NO321388B1 - Farmasoytisk sammensetning inneholdende en forbindelse med angiotensin II antagonistisk aktivitet i kombinasjon med en forbindelse som har insulinsensitivitetsstimulerende aktivitet, og anvendelse av samme for fremstilling av medikament. - Google Patents

Farmasoytisk sammensetning inneholdende en forbindelse med angiotensin II antagonistisk aktivitet i kombinasjon med en forbindelse som har insulinsensitivitetsstimulerende aktivitet, og anvendelse av samme for fremstilling av medikament. Download PDF

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Publication number
NO321388B1
NO321388B1 NO19984123A NO984123A NO321388B1 NO 321388 B1 NO321388 B1 NO 321388B1 NO 19984123 A NO19984123 A NO 19984123A NO 984123 A NO984123 A NO 984123A NO 321388 B1 NO321388 B1 NO 321388B1
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Norway
Prior art keywords
group
compound
methyl
angiotensin
ethoxy
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Application number
NO19984123A
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English (en)
Norwegian (no)
Other versions
NO984123D0 (no
NO984123L (no
Inventor
Hitoshi Ikeda
Norikazu Tamura
Takashi Sohada
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Takeda Pharmaceutical
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Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of NO984123D0 publication Critical patent/NO984123D0/no
Publication of NO984123L publication Critical patent/NO984123L/no
Publication of NO321388B1 publication Critical patent/NO321388B1/no

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • A61K31/222Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin with compounds having aromatic groups, e.g. dipivefrine, ibopamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41841,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
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    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
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    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
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    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
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    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P9/12Antihypertensives

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  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Neurosurgery (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
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  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
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  • Urology & Nephrology (AREA)
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  • Vascular Medicine (AREA)
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  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO19984123A 1996-04-05 1998-09-07 Farmasoytisk sammensetning inneholdende en forbindelse med angiotensin II antagonistisk aktivitet i kombinasjon med en forbindelse som har insulinsensitivitetsstimulerende aktivitet, og anvendelse av samme for fremstilling av medikament. NO321388B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP8391796 1996-04-05
PCT/JP1997/001149 WO1997037688A2 (fr) 1996-04-05 1997-04-03 Combinaison pharmaceutique comprenant un compose contenant de l'angiotensine ii et presentant une activite antagoniste

Publications (3)

Publication Number Publication Date
NO984123D0 NO984123D0 (no) 1998-09-07
NO984123L NO984123L (no) 1998-09-07
NO321388B1 true NO321388B1 (no) 2006-05-02

Family

ID=13815962

Family Applications (1)

Application Number Title Priority Date Filing Date
NO19984123A NO321388B1 (no) 1996-04-05 1998-09-07 Farmasoytisk sammensetning inneholdende en forbindelse med angiotensin II antagonistisk aktivitet i kombinasjon med en forbindelse som har insulinsensitivitetsstimulerende aktivitet, og anvendelse av samme for fremstilling av medikament.

Country Status (22)

Country Link
US (2) US6107323A (fr)
EP (4) EP1192951A3 (fr)
JP (2) JPH09323940A (fr)
KR (2) KR19990087076A (fr)
CN (1) CN1215338A (fr)
AT (1) ATE220333T1 (fr)
AU (1) AU713277B2 (fr)
BR (1) BR9708517A (fr)
CA (3) CA2577233C (fr)
CY (1) CY2300B1 (fr)
CZ (1) CZ297941B6 (fr)
DE (1) DE69713890T3 (fr)
DK (1) DK0914158T4 (fr)
ES (1) ES2175385T5 (fr)
NO (1) NO321388B1 (fr)
NZ (1) NZ330774A (fr)
PL (2) PL193365B1 (fr)
PT (1) PT914158E (fr)
RU (1) RU2188013C2 (fr)
SI (1) SI0914158T2 (fr)
SK (1) SK283348B6 (fr)
WO (1) WO1997037688A2 (fr)

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EP0914158B1 (fr) 2002-07-10
CA2241466A1 (fr) 1997-10-16
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US6432996B1 (en) 2002-08-13
US6107323A (en) 2000-08-22
SK127898A3 (en) 1999-05-07
DE69713890D1 (de) 2002-08-14
ES2175385T3 (es) 2002-11-16
PL329188A1 (en) 1999-03-15
CA2241466C (fr) 2007-05-22
PL193365B1 (pl) 2007-02-28
WO1997037688A2 (fr) 1997-10-16
CA2650637A1 (fr) 1997-10-16
BR9708517A (pt) 1999-08-03
CN1215338A (zh) 1999-04-28
AU713277B2 (en) 1999-11-25
CZ297941B6 (cs) 2007-05-02
EP1192951A3 (fr) 2004-04-21
JP2008195736A (ja) 2008-08-28
PL189066B1 (pl) 2005-06-30
CY2300B1 (en) 2003-07-04
NZ330774A (en) 1999-06-29
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WO1997037688A3 (fr) 1998-03-05
EP0914158B2 (fr) 2006-01-25
CZ288698A3 (cs) 1998-12-16
DE69713890T3 (de) 2006-09-07
EP2253327A1 (fr) 2010-11-24
JPH09323940A (ja) 1997-12-16
CA2577233A1 (fr) 1997-10-16
SI0914158T1 (en) 2002-12-31
SI0914158T2 (sl) 2006-04-30
ATE220333T1 (de) 2002-07-15
KR19990087076A (ko) 1999-12-15
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EP1192951A2 (fr) 2002-04-03
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AU2178097A (en) 1997-10-29
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