pl unknown
- 1988-07-14 IL IL87105A patent/IL87105A0/xx unknown
- 1988-07-14 JP JP63176198A patent/JPS6445344A/ja active Pending
- 1988-07-14 NZ NZ225408A patent/NZ225408A/xx unknown
- 1988-07-14 AT AT88306446T patent/ATE70530T1/de not_active IP Right Cessation
- 1988-07-14 ES ES88306446T patent/ES2051854T3/es not_active Expired - Lifetime
- 1988-07-14 KR KR1019880008745A patent/KR890001966A/ko not_active Application Discontinuation
- 1988-07-14 DK DK392788A patent/DK392788A/da not_active Application Discontinuation
- 1988-07-14 MC MC881991A patent/MC1959A1/xx unknown
- 1988-07-14 FI FI883355A patent/FI883355A/fi not_active Application Discontinuation
- 1988-07-14 EP EP88306446A patent/EP0299761B1/en not_active Expired - Lifetime
- 1988-07-14 NO NO88883146A patent/NO883146L/no unknown
- 1988-07-14 HU HU883683A patent/HU203076B/hu unknown
- 1988-07-14 DE DE8888306446T patent/DE3866981D1/de not_active Expired - Fee Related
- 1988-07-14 AU AU19068/88A patent/AU603468B2/en not_active Ceased
- 1988-07-14 PT PT87987A patent/PT87987B/pt not_active IP Right Cessation
- 1988-07-14 US US07/219,096 patent/US4988733A/en not_active Expired - Fee Related
-
1991
- 1991-12-19 GR GR91401878T patent/GR3003393T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| KR890001966A (ko) | 1989-04-07 |
| PT87987B (pt) | 1995-03-01 |
| JPS6445344A (en) | 1989-02-17 |
| HU203076B (en) | 1991-05-28 |
| PL273728A1 (en) | 1989-04-03 |
| FI883355A (fi) | 1989-01-16 |
| ES2051854T3 (es) | 1994-07-01 |
| EP0299761A1 (en) | 1989-01-18 |
| PL154186B1 (en) | 1991-07-31 |
| PT87987A (pt) | 1989-06-30 |
| US4988733A (en) | 1991-01-29 |
| DK392788D0 (da) | 1988-07-14 |
| GR3003393T3 (en) | 1993-02-17 |
| DE3866981D1 (de) | 1992-01-30 |
| IL87105A0 (en) | 1988-12-30 |
| AU1906888A (en) | 1989-01-19 |
| ATE70530T1 (de) | 1992-01-15 |
| MC1959A1 (fr) | 1989-06-30 |
| FI883355A0 (fi) | 1988-07-14 |
| NO883146D0 (no) | 1988-07-14 |
| HUT48572A (en) | 1989-06-28 |
| DK392788A (da) | 1989-01-16 |
| NZ225408A (en) | 1991-09-25 |
| AU603468B2 (en) | 1990-11-15 |
| EP0299761B1 (en) | 1991-12-18 |
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