NO20064251L - Benzamidazolderivater og anvendelse derav - Google Patents

Benzamidazolderivater og anvendelse derav

Info

Publication number
NO20064251L
NO20064251L NO20064251A NO20064251A NO20064251L NO 20064251 L NO20064251 L NO 20064251L NO 20064251 A NO20064251 A NO 20064251A NO 20064251 A NO20064251 A NO 20064251A NO 20064251 L NO20064251 L NO 20064251L
Authority
NO
Norway
Prior art keywords
formula
present
benzamidazole
derivatives
compound
Prior art date
Application number
NO20064251A
Other languages
English (en)
Other versions
NO332344B1 (no
Inventor
N N
Original Assignee
Takeda Pharmaceutical
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34858222&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20064251(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of NO20064251L publication Critical patent/NO20064251L/no
Publication of NO332344B1 publication Critical patent/NO332344B1/no

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245—Oxadiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Abstract

Den foreliggende oppfinnelse vedrører en forbindelse som er representert ved formelen (T). hvori Rer en gruppe som er representert ved formelen, hvori R, R, R, R,, Rog Rhver for seg uavhengig er et hydrogenatom eller et Ci .6 alkyl, eller et salt derav. Forbindelsen ifølge den foreliggende oppfinnelse er egnet som et agens for profylakse eller behandling av sirkulatoriske sykdommer slik som hypertensjon og lignende og metaboliske sykdommer slik som diabetes og lignende.
NO20064251A 2004-02-25 2006-09-20 Benzimidazolderivat, fremgangsmate for fremstilling derav, medikament inneholdende denne forbindelsen samt anvendelse av forbindelsen. NO332344B1 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2004048928 2004-02-25
US11/031,057 US7157584B2 (en) 2004-02-25 2005-01-07 Benzimidazole derivative and use thereof
PCT/JP2005/003422 WO2005080384A2 (en) 2004-02-25 2005-02-23 Benzimidazole derivative and use as aii receptor antagonist

Publications (2)

Publication Number Publication Date
NO20064251L true NO20064251L (no) 2006-11-22
NO332344B1 NO332344B1 (no) 2012-09-03

Family

ID=34858222

Family Applications (2)

Application Number Title Priority Date Filing Date
NO20064251A NO332344B1 (no) 2004-02-25 2006-09-20 Benzimidazolderivat, fremgangsmate for fremstilling derav, medikament inneholdende denne forbindelsen samt anvendelse av forbindelsen.
NO2012017C NO2012017I1 (no) 2004-02-25 2012-11-09 Benzimidazolderivat, fremgangsmåte for fremstilling derav, medikament inneholdende denne forbindelsen samt anvendelse av forbindelsen.

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO2012017C NO2012017I1 (no) 2004-02-25 2012-11-09 Benzimidazolderivat, fremgangsmåte for fremstilling derav, medikament inneholdende denne forbindelsen samt anvendelse av forbindelsen.

Country Status (33)

Country Link
US (3) US7157584B2 (no)
EP (3) EP1857457B1 (no)
JP (2) JP4256852B2 (no)
KR (1) KR101080029B1 (no)
CN (2) CN101381366B (no)
AR (2) AR047972A1 (no)
AT (2) ATE440095T1 (no)
AU (1) AU2005214271B8 (no)
BR (2) BR122012009489B8 (no)
CA (1) CA2557538C (no)
CY (5) CY1107008T1 (no)
DE (3) DE602005002030T2 (no)
DK (3) DK1718641T3 (no)
ES (3) ES2388945T3 (no)
HK (2) HK1098472A1 (no)
HR (3) HRP20070510T3 (no)
HU (1) HUS1200008I1 (no)
IL (1) IL177533A (no)
LU (1) LU91962I2 (no)
MA (1) MA28478B1 (no)
ME (2) ME01643B (no)
MY (1) MY142807A (no)
NL (1) NL300802I2 (no)
NO (2) NO332344B1 (no)
NZ (1) NZ549755A (no)
PL (3) PL1718641T3 (no)
PT (3) PT2119715E (no)
RS (3) RS52376B (no)
RU (2) RU2369608C2 (no)
SI (3) SI1718641T1 (no)
TW (1) TWI336702B (no)
WO (1) WO2005080384A2 (no)
ZA (1) ZA200607241B (no)

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KR20240039252A (ko) 2022-09-19 2024-03-26 대봉엘에스 주식회사 안지오텐신 ⅱ 길항제로서의 아질사르탄 디시클로헥실아민 및 이를 유효성분으로 하는 심혈관질환 치료 또는 예방용 약학적 조성물

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