NO304515B1 - FremgangsmÕte for fremstilling av <beta>-fenylisoserin og analoger derav samt mellomprodukt - Google Patents

FremgangsmÕte for fremstilling av <beta>-fenylisoserin og analoger derav samt mellomprodukt

Info

Publication number
NO304515B1
NO304515B1 NO943280A NO943280A NO304515B1 NO 304515 B1 NO304515 B1 NO 304515B1 NO 943280 A NO943280 A NO 943280A NO 943280 A NO943280 A NO 943280A NO 304515 B1 NO304515 B1 NO 304515B1
Authority
NO
Norway
Prior art keywords
pct
phenylisoserine
general formula
beta
analogs
Prior art date
Application number
NO943280A
Other languages
English (en)
Other versions
NO943280D0 (no
NO943280L (no
Inventor
Jean-Dominique Bourzat
On Alain Commer
Original Assignee
Rh Ne Poulenc Rorer Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rh Ne Poulenc Rorer Sa filed Critical Rh Ne Poulenc Rorer Sa
Publication of NO943280D0 publication Critical patent/NO943280D0/no
Publication of NO943280L publication Critical patent/NO943280L/no
Publication of NO304515B1 publication Critical patent/NO304515B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/14—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof
    • C07C227/18—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof by reactions involving amino or carboxyl groups, e.g. hydrolysis of esters or amides, by formation of halides, salts or esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/22—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from lactams, cyclic ketones or cyclic oximes, e.g. by reactions involving Beckmann rearrangement
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Epoxy Compounds (AREA)
  • Steroid Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
NO943280A 1992-03-10 1994-09-05 FremgangsmÕte for fremstilling av <beta>-fenylisoserin og analoger derav samt mellomprodukt NO304515B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9202821A FR2688499B1 (fr) 1992-03-10 1992-03-10 Procede de preparation de la beta-phenylisoserine et de ses analogues.
PCT/FR1993/000224 WO1993017997A1 (fr) 1992-03-10 1993-03-08 PROCEDE DE PREPARATION DE LA β-PHENYLISOSERINE ET DE SES ANALOGUES

Publications (3)

Publication Number Publication Date
NO943280D0 NO943280D0 (no) 1994-09-05
NO943280L NO943280L (no) 1994-09-05
NO304515B1 true NO304515B1 (no) 1999-01-04

Family

ID=9427518

Family Applications (1)

Application Number Title Priority Date Filing Date
NO943280A NO304515B1 (no) 1992-03-10 1994-09-05 FremgangsmÕte for fremstilling av <beta>-fenylisoserin og analoger derav samt mellomprodukt

Country Status (25)

Country Link
US (2) US5608102A (no)
EP (1) EP0630365B1 (no)
JP (1) JP3278768B2 (no)
KR (1) KR100272650B1 (no)
AT (1) ATE159512T1 (no)
AU (1) AU667886B2 (no)
CA (1) CA2130333C (no)
CZ (1) CZ283613B6 (no)
DE (1) DE69314779T2 (no)
DK (1) DK0630365T3 (no)
ES (1) ES2109509T3 (no)
FI (1) FI113640B (no)
FR (1) FR2688499B1 (no)
GE (1) GEP19981430B (no)
GR (1) GR3025117T3 (no)
HU (1) HU213621B (no)
MX (1) MX9301268A (no)
NO (1) NO304515B1 (no)
NZ (1) NZ249899A (no)
PL (1) PL171551B1 (no)
RU (1) RU2103258C1 (no)
SK (1) SK281297B6 (no)
TW (1) TW252971B (no)
WO (1) WO1993017997A1 (no)
ZA (1) ZA931677B (no)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI9520078B (sl) * 1994-07-26 1998-12-31 Indena S.P.A. Polsintetski taksani z antitumorsko aktivnostjo
US6765015B2 (en) * 1995-12-13 2004-07-20 Xechem International, Inc. Halogenated paclitaxel derivatives
AU739303B2 (en) 1997-08-21 2001-10-11 Florida State University Method for the synthesis of taxanes
WO1999025334A1 (en) * 1997-11-19 1999-05-27 Xechem International, Inc. Halogenated paclitaxel derivatives
ITMI991483A1 (it) 1999-07-06 2001-01-06 Indena Spa Derivati tassanici e procedimenti per la loro preparazione
AU775373B2 (en) 1999-10-01 2004-07-29 Immunogen, Inc. Compositions and methods for treating cancer using immunoconjugates and chemotherapeutic agents
JP2002080435A (ja) * 2000-06-26 2002-03-19 Kanegafuchi Chem Ind Co Ltd ３−アミノ−２−ヒドロキシプロピオン酸誘導体の製造法
JP4142444B2 (ja) 2001-03-07 2008-09-03 第一三共株式会社 ２−アゼチジノン誘導体の製造方法
SI1961735T1 (sl) * 2007-02-22 2010-01-29 Indena Spa Postopek za pripravo acetatne soli (2r,3s)-3-fenilizoserin-metilestra
ES2389518T3 (es) 2008-01-18 2012-10-26 Indena S.P.A. Formas sólidas de ortataxel
CN102408356A (zh) * 2011-09-28 2012-04-11 北京东方协和医药生物技术有限公司 一种多西他赛手性侧链中间体的制备方法
KR101900584B1 (ko) * 2014-02-03 2018-09-19 콰드리가 바이오사이언시스 인코포레이티드 화학치료제로서의 베타-치환된 베타-아미노산 및 유사체
CN111100026A (zh) * 2019-12-30 2020-05-05 重庆市碚圣医药科技股份有限公司 一种紫杉醇恶唑环侧链中间体的制备方法
CN112574134A (zh) * 2020-12-30 2021-03-30 重庆市碚圣医药科技股份有限公司 一种多西紫杉醇侧链的合成方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2629819B1 (fr) * 1988-04-06 1990-11-16 Rhone Poulenc Sante Procede de preparation de derives de la baccatine iii et de la desacetyl-10 baccatine iii
IT1231751B (it) * 1989-04-12 1991-12-21 Sigma Tau Ind Farmaceuti Procedimento per la produzione di r(+) amminocarnitina e s(-) amminocarnitina
US5175315A (en) * 1989-05-31 1992-12-29 Florida State University Method for preparation of taxol using β-lactam
US5304670A (en) * 1989-08-23 1994-04-19 Centre National De La Recherche Scientifique Process for the enantioselective preparation of phenylisoserine derivatives
FR2658510B1 (fr) * 1990-02-21 1992-04-30 Rhone Poulenc Sante Nouveau derive de la beta-phenylisoserine, sa preparation et son emploi.
US5294737A (en) * 1992-02-27 1994-03-15 The Research Foundation State University Of New York Process for the production of chiral hydroxy-β-lactams and hydroxyamino acids derived therefrom

Also Published As

Publication number Publication date
NO943280D0 (no) 1994-09-05
DE69314779D1 (de) 1997-11-27
WO1993017997A1 (fr) 1993-09-16
ATE159512T1 (de) 1997-11-15
CZ283613B6 (cs) 1998-05-13
GEP19981430B (en) 1998-10-30
KR950700234A (ko) 1995-01-16
RU2103258C1 (ru) 1998-01-27
DK0630365T3 (da) 1998-03-02
GR3025117T3 (en) 1998-01-30
HU213621B (en) 1997-08-28
FI113640B (fi) 2004-05-31
EP0630365A1 (fr) 1994-12-28
SK281297B6 (sk) 2001-02-12
FR2688499A1 (fr) 1993-09-17
CA2130333A1 (fr) 1993-09-16
EP0630365B1 (fr) 1997-10-22
NO943280L (no) 1994-09-05
FI944169A0 (fi) 1994-09-09
RU94045799A (ru) 1996-07-20
KR100272650B1 (ko) 2000-11-15
FR2688499B1 (fr) 1994-05-06
MX9301268A (es) 1993-09-01
US5608102A (en) 1997-03-04
HUT68540A (en) 1995-06-28
ES2109509T3 (es) 1998-01-16
CA2130333C (fr) 2002-11-26
HU9402590D0 (en) 1994-11-28
AU667886B2 (en) 1996-04-18
FI944169A (fi) 1994-09-09
JPH07504425A (ja) 1995-05-18
AU3755793A (en) 1993-10-05
NZ249899A (en) 1996-01-26
CZ218594A3 (en) 1995-11-15
TW252971B (no) 1995-08-01
ZA931677B (en) 1993-10-06
US5763628A (en) 1998-06-09
JP3278768B2 (ja) 2002-04-30
PL171551B1 (pl) 1997-05-30
SK108594A3 (en) 1995-02-08
DE69314779T2 (de) 1998-02-26

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