SI1961735T1 - Postopek za pripravo acetatne soli (2r,3s)-3-fenilizoserin-metilestra - Google Patents

Postopek za pripravo acetatne soli (2r,3s)-3-fenilizoserin-metilestra

Info

Publication number
SI1961735T1
SI1961735T1 SI200730119T SI200730119T SI1961735T1 SI 1961735 T1 SI1961735 T1 SI 1961735T1 SI 200730119 T SI200730119 T SI 200730119T SI 200730119 T SI200730119 T SI 200730119T SI 1961735 T1 SI1961735 T1 SI 1961735T1
Authority
SI
Slovenia
Prior art keywords
methyl ester
acetate salt
preparation
ester acetate
phenylisoserine
Prior art date
Application number
SI200730119T
Other languages
English (en)
Inventor
Daniele Ciceri
Bruno Gabetta
Nicola Vignola
Frieder Mitzel
Beat T Weber
Original Assignee
Indena Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Indena Spa filed Critical Indena Spa
Publication of SI1961735T1 publication Critical patent/SI1961735T1/sl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/30Preparation of optical isomers
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/34Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00Carboxylic acid amides
    • C07C233/01Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/02Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having nitrogen atoms of carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • C07C233/08Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having nitrogen atoms of carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with carbon atoms of carboxamide groups bound to acyclic carbon atoms of a saturated carbon skeleton containing rings
SI200730119T 2007-02-22 2007-02-22 Postopek za pripravo acetatne soli (2r,3s)-3-fenilizoserin-metilestra SI1961735T1 (sl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP07003642A EP1961735B1 (en) 2007-02-22 2007-02-22 Process for the preparation of (2r,3s)-3-phenylisoserine methyl ester acetate salt

Publications (1)

Publication Number Publication Date
SI1961735T1 true SI1961735T1 (sl) 2010-01-29

Family

ID=38230004

Family Applications (1)

Application Number Title Priority Date Filing Date
SI200730119T SI1961735T1 (sl) 2007-02-22 2007-02-22 Postopek za pripravo acetatne soli (2r,3s)-3-fenilizoserin-metilestra

Country Status (19)

Country Link
US (1) US8106231B2 (sl)
EP (1) EP1961735B1 (sl)
JP (1) JP5352478B2 (sl)
KR (1) KR101499817B1 (sl)
CN (1) CN101675028B (sl)
AT (1) ATE449062T1 (sl)
AU (1) AU2008217318B2 (sl)
CA (1) CA2679159C (sl)
DE (1) DE602007003312D1 (sl)
DK (1) DK1961735T3 (sl)
ES (1) ES2333266T3 (sl)
HK (1) HK1121735A1 (sl)
IL (1) IL200537A (sl)
MX (1) MX2009008985A (sl)
PL (1) PL1961735T3 (sl)
PT (1) PT1961735E (sl)
RU (1) RU2459802C2 (sl)
SI (1) SI1961735T1 (sl)
WO (1) WO2008101608A1 (sl)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK2380871T3 (da) * 2010-04-15 2013-04-08 Indena Spa Fremgangsmåde til fremstilling af isoserin-derivater
EP2399904A1 (en) * 2010-05-26 2011-12-28 Nabriva Therapeutics AG Process for the preparation of pleuromutilins

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2275378A (en) * 1937-09-10 1942-03-03 Rohm & Haas Polyalkylene ether disulphonyl halides and a process of making them
US4695589A (en) * 1976-06-25 1987-09-22 Sterling Drug Inc. Alpha-(aminoalkyl-4-hydroxy-3-(alkylthio)benzenemethanols
FR2415640A1 (fr) * 1978-01-27 1979-08-24 Nativelle Sa Ets Derives d'amino-3-cardenolides, procede pour leur preparation, et medicaments les contenant
ZA794872B (en) * 1978-09-20 1980-11-26 Schering Corp A phenylalkylaminoethylsalicylamide,its preparation and pharmaceutical compositions containing it
FR2688499B1 (fr) * 1992-03-10 1994-05-06 Rhone Poulenc Rorer Sa Procede de preparation de la beta-phenylisoserine et de ses analogues.
JPH06271512A (ja) * 1993-03-22 1994-09-27 Toray Ind Inc 光学活性トランス−1,2−ジアミノ−4−シクロヘキセンの製造方法
US6025516A (en) * 1998-10-14 2000-02-15 Chiragene, Inc. Resolution of 2-hydroxy-3-amino-3-phenylpropionamide and its conversion to C-13 sidechain of taxanes
EP1383754B1 (en) * 2001-03-23 2011-02-23 ScinoPharm Taiwan, Ltd. Process for making taxane derivatives
JP2005500322A (ja) * 2001-07-03 2005-01-06 アルタナ ファルマ アクチエンゲゼルシャフト 3−フェニルイソセリンの製法
CN1315777C (zh) * 2003-01-16 2007-05-16 东丽泛应化学(股) 旋光二酰基酒石酸的回收方法
FR2861073B1 (fr) * 2003-10-17 2006-01-06 Sanofi Synthelabo Derives de n-[heteroaryl(piperidin-2-yl)methyl]benzamide, leur preparation et leur application en therapeutique
JP2008507487A (ja) * 2004-07-23 2008-03-13 ディーエスエム アイピー アセッツ ビー.ブイ. (2r,3r)−2−ヒドロキシ−3−アミノ−3−アリール−プロピオンアミドおよび(2r,3r)−2−ヒドロキシ−3−アミノ−3−アリール−プロピオン酸アルキルエステルの調製方法
AR057061A1 (es) * 2005-06-16 2007-11-14 Altana Pharma Ag Espiro-bencimidazoles farmaceuticamente activos y su uso en la fabricacion de medicamentos
JP2009114065A (ja) * 2006-02-21 2009-05-28 Kaneka Corp (2r,3r)および(2s,3s)−3−フェニルイソセリン誘導体の製造法

Also Published As

Publication number Publication date
KR101499817B1 (ko) 2015-03-06
ES2333266T3 (es) 2010-02-18
ATE449062T1 (de) 2009-12-15
DK1961735T3 (da) 2010-03-29
WO2008101608A1 (en) 2008-08-28
CN101675028A (zh) 2010-03-17
PL1961735T3 (pl) 2010-04-30
US8106231B2 (en) 2012-01-31
RU2009131595A (ru) 2011-02-27
CN101675028B (zh) 2013-01-30
US20100168460A1 (en) 2010-07-01
IL200537A (en) 2013-03-24
MX2009008985A (es) 2009-09-02
RU2459802C2 (ru) 2012-08-27
CA2679159A1 (en) 2008-08-28
AU2008217318B2 (en) 2013-01-17
JP5352478B2 (ja) 2013-11-27
CA2679159C (en) 2015-11-03
JP2010519262A (ja) 2010-06-03
KR20090113859A (ko) 2009-11-02
EP1961735A1 (en) 2008-08-27
IL200537A0 (en) 2010-04-29
EP1961735B1 (en) 2009-11-18
PT1961735E (pt) 2009-12-21
DE602007003312D1 (de) 2009-12-31
HK1121735A1 (en) 2009-04-30
AU2008217318A1 (en) 2008-08-28

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