NO315855B1 - Kondenserte 1,2,4-tiadiazinderivater, fremgangsmåte for deres fremstilling,anvendelse derav til fremstilling av medikamenter, samtfarmasöytiske preparater som omfatter derivatene, og fremgangsmåte for fremstilling avpreparatene - Google Patents
Kondenserte 1,2,4-tiadiazinderivater, fremgangsmåte for deres fremstilling,anvendelse derav til fremstilling av medikamenter, samtfarmasöytiske preparater som omfatter derivatene, og fremgangsmåte for fremstilling avpreparatene Download PDFInfo
- Publication number
- NO315855B1 NO315855B1 NO19983286A NO983286A NO315855B1 NO 315855 B1 NO315855 B1 NO 315855B1 NO 19983286 A NO19983286 A NO 19983286A NO 983286 A NO983286 A NO 983286A NO 315855 B1 NO315855 B1 NO 315855B1
- Authority
- NO
- Norway
- Prior art keywords
- compound
- formula
- thiadiazine
- thieno
- dioxide
- Prior art date
Links
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Classifications
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/12—Antidiarrhoeals
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
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- A61P9/08—Vasodilators for multiple indications
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Diabetes (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Urology & Nephrology (AREA)
- Emergency Medicine (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pulmonology (AREA)
- Dermatology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (9)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DK4196 | 1996-01-17 | ||
DK25296 | 1996-03-05 | ||
DK25196 | 1996-03-05 | ||
DK25096 | 1996-03-05 | ||
DK25396 | 1996-03-05 | ||
DK25696 | 1996-03-05 | ||
DK25996 | 1996-03-05 | ||
DK90396 | 1996-08-27 | ||
PCT/DK1997/000019 WO1997026265A1 (fr) | 1996-01-17 | 1997-01-16 | Derives de 1,2,4-thiadiazine fusionnee et de 1,4-thiazine fusionnee, leur preparation et utilisation |
Publications (3)
Publication Number | Publication Date |
---|---|
NO983286D0 NO983286D0 (no) | 1998-07-16 |
NO983286L NO983286L (no) | 1998-09-16 |
NO315855B1 true NO315855B1 (no) | 2003-11-03 |
Family
ID=27570780
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO19983286A NO315855B1 (no) | 1996-01-17 | 1998-07-16 | Kondenserte 1,2,4-tiadiazinderivater, fremgangsmåte for deres fremstilling,anvendelse derav til fremstilling av medikamenter, samtfarmasöytiske preparater som omfatter derivatene, og fremgangsmåte for fremstilling avpreparatene |
Country Status (14)
Country | Link |
---|---|
US (1) | US5889002A (fr) |
EP (1) | EP0876379A1 (fr) |
JP (1) | JP3071832B2 (fr) |
KR (1) | KR19990077319A (fr) |
CN (1) | CN1158290C (fr) |
AU (1) | AU727775B2 (fr) |
BR (1) | BR9707003A (fr) |
CA (1) | CA2241567A1 (fr) |
CZ (1) | CZ220498A3 (fr) |
HU (1) | HUP9902056A3 (fr) |
IL (1) | IL125071A0 (fr) |
NO (1) | NO315855B1 (fr) |
PL (1) | PL327938A1 (fr) |
WO (1) | WO1997026265A1 (fr) |
Families Citing this family (189)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6225310B1 (en) | 1996-01-17 | 2001-05-01 | Novo Nordisk A/S | Fused 1,2,4-thiadiazine derivatives, their preparation and use |
AUPO227896A0 (en) * | 1996-09-13 | 1996-10-03 | Fujisawa Pharmaceutical Co., Ltd. | Novel compounds and their preparation |
ES2136013B1 (es) * | 1997-04-15 | 2000-07-01 | Consejo Superior Investigacion | Derivados de tieno y pirazolo (1,2,4) tiadiazina-1,1-dioxido farmacologicamente activos. |
CA2294830A1 (fr) * | 1997-07-16 | 1999-01-28 | John Bondo Hansen | Derives de 1,2,4-thiadiazine fusionnee, leur preparation et utilisation |
WO1999032494A1 (fr) * | 1997-12-19 | 1999-07-01 | Novo Nordisk A/S | Derives condenses de 1,2,4-thiadizine, leur preparation et leur utilisation |
US6329367B1 (en) | 1998-12-18 | 2001-12-11 | Novo Nordisk A/S | Fused 1,2,4-thiadiazine derivatives, their preparation and use |
DK1140945T3 (da) * | 1998-12-18 | 2003-09-15 | Novo Nordisk As | Kondenserede 1,2,4-thiadiazinderivater, deres fremstilling og anvendelse |
US6232310B1 (en) | 1999-03-12 | 2001-05-15 | Novo Nordisk A/S | Fused 1,4-thiazine-2-carbonitrile derivatives, their preparation and use |
WO2000055147A1 (fr) * | 1999-03-12 | 2000-09-21 | Novo Nordisk A/S | Derives de 1,4-thiazine-2-carbonitrile fusionnes, leur preparation et leur utilisation |
US6197765B1 (en) | 1999-06-08 | 2001-03-06 | Pnina Vardi | Use of diazoxide for the treatment of metabolic syndrome and diabetes complications |
WO2001002410A1 (fr) * | 1999-06-30 | 2001-01-11 | Novo Nordisk A/S | Nouveau procede |
US6878749B2 (en) * | 1999-09-17 | 2005-04-12 | Novartis Ag | Method of treating metabolic disorders, especially diabetes, or a disease or condition associated with diabetes |
WO2002000665A1 (fr) * | 2000-06-26 | 2002-01-03 | Novo Nordisk A/S | Utilisation d'elements d'ouverture du canal a potassium, pour le traitement de l'insulite |
WO2002000223A1 (fr) * | 2000-06-26 | 2002-01-03 | Novo Nordisk A/S | Utilisation d'agonistes des canaux potassiques pour reduire la consommation d'aliments gras |
WO2002050085A1 (fr) * | 2000-12-21 | 2002-06-27 | Novo Nordisk A/S | Nouveau procede de preparation de derives de 1,2,4-thiadiazine condenses |
ATE349425T1 (de) | 2000-12-21 | 2007-01-15 | Sanofi Aventis Deutschland | Neue diphenzylazetidinone, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung zur behandlung von lipidstoffwechselstörungen |
KR20030063462A (ko) | 2000-12-21 | 2003-07-28 | 아벤티스 파마 도이칠란트 게엠베하 | 디페닐 아제티디논 유도체, 이의 제조 방법, 이들화합물을 함유하는 약제 및 이의 용도 |
DE10110747A1 (de) * | 2001-03-07 | 2002-09-12 | Bayer Ag | Substituierte 2,6-Diamino-3,5-dicyano-4-aryl-pyridine und ihre Verwendung |
DE10142660A1 (de) | 2001-08-31 | 2003-03-20 | Aventis Pharma Gmbh | Verwendung von Derivaten von C2-substituierten Indan-1-ol-Systemen zur Herstellung von Medikamenten zur Prophylaxe oder Behandlung von Obesitas |
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EP3596107A1 (fr) | 2017-03-15 | 2020-01-22 | Novo Nordisk A/S | Composés bicycliques aptes à se lier au récepteur de mélanocortine 4 |
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Publication number | Priority date | Publication date | Assignee | Title |
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GB1368948A (en) * | 1970-11-11 | 1974-10-02 | Manuf Prod Pharma | Pyridine derivatives |
US3775312A (en) * | 1971-09-22 | 1973-11-27 | Petro Tex Chem Corp | Treatment of process water |
FR2703051B1 (fr) * | 1993-03-26 | 1995-04-28 | Adir | Nouvelles pyridothiadiazines, leurs procédés de préparation, et les compositions pharmaceutiques qui les contiennent. |
-
1997
- 1997-01-16 CA CA002241567A patent/CA2241567A1/fr not_active Abandoned
- 1997-01-16 IL IL12507197A patent/IL125071A0/xx not_active IP Right Cessation
- 1997-01-16 CN CNB971917493A patent/CN1158290C/zh not_active Expired - Fee Related
- 1997-01-16 WO PCT/DK1997/000019 patent/WO1997026265A1/fr not_active Application Discontinuation
- 1997-01-16 KR KR1019980705466A patent/KR19990077319A/ko not_active Application Discontinuation
- 1997-01-16 EP EP97900934A patent/EP0876379A1/fr not_active Withdrawn
- 1997-01-16 CZ CZ982204A patent/CZ220498A3/cs unknown
- 1997-01-16 PL PL97327938A patent/PL327938A1/xx unknown
- 1997-01-16 JP JP9523981A patent/JP3071832B2/ja not_active Expired - Fee Related
- 1997-01-16 AU AU14371/97A patent/AU727775B2/en not_active Ceased
- 1997-01-16 BR BR9707003A patent/BR9707003A/pt not_active Application Discontinuation
- 1997-01-16 HU HU9902056A patent/HUP9902056A3/hu unknown
- 1997-01-17 US US08/785,438 patent/US5889002A/en not_active Expired - Fee Related
-
1998
- 1998-07-16 NO NO19983286A patent/NO315855B1/no not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
NO983286L (no) | 1998-09-16 |
AU727775B2 (en) | 2000-12-21 |
BR9707003A (pt) | 1999-07-20 |
HUP9902056A2 (hu) | 1999-10-28 |
HUP9902056A3 (en) | 2002-02-28 |
KR19990077319A (ko) | 1999-10-25 |
CN1208417A (zh) | 1999-02-17 |
EP0876379A1 (fr) | 1998-11-11 |
PL327938A1 (en) | 1999-01-04 |
WO1997026265A1 (fr) | 1997-07-24 |
JPH10508881A (ja) | 1998-09-02 |
US5889002A (en) | 1999-03-30 |
JP3071832B2 (ja) | 2000-07-31 |
AU1437197A (en) | 1997-08-11 |
CN1158290C (zh) | 2004-07-21 |
CZ220498A3 (cs) | 1998-11-11 |
CA2241567A1 (fr) | 1997-07-24 |
IL125071A0 (en) | 1999-01-26 |
NO983286D0 (no) | 1998-07-16 |
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