NO20061092L - Heteroarvlaminosulfonvlfenvl-derivater for anvendelse som natrium- eller kalslumkanalblokkere i behandlingen av smerte - Google Patents
Heteroarvlaminosulfonvlfenvl-derivater for anvendelse som natrium- eller kalslumkanalblokkere i behandlingen av smerteInfo
- Publication number
- NO20061092L NO20061092L NO20061092A NO20061092A NO20061092L NO 20061092 L NO20061092 L NO 20061092L NO 20061092 A NO20061092 A NO 20061092A NO 20061092 A NO20061092 A NO 20061092A NO 20061092 L NO20061092 L NO 20061092L
- Authority
- NO
- Norway
- Prior art keywords
- treatment
- heteroarvlaminosulfonylphenyl
- pain
- derivatives
- sodium
- Prior art date
Links
- 229940127291 Calcium channel antagonist Drugs 0.000 title 1
- DGAQECJNVWCQMB-PUAWFVPOSA-M Ilexoside XXIX Chemical compound C[C@@H]1CC[C@@]2(CC[C@@]3(C(=CC[C@H]4[C@]3(CC[C@@H]5[C@@]4(CC[C@@H](C5(C)C)OS(=O)(=O)[O-])C)C)[C@@H]2[C@]1(C)O)C)C(=O)O[C@H]6[C@@H]([C@H]([C@@H]([C@H](O6)CO)O)O)O.[Na+] DGAQECJNVWCQMB-PUAWFVPOSA-M 0.000 title 1
- 239000000480 calcium channel blocker Substances 0.000 title 1
- 229910052708 sodium Inorganic materials 0.000 title 1
- 239000003195 sodium channel blocking agent Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 108010052164 Sodium Channels Proteins 0.000 abstract 1
- 102000018674 Sodium Channels Human genes 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
Classifications
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- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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- C04B35/63—Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B using additives specially adapted for forming the products, e.g.. binder binders
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- C07C311/30—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
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Abstract
Det beskrives forbindelser som er nyttige som inhibitorer av spenningsportstyrte natriumkanaler. Det beskrives også farmasøytisk akseptable sammensetninger som omfatter forbindelsene, og fremgangsmåter for anvendelse av sammensetningene ved behandling av forskjellige forstyrrelser.
Applications Claiming Priority (3)
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US49365903P | 2003-08-08 | 2003-08-08 | |
US58471704P | 2004-07-01 | 2004-07-01 | |
PCT/US2004/025827 WO2005013914A2 (en) | 2003-08-08 | 2004-08-09 | Heteroarylaminosulfonylphenyl derivatives for use as sodium or calcium channel blockers in the treatment of pain |
Publications (1)
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NO20061092L true NO20061092L (no) | 2006-04-27 |
Family
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NO20061092A NO20061092L (no) | 2003-08-08 | 2006-03-07 | Heteroarvlaminosulfonvlfenvl-derivater for anvendelse som natrium- eller kalslumkanalblokkere i behandlingen av smerte |
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US (3) | US8202861B2 (no) |
EP (3) | EP1673357A2 (no) |
JP (2) | JP2007501804A (no) |
KR (1) | KR20060073930A (no) |
AR (1) | AR045238A1 (no) |
AU (1) | AU2004263179B8 (no) |
CA (1) | CA2539227A1 (no) |
IL (1) | IL173602A0 (no) |
NO (1) | NO20061092L (no) |
NZ (2) | NZ545710A (no) |
PE (1) | PE20050358A1 (no) |
TW (1) | TW200524888A (no) |
WO (1) | WO2005013914A2 (no) |
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US20130184258A1 (en) | 2013-07-18 |
AR045238A1 (es) | 2005-10-19 |
EP2332912A1 (en) | 2011-06-15 |
US8309543B2 (en) | 2012-11-13 |
TW200524888A (en) | 2005-08-01 |
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