NO331689B1 - Oral farmasoytisk sammensetning omfattende rivastigmin, samt anvendelse av rivastigmin - Google Patents
Oral farmasoytisk sammensetning omfattende rivastigmin, samt anvendelse av rivastigmin Download PDFInfo
- Publication number
- NO331689B1 NO331689B1 NO20011471A NO20011471A NO331689B1 NO 331689 B1 NO331689 B1 NO 331689B1 NO 20011471 A NO20011471 A NO 20011471A NO 20011471 A NO20011471 A NO 20011471A NO 331689 B1 NO331689 B1 NO 331689B1
- Authority
- NO
- Norway
- Prior art keywords
- rivastigmine
- composition
- pharmaceutical composition
- cellulose
- water
- Prior art date
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- 239000008203 oral pharmaceutical composition Substances 0.000 title claims description 7
- XSVMFMHYUFZWBK-NSHDSACASA-N Rivastigmine Chemical compound CCN(C)C(=O)OC1=CC=CC([C@H](C)N(C)C)=C1 XSVMFMHYUFZWBK-NSHDSACASA-N 0.000 claims abstract description 53
- 229960004136 rivastigmine Drugs 0.000 claims abstract description 50
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Classifications
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/27—Esters, e.g. nitroglycerine, selenocyanates of carbamic or thiocarbamic acids, meprobamate, carbachol, neostigmine
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- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2886—Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
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- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Emergency Medicine (AREA)
- Biomedical Technology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Cosmetics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9821299.6A GB9821299D0 (en) | 1998-10-01 | 1998-10-01 | Organic compounds |
| GBGB9821298.8A GB9821298D0 (en) | 1998-10-01 | 1998-10-01 | Organic compoundsq |
| GBGB9826654.7A GB9826654D0 (en) | 1998-12-03 | 1998-12-03 | Organic compounds |
| GBGB9827624.9A GB9827624D0 (en) | 1998-12-16 | 1998-12-16 | Organic compounds |
| GBGB9907822.2A GB9907822D0 (en) | 1999-04-06 | 1999-04-06 | Organic compounds |
| GBGB9907823.0A GB9907823D0 (en) | 1999-04-06 | 1999-04-06 | Organic compounds |
| PCT/EP1999/007298 WO2000019985A2 (en) | 1998-10-01 | 1999-10-01 | New sustained release oral formulations |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20011471D0 NO20011471D0 (no) | 2001-03-22 |
| NO20011471L NO20011471L (no) | 2001-03-22 |
| NO331689B1 true NO331689B1 (no) | 2012-02-27 |
Family
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| Application Number | Title | Priority Date | Filing Date |
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| NO20011471A NO331689B1 (no) | 1998-10-01 | 2001-03-22 | Oral farmasoytisk sammensetning omfattende rivastigmin, samt anvendelse av rivastigmin |
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| EP (1) | EP1121104B1 (cs) |
| JP (1) | JP4012689B2 (cs) |
| KR (1) | KR100603900B1 (cs) |
| CN (1) | CN1406126A (cs) |
| AT (1) | ATE286725T1 (cs) |
| AU (1) | AU764866B2 (cs) |
| BR (1) | BR9914251A (cs) |
| CA (1) | CA2342340C (cs) |
| CZ (1) | CZ302888B6 (cs) |
| DE (1) | DE69923200T2 (cs) |
| ES (1) | ES2237163T3 (cs) |
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| HU (1) | HUP0103883A3 (cs) |
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| NO (1) | NO331689B1 (cs) |
| NZ (1) | NZ510683A (cs) |
| PL (1) | PL196945B1 (cs) |
| PT (1) | PT1121104E (cs) |
| SK (1) | SK285250B6 (cs) |
| TR (1) | TR200100931T2 (cs) |
| WO (1) | WO2000019985A2 (cs) |
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| AU6715600A (en) * | 1999-08-26 | 2001-03-19 | Elan Corporation, Plc | Pharmaceutical formulations |
| GB9923045D0 (en) * | 1999-09-29 | 1999-12-01 | Novartis Ag | New oral formulations |
| CN1466451B (zh) * | 2000-09-29 | 2010-05-12 | 索尔瓦药物有限公司 | 不受离子强度影响的持续释放的医药制剂 |
| JP5023412B2 (ja) * | 2001-05-09 | 2012-09-12 | 吉澤石灰工業株式会社 | ホルムアルデヒド廃液の処理剤 |
| PT1424997E (pt) * | 2001-09-14 | 2008-02-28 | Scolr Inc | Forma de dosagem de libertação prolongada modulada por aminoácidos |
| JP2005525299A (ja) * | 2001-09-14 | 2005-08-25 | スコラー インコーポレイテッド | アミノ酸調節性の長期放出投薬形態 |
| KR100453288B1 (ko) * | 2002-03-12 | 2004-10-21 | 한국화학연구원 | 약물의 제어 방출을 위한 스퀴즈-유형의 삼투성 약물 전달장치 |
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| KR100990590B1 (ko) * | 2005-09-01 | 2010-10-29 | 에자이 알앤드디 매니지먼트 가부시키가이샤 | 붕해성이 개선된 의약 조성물의 제조 방법 |
| GB0525461D0 (en) | 2005-12-15 | 2006-01-25 | Archimedes Dev Ltd | Pharmaceutical compositions |
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| CN1158071C (zh) * | 1997-05-30 | 2004-07-21 | 渗透有限公司 | 多层渗透装置 |
| GB9800526D0 (en) * | 1998-01-12 | 1998-03-11 | Ciba Geigy Ag | Organic compounds |
| TR200100931T2 (tr) | 1998-10-01 | 2001-10-22 | Novartis Ag | Yeni sürekli salınımlı oral formülasyonlar |
| US6534541B1 (en) | 1999-10-19 | 2003-03-18 | Novartis Ag | Treatment of ocular disorders |
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1999
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- 1999-10-01 CN CN99811633A patent/CN1406126A/zh active Pending
- 1999-10-01 ID IDW20010671A patent/ID27504A/id unknown
- 1999-10-01 WO PCT/EP1999/007298 patent/WO2000019985A2/en not_active Ceased
- 1999-10-01 ES ES99950595T patent/ES2237163T3/es not_active Expired - Lifetime
- 1999-10-01 BR BR9914251-1A patent/BR9914251A/pt not_active Application Discontinuation
- 1999-10-01 NZ NZ510683A patent/NZ510683A/en not_active IP Right Cessation
- 1999-10-01 HU HU0103883A patent/HUP0103883A3/hu unknown
- 1999-10-01 PT PT99950595T patent/PT1121104E/pt unknown
- 1999-10-01 CA CA002342340A patent/CA2342340C/en not_active Expired - Fee Related
- 1999-10-01 CZ CZ20011155A patent/CZ302888B6/cs not_active IP Right Cessation
- 1999-10-01 EP EP99950595A patent/EP1121104B1/en not_active Expired - Lifetime
- 1999-10-01 HK HK03104925.9A patent/HK1052473A1/zh unknown
- 1999-10-01 PL PL348734A patent/PL196945B1/pl not_active IP Right Cessation
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2001
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- 2001-03-27 US US09/818,690 patent/US20010033866A1/en not_active Abandoned
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2002
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2003
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2005
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2006
- 2006-11-03 US US11/592,853 patent/US20070053982A1/en not_active Abandoned
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