NO317947B1 - Hemmere av interleukin-1<beta> omdannende enzym - Google Patents
Hemmere av interleukin-1<beta> omdannende enzym Download PDFInfo
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- NO317947B1 NO317947B1 NO19965365A NO965365A NO317947B1 NO 317947 B1 NO317947 B1 NO 317947B1 NO 19965365 A NO19965365 A NO 19965365A NO 965365 A NO965365 A NO 965365A NO 317947 B1 NO317947 B1 NO 317947B1
- Authority
- NO
- Norway
- Prior art keywords
- group
- optionally substituted
- phenyl
- alkyl
- amino
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/0202—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-X-X-C(=0)-, X being an optionally substituted carbon atom or a heteroatom, e.g. beta-amino acids
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/06—Tripeptides
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/07—Tetrapeptides
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
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- A—HUMAN NECESSITIES
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US08/440,898 US5847135A (en) | 1994-06-17 | 1995-05-25 | Inhibitors of interleukin-1β converting enzyme |
PCT/US1995/007617 WO1995035308A1 (en) | 1994-06-17 | 1995-06-16 | INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME |
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JPH0789951A (ja) * | 1993-06-03 | 1995-04-04 | Sterling Winthrop Inc | インターロイキン−1β転換酵素阻害剤 |
JPH0725887A (ja) * | 1993-06-04 | 1995-01-27 | Sterling Winthrop Inc | インターロイキン−1β転換酵素阻害剤 |
DE69408598T2 (de) * | 1993-06-08 | 1998-09-17 | Vertex Pharmaceuticals Inc Cam | Pyridazine als Interleukin-1-beta Verwandlungsenzym Inhibitoren |
US6083735A (en) * | 1993-06-24 | 2000-07-04 | The General Hospital Corporation | Programmed cell death genes and proteins |
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CA2186511C (en) * | 1994-03-31 | 2009-02-10 | Roland E. Dolle | Pyrimidinyl derivatives as interleukin inhibitors |
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US5565430A (en) * | 1994-08-02 | 1996-10-15 | Sterling Winthrop Inc. | Azaaspartic acid analogs as interleukin-1β converting enzyme inhibitors |
US5498616A (en) * | 1994-11-04 | 1996-03-12 | Cephalon, Inc. | Cysteine protease and serine protease inhibitors |
US5585537A (en) * | 1995-03-03 | 1996-12-17 | Pioneer Hi-Bred International, Inc. | Hybrid maize plant & seed (3753) |
-
1994
- 1994-06-17 US US08/261,452 patent/US5756466A/en not_active Expired - Lifetime
-
1995
- 1995-03-17 US US08/405,581 patent/US5656627A/en not_active Expired - Lifetime
- 1995-06-05 US US08/460,973 patent/US6025147A/en not_active Expired - Lifetime
- 1995-06-05 US US08/465,216 patent/US6103711A/en not_active Expired - Lifetime
- 1995-06-15 ZA ZA954988A patent/ZA954988B/xx unknown
- 1995-06-16 PL PL95354005A patent/PL193391B1/pl not_active IP Right Cessation
- 1995-06-16 EP EP09004745A patent/EP2123665A3/en not_active Withdrawn
- 1995-06-16 KR KR10-2004-7016887A patent/KR100478323B1/ko not_active IP Right Cessation
- 1995-06-16 EP EP03022215A patent/EP1394175A1/en not_active Withdrawn
- 1995-06-16 TN TNTNSN95066A patent/TNSN95066A1/fr unknown
- 1995-06-16 UA UA97010184A patent/UA66745C2/xx unknown
-
1996
- 1996-12-13 NO NO19965365A patent/NO317947B1/no not_active IP Right Cessation
-
2008
- 2008-06-25 JP JP2008166634A patent/JP2008291039A/ja not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
EP2123665A3 (en) | 2010-02-03 |
EP2123665A2 (en) | 2009-11-25 |
JP2008291039A (ja) | 2008-12-04 |
KR100478323B1 (ko) | 2005-03-24 |
TNSN95066A1 (fr) | 1996-02-06 |
PL193391B1 (pl) | 2007-02-28 |
US5756466A (en) | 1998-05-26 |
US6103711A (en) | 2000-08-15 |
US6025147A (en) | 2000-02-15 |
UA66745C2 (en) | 2004-06-15 |
NO965365D0 (no) | 1996-12-13 |
US5656627A (en) | 1997-08-12 |
ZA954988B (en) | 1996-12-17 |
NO965365L (no) | 1997-02-17 |
EP1394175A1 (en) | 2004-03-03 |
KR20040098075A (ko) | 2004-11-18 |
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