NO20075385L - 7-aminoalkylidenyl-heterocykliske kinoloner og naftyridoner - Google Patents
7-aminoalkylidenyl-heterocykliske kinoloner og naftyridonerInfo
- Publication number
- NO20075385L NO20075385L NO20075385A NO20075385A NO20075385L NO 20075385 L NO20075385 L NO 20075385L NO 20075385 A NO20075385 A NO 20075385A NO 20075385 A NO20075385 A NO 20075385A NO 20075385 L NO20075385 L NO 20075385L
- Authority
- NO
- Norway
- Prior art keywords
- aminoalkylidenyl
- naphthyridones
- quinolones
- heterocyclic
- heterocyclic quinolones
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Abstract
Foreliggende oppfinnelse angår forbindelser som har strukturen i henhold til formel (I), hvor n, m, z, R, R2, R3, R4, R5, R6, A, E, X, Y, a og b er som definert i beskrivelsen; eller en optisk isomer, diastereomer, enantiomer, farmasøytisk akseptabelt salt, hydrat eller prodrug derav.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US11/084,987 US7732612B2 (en) | 2004-09-09 | 2005-03-21 | 7-amino alkylidenyl-heterocyclic quinolones and naphthyridones |
PCT/US2006/003657 WO2006101603A1 (en) | 2005-03-21 | 2006-02-02 | 7-amino alkylidenyl-heterocyclic quinolones and naphthyridones |
Publications (2)
Publication Number | Publication Date |
---|---|
NO20075385L true NO20075385L (no) | 2007-12-14 |
NO340833B1 NO340833B1 (no) | 2017-06-26 |
Family
ID=36648281
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20075385A NO340833B1 (no) | 2005-03-21 | 2007-10-22 | 7-aminoalkylidenylheterocykliske kinolon- og naftyridon-forbindelser og farmasøytiske sammensetninger |
Country Status (22)
Country | Link |
---|---|
US (1) | US7732612B2 (no) |
EP (1) | EP1861401B1 (no) |
JP (1) | JP4977684B2 (no) |
KR (1) | KR101323665B1 (no) |
CN (1) | CN101248070B (no) |
AR (1) | AR053342A1 (no) |
AU (1) | AU2006227984A1 (no) |
BR (1) | BRPI0609426B8 (no) |
CA (1) | CA2602140C (no) |
CR (1) | CR9458A (no) |
DK (1) | DK1861401T3 (no) |
EA (1) | EA014554B1 (no) |
ES (1) | ES2561834T3 (no) |
IL (1) | IL186041A (no) |
MX (1) | MX2007011774A (no) |
MY (1) | MY147638A (no) |
NO (1) | NO340833B1 (no) |
NZ (1) | NZ561651A (no) |
TW (1) | TWI444380B (no) |
UA (1) | UA93672C2 (no) |
WO (1) | WO2006101603A1 (no) |
ZA (1) | ZA200708868B (no) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7913302B2 (en) * | 2004-05-02 | 2011-03-22 | Markmonitor, Inc. | Advanced responses to online fraud |
US20090156577A1 (en) * | 2004-09-09 | 2009-06-18 | Benjamin Davis | 7-amino alkylidenyl-heterocyclic quinolones and naphthyridones |
EA200801128A1 (ru) * | 2005-10-21 | 2008-10-30 | Глэксо Груп Лимитед | Пери-конденсированные трициклические соединения, полезные в качестве антибактериальных средств |
EP1963324B1 (en) | 2005-12-22 | 2010-04-21 | Glaxo Group Limited | Heterocyclic compounds, their preparation and their use as antibacterials |
ATE507219T1 (de) * | 2006-03-28 | 2011-05-15 | Warner Chilcott Co Llc | Malatsalze und polymorphe von (3s,5s)-7-ä3-amino- 5-methyl-piperidinylü-1-cyclopropyl-1,4-dihydro 8-methoxy-4-oxo-3-chinolincarbonsäure |
KR101084521B1 (ko) | 2006-03-28 | 2011-11-18 | 워너 칠콧 컴퍼니 엘엘씨 | 퀴놀론 중간체를 제조하기 위한 커플링 방법 |
KR101245938B1 (ko) | 2008-05-29 | 2013-03-21 | 블루스타 실리콘즈 프랑스 에스에이에스 | 수계, 특히 해양 용도를 위한 방오 특성을 가진 물품 |
EA201490435A1 (ru) | 2011-08-10 | 2014-06-30 | ЯНССЕН Ар ЭНД Ди АЙРЛЭНД | Антибактериальные 3,4-дигидро-1н-[1,8]нафтиридиноны, замещенные пиперидинилом |
JO3611B1 (ar) | 2011-08-10 | 2020-08-27 | Janssen Sciences Ireland Uc | سايكلو بنتا (سي (بيرول 4,3 ثاني هيدرو 1 hمستبدله [8,1] نافثيريدينونات مضادة للجراثيم |
CN105237464B (zh) * | 2011-09-30 | 2018-06-01 | 詹森药业有限公司 | 用于制备2-[(2e)-2-氟-2-(3-亚哌啶基)乙基]-1h-异吲哚-1,3(2h)-二酮的改进方法 |
US9388178B2 (en) * | 2012-12-04 | 2016-07-12 | Mankind Research Centre | Process for the preparation of moxifloxacin hydrochloride |
WO2016079757A2 (en) * | 2014-11-19 | 2016-05-26 | Symed Labs Limited | Novel processes for preparing 5-hydroxymethyl-oxazolidin-2-one derivatives |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK164287A (da) | 1986-03-31 | 1987-10-01 | Sankyo Co | Quinolin-3-carboxylsyrederivater og fremgangsmaade til fremstilling deraf og deres anvendelse |
JPH0262875A (ja) * | 1988-05-23 | 1990-03-02 | Wakunaga Pharmaceut Co Ltd | 新規イソインドリン誘導体 |
CA1332605C (en) * | 1988-10-03 | 1994-10-18 | Yasuhiro Nishitani | Pyridonecarboxylic acids |
US5580872A (en) * | 1990-05-02 | 1996-12-03 | Abbott Laboratories | Quinolizinone type compounds |
FR2692577B1 (fr) * | 1992-05-26 | 1996-02-02 | Bouchara Sa | Nouvelles quinolones fluorees, leur procede de preparation et les compositions pharmaceutiques en renfermant. |
NO304832B1 (no) * | 1992-05-27 | 1999-02-22 | Ube Industries | Aminokinolonderivater samt middel mot HIV |
JPH07300472A (ja) * | 1992-12-28 | 1995-11-14 | Korea Res Inst Chem Technol | 新規キノロンカルボン酸誘導体およびその製造方法 |
JPH06263754A (ja) | 1993-03-12 | 1994-09-20 | Hokuriku Seiyaku Co Ltd | 7−アミノピロリジニルキノリン−3−カルボン酸誘導体 |
CZ299554B6 (cs) | 1997-09-15 | 2008-09-03 | The Procter & Gamble Company | Sloucenina se strukturou chinolonu, farmaceutickýprostredek ji obsahující a použití |
US6878713B2 (en) * | 2001-04-25 | 2005-04-12 | Wockhardt Limited | Generation triple-targeting, chiral, broad-spectrum antimicrobial 7-substituted piperidino-quinolone carboxylic acid derivatives, their preparation, compositions and use as medicaments |
US6964966B2 (en) | 2001-04-25 | 2005-11-15 | Wockhardt Limited | Generation triple-targeting, chiral, broad-spectrum antimicrobial 7-substituted piperidino-quinolone carboxylic acid derivatives, their preparation, compositions and use as medicaments |
BRPI0414573A (pt) * | 2003-09-22 | 2006-11-07 | Janssen Pharmaceutica Nv | 7-amino alquilidenil-quinolonas e naftiridonas heterocìclicas |
-
2005
- 2005-03-21 US US11/084,987 patent/US7732612B2/en not_active Expired - Fee Related
-
2006
- 2006-02-02 JP JP2008502985A patent/JP4977684B2/ja not_active Expired - Fee Related
- 2006-02-02 CA CA2602140A patent/CA2602140C/en not_active Expired - Fee Related
- 2006-02-02 EA EA200702039A patent/EA014554B1/ru unknown
- 2006-02-02 BR BRPI0609426A patent/BRPI0609426B8/pt not_active IP Right Cessation
- 2006-02-02 WO PCT/US2006/003657 patent/WO2006101603A1/en active Application Filing
- 2006-02-02 DK DK06720136.8T patent/DK1861401T3/en active
- 2006-02-02 NZ NZ561651A patent/NZ561651A/en not_active IP Right Cessation
- 2006-02-02 MX MX2007011774A patent/MX2007011774A/es active IP Right Grant
- 2006-02-02 AU AU2006227984A patent/AU2006227984A1/en not_active Abandoned
- 2006-02-02 UA UAA200710571A patent/UA93672C2/ru unknown
- 2006-02-02 CN CN200680017405XA patent/CN101248070B/zh not_active Expired - Fee Related
- 2006-02-02 EP EP06720136.8A patent/EP1861401B1/en active Active
- 2006-02-02 ES ES06720136.8T patent/ES2561834T3/es active Active
- 2006-02-02 KR KR1020077024070A patent/KR101323665B1/ko active IP Right Grant
- 2006-03-20 AR ARP060101080A patent/AR053342A1/es active IP Right Grant
- 2006-03-20 TW TW095109374A patent/TWI444380B/zh not_active IP Right Cessation
- 2006-03-21 MY MYPI20061247A patent/MY147638A/en unknown
-
2007
- 2007-09-18 IL IL186041A patent/IL186041A/en active IP Right Grant
- 2007-10-19 CR CR9458A patent/CR9458A/es not_active Application Discontinuation
- 2007-10-19 ZA ZA200708868A patent/ZA200708868B/xx unknown
- 2007-10-22 NO NO20075385A patent/NO340833B1/no not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
TWI444380B (zh) | 2014-07-11 |
EP1861401A1 (en) | 2007-12-05 |
CN101248070B (zh) | 2011-12-14 |
CN101248070A (zh) | 2008-08-20 |
CA2602140A1 (en) | 2006-09-28 |
UA93672C2 (en) | 2011-03-10 |
AR053342A1 (es) | 2007-05-02 |
BRPI0609426A2 (pt) | 2010-04-06 |
IL186041A (en) | 2016-05-31 |
CA2602140C (en) | 2015-04-14 |
US20060052359A1 (en) | 2006-03-09 |
TW200700418A (en) | 2007-01-01 |
KR20070113304A (ko) | 2007-11-28 |
ZA200708868B (en) | 2009-01-28 |
JP4977684B2 (ja) | 2012-07-18 |
EP1861401B1 (en) | 2015-11-18 |
CR9458A (es) | 2008-09-09 |
BRPI0609426B8 (pt) | 2021-05-25 |
MX2007011774A (es) | 2008-03-10 |
NZ561651A (en) | 2011-09-30 |
US7732612B2 (en) | 2010-06-08 |
ES2561834T3 (es) | 2016-03-01 |
AU2006227984A1 (en) | 2006-09-28 |
WO2006101603A1 (en) | 2006-09-28 |
BRPI0609426B1 (pt) | 2020-09-24 |
MY147638A (en) | 2012-12-31 |
EA014554B1 (ru) | 2010-12-30 |
JP2008538110A (ja) | 2008-10-09 |
EA200702039A1 (ru) | 2008-02-28 |
DK1861401T3 (en) | 2015-12-07 |
IL186041A0 (en) | 2008-02-09 |
KR101323665B1 (ko) | 2013-10-31 |
NO340833B1 (no) | 2017-06-26 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM1K | Lapsed by not paying the annual fees |