NO309651B1 - (R)-3-(1H-indol-3-yl)-1-[N-(2-metoksybenzyl)acetylamino]-2-[N- - Google Patents
(R)-3-(1H-indol-3-yl)-1-[N-(2-metoksybenzyl)acetylamino]-2-[N- Download PDFInfo
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- NO309651B1 NO309651B1 NO970078A NO970078A NO309651B1 NO 309651 B1 NO309651 B1 NO 309651B1 NO 970078 A NO970078 A NO 970078A NO 970078 A NO970078 A NO 970078A NO 309651 B1 NO309651 B1 NO 309651B1
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- Norway
- Prior art keywords
- mol
- indol
- solution
- methoxybenzyl
- piperidin
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Landscapes
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Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
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US27170894A | 1994-07-12 | 1994-07-12 | |
PCT/US1995/008300 WO1996001819A1 (en) | 1994-07-12 | 1995-06-30 | Heterocyclic tachykinin receptor antagonists |
Publications (3)
Publication Number | Publication Date |
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NO970078L NO970078L (no) | 1997-01-09 |
NO970078D0 NO970078D0 (no) | 1997-01-09 |
NO309651B1 true NO309651B1 (no) | 2001-03-05 |
Family
ID=23036729
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO970078A NO309651B1 (no) | 1994-07-12 | 1997-01-09 | (R)-3-(1H-indol-3-yl)-1-[N-(2-metoksybenzyl)acetylamino]-2-[N- |
Country Status (25)
Country | Link |
---|---|
US (1) | US5530009A (da) |
EP (1) | EP0693489B1 (da) |
JP (1) | JPH10502640A (da) |
CN (1) | CN1067067C (da) |
AT (1) | ATE205491T1 (da) |
AU (1) | AU688072B2 (da) |
BR (1) | BR9508375A (da) |
CA (1) | CA2194471C (da) |
CO (1) | CO4410196A1 (da) |
CZ (1) | CZ288434B6 (da) |
DE (1) | DE69522619T2 (da) |
DK (1) | DK0693489T3 (da) |
ES (1) | ES2163475T3 (da) |
FI (1) | FI970107A (da) |
HU (1) | HUT77948A (da) |
IL (1) | IL114474A (da) |
MX (1) | MX9700271A (da) |
NO (1) | NO309651B1 (da) |
NZ (1) | NZ289652A (da) |
PL (1) | PL180866B1 (da) |
PT (1) | PT693489E (da) |
RU (1) | RU2151769C1 (da) |
TR (1) | TR199500844A1 (da) |
WO (1) | WO1996001819A1 (da) |
ZA (1) | ZA955639B (da) |
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JP2000506527A (ja) * | 1996-03-11 | 2000-05-30 | イーライ・リリー・アンド・カンパニー | 間質性膀胱炎の治療または予防方法 |
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AU7580998A (en) * | 1997-05-21 | 1998-12-11 | Eli Lilly And Company | 3-arylpropylamino neuropeptide y receptor antagonists |
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EP1556054A4 (en) * | 2002-05-29 | 2007-09-05 | Univ California | ANTAGONIZING NK1 RECEPTORS RESTRICT DRUG ABUSE |
KR101389246B1 (ko) | 2004-07-15 | 2014-04-24 | 브리스톨-마이어스스퀴브컴파니 | 아릴- 및 헤테로아릴-치환된 테트라히드로이소퀴놀린, 및 이것의 노르에피네프린, 도파민 및 세로토닌의 재흡수를 차단하기 위한 용도 |
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KR101591656B1 (ko) | 2007-01-10 | 2016-02-19 | 엠에스디 이탈리아 에스.알.엘. | 폴리(adp-리보오스) 폴리머라아제(parp) 억제제로서의 아미드 치환된 인다졸 |
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JP5739415B2 (ja) | 2009-05-12 | 2015-06-24 | ブリストル−マイヤーズ スクウィブ カンパニー | (S)−7−([1,2,4]トリアゾロ[1,5−a]ピリジン−6−イル)−4−(3,4−ジクロロフェニル)−1,2,3,4−テトラヒドロイソキノリンの結晶形態およびその使用 |
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MX2012004377A (es) | 2009-10-14 | 2012-06-01 | Merck Sharp & Dohme | Piperidinas sustituidas que aumentan la actividad de p53 y sus usos. |
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EP2613782B1 (en) | 2010-09-01 | 2016-11-02 | Merck Sharp & Dohme Corp. | Indazole derivatives useful as erk inhibitors |
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US9260471B2 (en) | 2010-10-29 | 2016-02-16 | Sirna Therapeutics, Inc. | RNA interference mediated inhibition of gene expression using short interfering nucleic acids (siNA) |
US9351965B2 (en) | 2010-12-21 | 2016-05-31 | Merck Sharp & Dohme Corp. | Indazole derivatives useful as ERK inhibitors |
AU2012245971A1 (en) | 2011-04-21 | 2013-10-17 | Piramal Enterprises Limited | A crystalline form of a salt of a morpholino sulfonyl indole derivative and a process for its preparation |
WO2013063214A1 (en) | 2011-10-27 | 2013-05-02 | Merck Sharp & Dohme Corp. | Novel compounds that are erk inhibitors |
EP3919620A1 (en) | 2012-05-02 | 2021-12-08 | Sirna Therapeutics, Inc. | Short interfering nucleic acid (sina) compositions |
MX2015004041A (es) | 2012-09-28 | 2015-07-06 | Merck Sharp & Dohme | Compuestos novedosos que son inhibidores de erk. |
CA2892361A1 (en) | 2012-11-28 | 2014-06-05 | Merck Sharp & Dohme Corp. | Use of a wee1 inhibitor for treating a cancer characterized by low pkmyt1 expression levels |
ES2707305T3 (es) | 2012-12-20 | 2019-04-03 | Merck Sharp & Dohme | Imidazopiridinas sustituidas como inhibidores de HDM2 |
WO2014120748A1 (en) | 2013-01-30 | 2014-08-07 | Merck Sharp & Dohme Corp. | 2,6,7,8 substituted purines as hdm2 inhibitors |
EP3041938A1 (en) | 2013-09-03 | 2016-07-13 | Moderna Therapeutics, Inc. | Circular polynucleotides |
WO2019094311A1 (en) | 2017-11-08 | 2019-05-16 | Merck Sharp & Dohme Corp. | Prmt5 inhibitors |
US11981701B2 (en) | 2018-08-07 | 2024-05-14 | Merck Sharp & Dohme Llc | PRMT5 inhibitors |
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EP0104848B1 (en) * | 1982-09-18 | 1986-11-26 | Lillywhites Cantabrian Limited | Display unit |
US5331089A (en) | 1988-03-25 | 1994-07-19 | Merck Sharpe & Dohme, Ltd. | Peptides useful as tachykinin agonists |
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IL99320A (en) * | 1990-09-05 | 1995-07-31 | Sanofi Sa | Arylalkylamines, their preparation and pharmaceutical preparations containing them |
FR2676053B1 (fr) * | 1991-05-03 | 1993-08-27 | Sanofi Elf | Nouveaux composes dialkylenepiperidino et leurs enantiomeres, procede pour leur preparation et compositions pharmaceutiques les contenant. |
FR2676055B1 (fr) * | 1991-05-03 | 1993-09-03 | Sanofi Elf | Composes polycycliques amines et leurs enantiomeres, procede pour leur preparation et compositions pharmaceutiques les contenant. |
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FR2696178B1 (fr) | 1992-09-30 | 1994-12-30 | Sanofi Elf | Amides basiques quaternaires, procédé pour leur préparation et compositions pharmaceutiques en contenant. |
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EP0686629A3 (en) * | 1994-06-10 | 1999-02-10 | Eli Lilly And Company | Cyclohexyl tachykinine receptor antagonists |
-
1995
- 1995-06-30 CN CN95194996A patent/CN1067067C/zh not_active Expired - Fee Related
- 1995-06-30 HU HU9700069A patent/HUT77948A/hu unknown
- 1995-06-30 CA CA002194471A patent/CA2194471C/en not_active Expired - Fee Related
- 1995-06-30 PL PL95318327A patent/PL180866B1/pl unknown
- 1995-06-30 RU RU97102050/04A patent/RU2151769C1/ru active
- 1995-06-30 NZ NZ289652A patent/NZ289652A/en unknown
- 1995-06-30 AU AU29560/95A patent/AU688072B2/en not_active Ceased
- 1995-06-30 JP JP8504355A patent/JPH10502640A/ja not_active Ceased
- 1995-06-30 WO PCT/US1995/008300 patent/WO1996001819A1/en active IP Right Grant
- 1995-06-30 BR BR9508375A patent/BR9508375A/pt not_active Application Discontinuation
- 1995-06-30 CZ CZ199757A patent/CZ288434B6/cs not_active IP Right Cessation
- 1995-06-30 MX MX9700271A patent/MX9700271A/es unknown
- 1995-07-06 ZA ZA955639A patent/ZA955639B/xx unknown
- 1995-07-06 IL IL11447495A patent/IL114474A/xx not_active IP Right Cessation
- 1995-07-07 EP EP95304750A patent/EP0693489B1/en not_active Expired - Lifetime
- 1995-07-07 DE DE69522619T patent/DE69522619T2/de not_active Expired - Fee Related
- 1995-07-07 DK DK95304750T patent/DK0693489T3/da active
- 1995-07-07 PT PT95304750T patent/PT693489E/pt unknown
- 1995-07-07 ES ES95304750T patent/ES2163475T3/es not_active Expired - Lifetime
- 1995-07-07 AT AT95304750T patent/ATE205491T1/de not_active IP Right Cessation
- 1995-07-10 CO CO95029998A patent/CO4410196A1/es unknown
- 1995-07-11 TR TR95/00844A patent/TR199500844A1/xx unknown
-
1996
- 1996-06-05 US US08/462,413 patent/US5530009A/en not_active Expired - Fee Related
-
1997
- 1997-01-09 NO NO970078A patent/NO309651B1/no not_active IP Right Cessation
- 1997-01-10 FI FI970107A patent/FI970107A/fi unknown
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